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BindingDB Data by Target and Substrate


Target NameSubstrate NameEnz. Inhib.
Data
11-beta-Hydroxysteroid Dehydrogenase 1 (11-beta-HSD1) cortisone 73
[3H]-cortisone 159
[3H]cortisone 26
11-beta-Hydroxysteroid Dehydrogenase 2 (11-beta-HSD2) cortisol 42
[3H]cortisol 11
15-Lipoxygenase Linoleic Acid 115
17-beta-Hydroxysteroid Dehydrogenase 1 (17-beta-HSD1) 17beta-estradiol (E2) 3
Estrone (E1) 3
[2,4,6,7-3H]-E1 39
17-beta-Hydroxysteroid Dehydrogenase 2 (17-beta-HSD2) [2,4,6,7-3H]-E2 16
17-beta-Hydroxysteroid Dehydrogenase 5 (17-beta-HSD5, AKR1C3) 3alpha-Androstanediol 2
Androstenedione 3
Androsterone 2
S-(+)-1,2,3,4-tetrahydro-1-naphthol 1
testosterone 1
20-alpha-Hydroxysteroid Dehydrogenase (AKR1C1) 5Beta-pregnane-3alpha,20alpha-diol 1
20-alpha-Hydroxysteroid Dehydrogenase (AKR1C1) Mutant (H222S) 5Beta-pregnane-3alpha,20alpha-diol 1
20-alpha-Hydroxysteroid Dehydrogenase (AKR1C1) Mutant (L306A) 5Beta-pregnane-3alpha,20alpha-diol 1
20-alpha-Hydroxysteroid Dehydrogenase (AKR1C1) Mutant (L308A) 5Beta-pregnane-3alpha,20alpha-diol 1
20-alpha-Hydroxysteroid Dehydrogenase (AKR1C1) Mutant (L54V) 5Beta-pregnane-3alpha,20alpha-diol 1
2C-methyl-D-erythritol-2,4-cyclodiphosphate synthase (IspF) 4-diphosphocytidyl-2C-methyl-D-erythritol-2-phosphate 9
3-alpha-Hydroxysteroid Dehydrogenase Type 1 (AKR1C4) S-(+)-1,2,3,4-tetrahydro-1-naphthol 1
3-alpha-Hydroxysteroid Dehydrogenase Type 3 (AKR1C2) S-(+)-1,2,3,4-tetrahydro-1-naphthol 1
3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) AKT2 75
PDK1 Peptide Substrate 1
PDKtide 11
SGK1 50
3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (A162V) PDKtide 2
3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (E166D) PDKtide 2
3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (L159M) PDKtide 2
3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (T222A) PDKtide 2
3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (V143T) PDKtide 2
3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (V143T/T222A) PDKtide 2
5-Lipoxygenase Arachidonic acid 74
Linoleic Acid 28
Abhydrolase Domain-Containing Protein 6 FP-rhodamine 1
ABL Biotinylated peptide substrate 14
biotinylated SB202190 7
[Val5]-Angiotensin II 30
ABL Mutant (E255K) biotinylated SB202190 7
ABL Mutant (F359V) biotinylated SB202190 7
ABL Mutant (H396P) biotinylated SB202190 7
ABL Mutant (M351T) biotinylated SB202190 7
ABL Mutant (Q252H) biotinylated SB202190 7
ABL Mutant (T315I) biotinylated affinity ligand 20
biotinylated SB202190 7
ABL Mutant (T315N) biotinylated SB202190 7
ABL Mutant (Y253F) biotinylated SB202190 7
Acetylcholinesterase (AChE) acetylcholine 93
acetylcholine chloride 15
acetylthiocholine chloride 15
acetylthiocholine iodide 873
Activated Protein C (APC) Chromogenic Substrate S-2366 1
Acyl Cholesterol Acyltransferase 1 (ACAT-1) [14C] oleoyl coenzyme A 7
ADAMTS-4 (Aggrecanase-1) Fluorescent peptide WAAG-3R 30
ADAMTS-5 (Aggrecanase-2) QF-peptide 30
WAAG-3R 35
Adenosine A3 Receptor [3H]AB-MECA 29
Adenosine Deaminase Adenosine 59
Adenosine Kinase (AK) Adenosine 8
Adenosine Phosphosulfate Reductase (APSR) Adenosine Phosphosulfate (APS) 10
Adenosine Receptor A1 Not Available 71
[3H]DPCPX 103
Adenosine Receptor A2A [3H]-CGS 21680 71
[3H]-ZM241385 86
[3H]NECA 29
Adenosine Receptor A2B Not Available 7
Adenosine Receptor A3 Not Available 7
AICAR Tfase AICAR 19
Aldehyde Reductase (ALR1) D,L-glyceraldehyde 40
Aldose Reductase (ALR2) benzyl alcohol 15
D,L-glyceraldehyde 50
D-glyceraldehyde 77
D-xylose 4
xylitol 10
Aldose Reductase (ALR2) Mutant (C298A) benzyl alcohol 2
Aldose Reductase (ALR2) Mutant (C298A/W219Y) xylitol 12
Aldosterone Synthase (CYP11B2) deoxycorticosterone 94
[4-14C]-11-deoxycorticosterone 16
Alpha-1 Adrenergic Receptor [3H]-Prazosin 12
alpha-Amylase Potato starch 20
alpha-Carbonic Anhydrase Carbon Dioxide 17
alpha-Chymotrypsin Not Available 1
alpha-Glucosidase (alpha-Glu) 4-methylumbelliferyl alpha-glucoside 14
pNPG 21
alpha-Methylacyl-CoA Racemase (25S)-THC-CoA 10
Alpha2 Adrenoreceptor Clonidine 4
Aminopeptidase M L-alanyl-p-nitroanilide 27
L-Leucine-para-nitroanilide 19
Androgen Receptor (AR) DHT 167
Not Available 27
SRC2-3 peptide 11
Testosterone 11
[3H]DHT 49
[3H]MIB 70
Angiotensin-Converting Enzyme Abz-Gly-p-nitro-Phe-Pro-OH 6
Mca-Ala-Ser-Asp-Lys-Dpa-OH 4
N-Cbz-Phe-His-Leu 29
Angiotensin-Converting Enzyme 2 Mca-APK(Dnp)OH 36
Anthrax Lethal Factor (LF) fluorogenic LF protease substrate III 21
Fluorogenic LF Substrate 28
MAPKKide 147
Peptide Substrate 50
Apoptosis Regulator Bcl-2 FITC-conjugated-Bim BH3 Peptide 10
Fluorescein-labeled BAX peptide 52
Apoptosis Regulator Bcl-xL Bak-BH3 peptide 19
F-BakBH3 10
F-Bim 78
Fl-Bak peptide 50
Fluorescein-labeled BAD peptide 52
Apurinic-Apyrimidinic Endonuclease 1 (APE1) DNA Substrate 47
Aromatase (CYP19) Androstenedione 279
dibenzylfluorescein (DBF) 21
Testosterone 60
[1beta-3H] androstenedione 53
Aryl Hydrocarbon Receptor (AhR) [3H]-TCDD 25
Asparaginyl Endopeptidase (AE) Cbz-Ala-Ala-Asn-AMC 89
ATP Phosphoribosyltransferase Phosphoribosyl Pyrophosphate (PRPP) 11
ATP-Binding Cassette Transporter ABCG2 PhA 21
Aurora Kinase A (Aurora-A) Aurora Peptide Substrate 23
biotinylated affinity ligand 11
Biotinylated Cross-tide Substrate 13
Biotinylated Peptide Substrate 47
CHOCKtide 131
FAM-PKAtide 26
Histone H3 84
Kemptide 1
Not Specified 1
PKAtide 2
Substrate Peptide SerThr 01 1
Aurora Kinase B (Aurora-B) Aurora B Substrate Peptide 1
biotinylated affinity ligand 13
Biotinylated Cross-tide Substrate 13
Biotinylated Peptide Substrate 37
CHOCKtide 6
FAM-PKAtide 13
Histone H3 16
Not Specified 1
Aurora Kinase C (Aurora-C) biotinylated affinity ligand 18
Not Specified 1
AXL Receptor Tyrosine Kinase biotinylated affinity ligand 16
B-Raf Protein Kinase biotin-MEK 1
GST-MEK 38
GST-MEK1 16
MEK-1 1
Rhodamine green labeled ligand 17
B-Raf Protein Kinase Mutant (V599E) MEK-1 1
B-Raf Protein Kinase Mutant (V600E) biotin-MEK 13
GST-MEK1 101
MEK Inactive Mutant 32
Bacterial Leucyl Aminopeptidase L-Leucine-para-nitroanilide 19
Bacteriophage T4 DNA Ligase 32P-labeled nicked duplex DNA substrate 7
Beta-1 Adrenergic Receptor [3H]CGP 12177 25
Beta-2 Adrenergic Receptor [125I]-(-)iodopindolol 7
[3H]CGP 12177 32
Beta-3 Adrenergic Receptor [3H]CGP 12177 25
beta-Carbonic Anhydrase Carbon Dioxide 37
beta-Hydroxyacyl-Acyl Carrier Protein Dehydratase (FabZ) crotonoyl-CoA 53
beta-Ketoacyl-ACP Synthase III (FabH) Malonyl-ACP 58
beta-Secretase (BACE-1) APP_NFEV 23
BACE Peptide Substrate 62
BACE Substrate Peptide 85
BACE-1 Peptide Substrate 16
BACE-1 Substrate Peptide 47
ELGY-9 7
Fluorescent Substrate 110
fluorescent substrate FS-2 7
Fluorogenic Substrate 37
FS1 FRET Substrate 4
MBPAPPC125 30
beta-Secretase (BACE-2) BACE Peptide Substrate 5
BACE Substrate Peptide 7
Fluorescent Substrate 100
Fluorogenic Substrate 12
Bfl-1 F-Bim 198
FITC-conjugated-Bim BH3 Peptide 8
Bfl-1 FITC-Ahx-EDIIRNIARHLAQVGDSMDR 44
Biotin Carboxylase Biotinyl-BCCP 14
Bone Morphogenetic Protein Receptor type II (BMPR2) biotinylated affinity ligand 6
Botulinum Neurotoxin Type A SNAP-25 substrate peptide 18
SNAP-25-based peptide substrate 16
SNAPtide 99
Butyrylcholinesterase (BuChE) butyrylthiocholine 603
butyrylthiocholine chloride 28
C-Raf Protein Kinase MEK Inactive Mutant 34
Calcium-Sensing Receptor (CaSR) Not Available 44
Calpain-1 BODIPY FL casein 10
Suc-Leu-Tyr-AMC 11
Calpain-2 BODIPY FL casein 10
CaM Kinase II Autocamtide-2 38
CaM Kinase II Peptide Substrate 4
cAMP-Dependent Protein Kinase (PKA) biotinylated kemptide 30
Fluorescent probe ARC-583 27
histone (type H IIas) 15
histone (type Vs) 61
Histone H1 10
Histone type HL 67
Histone VII-S 13
ING Peptide 16
Kemptide 81
Lys-rich histone 97
Peptide Substrate 11
PKA Peptide Substrate 5
PKA-specific peptide substrate 21
stathmin 1
cAMP-Dependent Protein Kinase (PKA) Mutant PKAR1 (1) Kemptide 5
cAMP-Dependent Protein Kinase (PKA) Mutant PKAR1 (2) Kemptide 5
cAMP-Dependent Protein Kinase (PKA) Mutant PKAR1 (3) Kemptide 5
cAMP-Dependent Protein Kinase (PKA) Mutant PKAR1 (4) Kemptide 5
cAMP-Dependent Protein Kinase (PKA) Mutant PKAR2 (1) Kemptide 5
cAMP-Dependent Protein Kinase (PKA) Mutant PKAR2 (2) Kemptide 1
cAMP-Dependent Protein Kinase (PKA) Mutant PKAR2 (3) Kemptide 3
cAMP-Dependent Protein Kinase (PKA) Mutant PKAR3 Kemptide 5
cAMP-Dependent Protein Kinase (PKA) Mutant PKAR3 (1) Kemptide 5
cAMP-Dependent Protein Kinase (PKA) Mutant PKAR4 Kemptide 5
cAMP-Dependent Protein Kinase (PKA) Mutant PKAR5 Kemptide 5
Cannabinoid Receptor 1 GTP-gamma-S 19
[3H]CP55940 109
[3H]SR141716A 44
Cannabinoid Receptor 2 [3H]CP55940 122
[3H]SR141716A 10
Carbonic Anhydrase (hpCA) Carbon Dioxide 47
Carbonic Anhydrase (mtCA 1) Carbon Dioxide 37
Carbonic Anhydrase (mtCA 3) Carbon Dioxide 37
Carbonic Anhydrase 2 (Can2) Carbon Dioxide 37
Carbonic Anhydrase I 4-nitrophenyl acetate 139
Carbon Dioxide 315
dansylamide 5
Carbonic Anhydrase II 4-nitrophenyl acetate 173
Carbon Dioxide 401
dansylamide 52
Carbonic Anhydrase II Mutant (F131V) dansylamide 11
Carbonic Anhydrase III Carbon Dioxide 49
Carbonic Anhydrase IV 4-nitrophenyl acetate 133
Carbon Dioxide 134
Carbonic Anhydrase IX Carbon Dioxide 265
Carbonic Anhydrase VA Carbon Dioxide 149
Carbonic Anhydrase VB Carbon Dioxide 103
Carbonic Anhydrase VI Carbon Dioxide 85
Carbonic Anhydrase VII Carbon Dioxide 52
Carbonic Anhydrase XII Carbon Dioxide 69
Carbonic Anhydrase XIII Carbon Dioxide 51
Carbonic Anhydrase XIV Carbon Dioxide 53
Carbonic Anhydrase XV Carbon Dioxide 73
Carboxylesterase 1 Nitrophenyl Acetate 271
Carboxylesterase 2 (intestine, liver) Nitrophenyl Acetate 146
Carboxypeptidase A (CPA) Furylacryloyl-Phe-Phe 15
Casein Kinase I Casein 8
CK1 Peptide Substrate 4
CK1 Substrate Peptide 1
Casein Kinase II CK-2 Peptide Substrate 15
CK2 Peptide Substrate 1
Peptide Substrate 25
stathmin 1
Caspase-1 Caspase-1 Fluorogenic Substrate 115
Caspase-1 Fluorogenic Substrate Ac-Trp-Glu-His-Asp-AFC 9
Caspase-1 Substrate 20
Fluorometric Tetrapeptide Ac-DEVD-AMC 1
Caspase-2 Caspase Substrate 7
Caspase-2 Fluorogenic Substrate 8
Caspase-2 Fluorogenic Substrate Ac-Val-Asp-Val-Ala-Asp-AFC 9
Caspase-3 Ac-DEVD-AFC 42
Caspase Fluorogenic Substrate 188
Caspase-3 (7) Fluorogenic Substrate 11
Caspase-3 Fluorogenic Substrate 35
Caspase-3 Fluorogenic Substrate Ac-Asp-Glu-Val-Asp-AFC 49
Caspase-3 Substrate 73
Fluorometric Tetrapeptide Ac-DEVD-AMC 1
Caspase-4 Caspase-4 Fluorogenic Substrate 8
Caspase-4 Fluorometric Substrate Ac-Trp-Glu-His-Asp-AFC 9
Caspase-5 Caspase-5 Fluorometric Substrate Ac-Trp-Glu-His-Asp-AFC 9
Caspase-6 Caspase Fluorogenic Substrate 8
Caspase Substrate 7
Caspase-6 Fluorogenic Substrate 29
Caspase-6 Fluorometric Substrate Ac-Val-Glu-Ile-Asp-AFC 9
Caspase-6 Substrate 22
Caspase-7 Caspase Fluorogenic Substrate 85
Caspase Substrate 7
Caspase-3 (7) Fluorogenic Substrate 11
Caspase-7 Fluorometric Substrate Ac-Asp-Glu-Val-Asp-AFC 9
Caspase-7 Substrate 20
Caspase-8 Caspase Substrate 7
Caspase-8 Fluorogenic Substrate 96
Caspase-8 Fluorometric Substrate Ac-Ile-Glu-Thr-Asp-AFC 9
Caspase-8 Substrate 20
Caspase-9 Caspase-9 Fluorogenic Substrate 8
Cathepsin B Boc-Leu-Lys-Arg-AMC 100
Cbz-Phe-Arg-AMC 36
Z-Arg-Arg-AMC 24
Z-Phe-Arg-NMec 13
Cathepsin B Z-Arg-Arg-AMC 56
Cathepsin B-Like Cysteine Protease (TbcatB) Z-Phe-Arg-AMC 56
Cathepsin D Cathepsin D FRET Substrate 1
Cathepsin D Peptide Substrate 57
Cathepsin D/Pepsin Peptide Substrate 5
Fluorescent Substrate 100
MOCAc-Gly-Lys-Pro-Ile-Leu-Phe-Phe-Arg-Leu-Lys(Dnp)-D-Arg-NH2 27
Peptide Substrate 104
Cathepsin K Ac-Lys-His-Pro-Lys-ACMC 170
Cbz-Leu-Arg-AMC 173
Cbz-Phe-Arg-AMC 114
Z-Leu-Arg-NHMec 48
Z-Phe-Arg-AMC 24
Cathepsin L Ac-His-Lys-Phe-Lys-ACMC 170
Cbz-Leu-Arg-AMC 100
Cbz-Phe-Arg-AMC 87
Cbz-Phe-Arg-MCA 13
Z-Phe-Arg-AMC 24
Z-Phe-Arg-NHMec 52
Cathepsin L2 Z-Phe-Arg-AMC 24
Cathepsin S Ac-His-Pro-Val-Lys-ACMC 180
Cathepsin S Substrate Peptide 28
Cbz-Leu-Arg-AMC 8
Cbz-Phe-Arg-AMC 9
Z-Leu-Leu-Arg-AMC 43
Z-Phe-Arg-AMC 24
Z-Val-Val-Arg-AMC 130
Z-Val-Val-Arg-NHMec 48
Cathepsin V Cbz-Phe-Arg-AMC 2
Cdc7 Kinase His6-tagged MCM2 16
MCM2 85
Cell Division Cycle 2-Like 1(CDC2L1) biotinylated affinity ligand 7
Cell Division Cycle 2-Like 2 (CDC2L2) biotinylated affinity ligand 7
Cell Division Cycle 2-Like 6 (CDK11) biotinylated affinity ligand 11
cGMP-Dependent Protein Kinase Histone H1 10
Histone II-A 13
Checkpoint Kinase (Chk1) biotinylated CDC25C peptide 13
biotinylated cdc25c peptide substrate 2
biotinylated CHKtide 9
Biotinylated Peptide Substrate 24
Cdc25C peptide substrate 124
Chktide 31
Not Available 1
Synthetic Chk1 Peptide Substrate 3
Checkpoint Kinase (Chk2) biotinylated CDC25C peptide 4
Fam-CHK2tide 7
Histone H1 4
Chitinase fluorogenic substrate 12
Not Available 3
Chitinase Mutant (A217G) Not Available 3
Chitinase Mutant (D175A) Not Available 3
Chitinase Mutant (D246A) Not Available 1
Chitinase Mutant (E177A) Not Available 1
Chitinase Mutant (E322A) Not Available 3
Chitinase Mutant (M243A) Not Available 3
Chitinase Mutant (R301K) Not Available 3
Chitinase Mutant (T138A) Not Available 3
Chitinase Mutant (Y245F) Not Available 2
Cholecystokinin-1 Receptor [125I]CCK-8 17
Cholecystokinin-2 Receptor [125I]CCK-8 17
Chymase Chymase/Chymotrypsin Chromogenic Substrate 2
Chymotrypsin Chymase/Chymotrypsin Chromogenic Substrate 2
Suc-Ala-Ala-Pro-Phe-7-amino-4-methylcoumarin 27
cIAP-1 BIR3 AVP-diPhe-FAM 5
Smac-derived peptide 5
cIAP-2 BIR3 AVP-diPhe-FAM 5
Smac-derived peptide 5
cIAP1-BIR3 AVP-diPhe-FAM 5
cIAP2-BIR3 AVP-diPhe-FAM 3
CLK1 biotinylated affinity ligand 16
CLK4 biotinylated affinity ligand 13
Collagenase (ChC) Collagenase Substrate 187
Corticotropin-releasing Factor Receptor 1 125I-Tyr(0)-ovine-CRF 135
Cyclin-Dependent Kinase 1 (CDK1) biotinylated CDK peptide substrate 3
Biotinylated CDK1 Peptide Substrate 99
Biotinylated peptide substrate 4
GST-Rb fusion protein 85
Histidine-tagged retinoblastoma protein 26
Histone H1 652
Not Available 1
Peptide Substrate 102
Rb (Ser780) Biotinylated Peptide 4
S1 peptide 5
Substrate Peptide SerThr 18 3
Cyclin-Dependent Kinase 2 (CDK2) biotinylated CDK peptide substrate 3
Biotinylated peptide substrate 91
CDK2 biotinylated peptide substrate 4
CDK2 Peptide Subsrate 22
CDKtide 3
GST-Rb fusion protein 675
Histidine-tagged Rb 68
Histidine-tagged retinoblastoma protein 26
Histone H1 548
Histone type 3 20
ING Peptide 144
Not Available 1
Peptide Substrate 132
Rb(21) 8
S1 peptide 13
Cyclin-Dependent Kinase 2 (CDK2) Mutant (F82H) Histone H1 1
Cyclin-Dependent Kinase 2 (CDK2) Mutant (F82H/L83V/H84D) Histone H1 2
Cyclin-Dependent Kinase 2 (CDK2) Mutant (F82H/L83V/H84D/K89T) Histone H1 2
Cyclin-Dependent Kinase 2 (CDK2) Mutant (K89T) Histone H1 2
Cyclin-Dependent Kinase 2 (CDK2) Mutant (L83V/H84D) Histone H1 1
Cyclin-Dependent Kinase 4 (CDK4) Biotinylated Peptide Substrate 30
G1 peptide 43
GST-Rb fusion protein 665
Histidine-tagged retinoblastoma protein 26
Histone H1 9
ING Peptide 160
Rb 2
Rb(21) 95
Retinoblastoma (Rb) 13
Cyclin-Dependent Kinase 5 (CDK5) Cdk5 Substrate 1
Histone H1 301
Histone H1 Peptide 1
Cyclin-Dependent Kinase 6 (CDK6) G1 peptide 1
Histone H1 7
Cyclin-Dependent Kinase 7 (CDK7) biotinylated affinity ligand 12
Biotinylated Peptide Substrate 7
FAM-CDK7 derived peptide 18
Histone H1 4
Cyclin-Dependent Kinase 8 (CDK8) biotinylated affinity ligand 8
Cyclin-Dependent Kinase 9 (CDK9) biotinylated affinity ligand 6
Biotinylated Peptide Substrate 7
pRB 4
RNA Polymerase CTD Peptide 2
Cyclooxygenase-1 Arachidonic acid 33
[1-14C]Arachidonic acid 39
Cyclooxygenase-2 Arachidonic acid 30
[1-14C]Arachidonic acid 45
Cytochrome P450 1A2 Ethoxyresorufin 1
Cytochrome P450 2A6 Coumarin 31
Cytochrome P450 2C19 3-butyryl-7- methoxycoumarin 7
S-Mephenytoin 1
Cytochrome P450 2C9 7-methoxy-4-trifluoromethylcoumarin-3-acetic acid 7
Diclofenac 1
MFC 21
Cytochrome P450 2D6 4-Methylaminomethyl-7-methoxycoumarin 7
Bufuralol 1
Cytochrome P450 2E1 p-nitrophenol 9
Cytochrome P450 3A1 erythromycin 11
Cytochrome P450 3A4 7-Benzyloxyquinoline 7
BFC 31
Midazolam 1
Testosterone 52
Cytochrome P450 51(CYP51) Not Available 26
Cytochrome P450 51(CYP51) Mutant (F78L) Not Available 2
D-Amino Acid Oxidase (DAAO) D-Serine 61
Not Available 7
D-Aspartate Oxidase (DDO) D-Aspartic Acid 23
Delta Opioid Receptor [3H]-diprenorphine 69
[3H]-naltrindole 21
[3H]DPDPE 53
Dengue Virus 1 (DENV1) NS2B-NS3 Protease Bz-Nle-Lys-Arg-Arg-AMC 10
Dengue Virus 2 (DENV2) NS2B-NS3 Protease Boc-Gly-Arg-Arg-AMC 5
Bz-Nle-Lys-Arg-Arg-AMC 10
Dengue Virus 3 (DENV3) NS2B-NS3 Protease Bz-Nle-Lys-Arg-Arg-AMC 10
Dengue Virus 4 (DENV4) NS2B-NS3 Protease Bz-Nle-Lys-Arg-Arg-AMC 10
Diacyl Glycerolacyltransferase 1 (DGAT-1) didecanoyl glycerol 25
[14C] oleoyl coenzyme A 9
Diacyl Glycerolacyltransferase 2 (DGAT-2) [14C] oleoyl coenzyme A 2
Dihydrofolate Reductase (DHFR) dihydrofolic acid 612
Dihydrofolate Reductase (DHFR) Mutant (F98Y) dihydrofolic acid 2
Dihydrofolate Reductase (DHFR) Mutant (I100L) dihydrofolic acid 2
Dihydrofolate Reductase-Thymidylate Synthase (DHFR-TS) dihydrofolic acid 22
Dihydrofolate Reductase-Thymidylate Synthase (DHFR-TS) Mutant KICB1 dihydrofolic acid 3
Dihydrofolate Reductase-Thymidylate Synthase (DHFR-TS) Mutant SP21 dihydrofolic acid 19
Dihydrofolate Reductase-Thymidylate Synthase (DHFR-TS) Mutant V1/S dihydrofolic acid 3
Dihydroorotate Dehydrogenase (DHODH) Coenzyme Q1 9
Coenzyme Q6 18
Decylubiquinone 181
Ubiquinone-0 (CoQ0) 40
Dihydroorotate Dehydrogenase (DHODH) Mutant (H185A) Ubiquinone-0 (CoQ0) 13
Dihydroorotate Dehydrogenase (DHODH) Mutant (R265A) Ubiquinone-0 (CoQ0) 13
Dipeptidyl Peptidase II (DPP-II) (QPP) Nle-Pro-AMC 52
Dipeptidyl Peptidase IV (DPP-IV) Ala-Pro-7-amido-4-trifluoromethylcoumarin 48
Gly-Pro-AMC 501
Gly-Pro-pNA 149
H-Ala-Pro-pNA 49
Dipeptidyl Peptidase VII (DPP-VII) (QPP) Gly-Pro-pNA 47
Lys-Ala-pNA 67
Nle-Pro-AMC 215
DNA Gyrase ATP 44
Kinetoplast DNA 5
DNA Ligase (MtuLigA) 32P-labeled nicked duplex DNA substrate 7
DNA Ligase I 32P-labeled nicked duplex DNA substrate 4
DNA Polymerase alpha dGTP 2
DNA template-primer 10
DNA Polymerase beta DNA template-primer 10
DNA Polymerase gamma dGTP 2
DNA polymerase IIIC dGTP 2
DNA polymerase IIIE dGTP 4
DNA Topoisomerase IV ATP 22
Kinetoplast DNA 5
Dopamine Receptor D2 [3H]-Spiroperidol 39
Dopamine Transporter (DAT) [125I]RTI-55 64
[3H]WIN 35,428 19
DPP8 Ala-Pro-7-amido-4-trifluoromethylcoumarin 297
Gly-Pro-AMC 38
Gly-Pro-pNA 65
DPP9 Gly-Pro-AMC 275
Dual Specificity Protein Phosphatase 1 OMFP Substrate 165
DYRK1A myelin basic protein 3
EGF-R Tyrosine Kinase (Biotin)Poly(Glu:Tyr) 4
Angiotensin II 30
Biotinylated EGFR Peptide Substrate 19
biotinylated gastrin substrate 1
Biotinylated Peptide Substrate 41
EGF Receptor Substrate 23
EGF-R Substrate 325
EGFR Substrate 174
EGFR Substrate Peptide 22
N-biotinyl peptide substrate 1
Not Available 19
poly(E, A, Y) 93
poly(E,A,Y) 30
poly(E,Y) 13
Poly(E:A:Y) 3
Poly(E:Y) 131
Poly(GAT) 170
poly(Glu4-Tyr) 13
poly(Glu4/Tyr) 24
Tyr 04 Substrate Peptide 4
EGF-R Tyrosine Kinase Mutant (G719C) biotinylated affinity ligand 20
EGF-R Tyrosine Kinase Mutant (G719S) Not Available 2
EGF-R Tyrosine Kinase Mutant (L858R) Not Available 4
EGF-R Tyrosine Kinase Mutant (L858R/T790M) Not Available 2
EGF-R Tyrosine Kinase Mutant (T790M) Not Available 2
Tyr 04 Substrate Peptide 4
Endothelin-Converting Enzyme 1 Pya(21)-(p-NO2)Phe(22)bigET(19-35) 29
Enoyl-ACP Reductase (FabI) Crotonoyl-ACP 50
Crotonoyl-CoA 111
Enoyl-ACP Reductase (FabK) Crotonoyl-ACP 5
Enoyl-ACP Reductase (InhA) 2-trans-Octenoyl-CoA (OCoA) 100
trans-2-Dodecenoyl-Coenzyme A 13
Enoyl-ACP Reductase (PfENR) Crotonoyl-CoA 28
Epoxide Hydrolase B (EHB) alpha-cyanocarbonate epoxide 20
Equilibrative Nucleoside Transporter 1 (ENT1) 5-(SAENTA)-X8-fluorescein 80
ErbB-2 (HER2) Tyrosine Kinase Biotinylated ErbB-2 Peptide Substrate 19
Biotinylated Peptide Substrate 41
ErbB-2 Substrate Peptide 22
HER-2 Substrate 38
poly(Glu4/Tyr) 24
ErbB-4 (HER4) Tyrosine Kinase Biotinylated ErbB-4 Peptide Substrate 9
ERK-2 biotin-MBP protein 1
EGFR Peptide Substrate 2
ERK-2 Peptide Substrate 4
ERKtide 57
Histone H1 3
Substrate Peptide T669 5
ERK-8 biotinylated affinity ligand 9
Estrogen Receptor (ER-alpha) 17beta-estradiol (E2) 134
Estrone (E1) 56
[3H]-estradiol 25
[3H]]estradiol 15
Estrogen Receptor (ER-beta) 17beta-estradiol (E2) 134
Estrone (E1) 56
Estrogen-Related Receptor, alpha PGC-1 alpha derived peptide 2
Estrogen-Related Receptor, gamma Biotinylated RIP140 peptide 12
[3H]4-OHT 19
Factor IXa (fIXa) Chromogenic Substrate 7
Factor IX Chromogenic Substrate 85
Factor VIIa (fVIIa) Chromogenic Substrate 7
Chromozym tPA 66
Factor VII Chromogenic Substrate 108
Not Specified 3
Pefachrome FVIIa 96
Spectrozyme-FVIIa 46
Factor Xa (fXa) Chromogenic Substrate Pefachrome FXa 63
Chromogenic Substrate S-2222 461
Chromogenic Substrate S-2765 472
Chromogenic Substrate Spectrozyme FXa 37
Chromozym X 39
Factor Xa (fXa) Chromogenic Substrate 57
Factor Xa Chromogenic Substrate 7
Factor Xa Fluorogenic Substrate 24
MeSO2-D-Nle-Gly-Arg-pNA 54
Not Specified 3
rhodamime 110, bis-(Boc-L-glycylglycyl-L-arginine amide) 25
Factor XIa (fXIa) Boc-Glu-Ala-Arg-AMC 396
Fluorogenic Tripeptide Substrate 31
Not Specified 3
Factor XIIa (fXIIa) Boc-Gln-Gly-Arg-AMC 87
Chromogenic Substrate S-2302 36
Falcipain-2 Z-Leu-Arg-AMC 30
Farnesoid X-Activated Receptor biotin-tagged SRC-1 4
Biotinylated SRC-1 Peptide 5
Not Available 54
Fatty Acid Amide Hydrolase 14C-labeled oleamide 115
FP-rhodamine 1
Oleamide 16
[14C]Anandamide 39
[3H]Anandamide 82
Fatty Acid Synthase 4-methylumbelliferyl heptanoate (4-MUH) 46
FGFR-1 Tyrosine Kinase Biotinylated FGFR Peptide Substrate 2
biotinylated gastrin substrate 1
N-biotinyl peptide substrate 1
Poly (E:Y) 1
poly(E,A,Y) 67
Poly(E:Y) 486
Substrate Peptide Tyr 04 1
FGFR-2 Tyrosine Kinase (Biotin)Poly(Glu:Tyr) 3
FGFR Substrate 7
Fibroblast Activation Protein (FAP) Gly-Pro-pNA 18
Formyl Peptide Receptor-Like 1 Not Available 18
G-protein Coupled Receptor 40 Not Available 52
G-protein Coupled Receptor 54 [125I]Kisspeptin-15 12
GABAA Receptor Mutant, alpha-1 (A160C), beta-2, gamma-2 [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1 (D97C), beta-2, gamma-2 [3H]Ro15-1788 1
GABAA Receptor Mutant, alpha-1 (F99C), beta-2, gamma-2 [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1 (G157C), beta-2, gamma-2 [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1 (G200C), beta-2, gamma-2 [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1 (S204C), beta-2, gamma-2 [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1 (S205C), beta-2, gamma-2 [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1 (T162C), beta-2, gamma-2 [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1 (T206C), beta-2, gamma-2 [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1 (V202C), beta-2, gamma-2 [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1 (V211C), beta-2, gamma-2 [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1 (Y209C), beta-2, gamma-2 [3H]Ro15-1788 1
GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (A79C) [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (Chimera) [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (D56C) [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (F77C) [3H]Ro15-1788 1
GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (L140C) [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (M130C) [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (R132C) [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (R144C) [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (R185C) [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (R194C) [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (T126C) [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (T142C) [3H]Ro15-1788 3
GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (T81C) [3H]Ro15-1788 3
GABAA Receptor, alpha-1, beta-2, gamma-2 [3H]Ro15-1788 3
GABAA Receptor, alpha-1, beta-3, gamma-2 [3H]flunitrazepam 8
GABAA Receptor, alpha-2, beta-2, gamma-2 [3H]Ro15-1788 3
GABAA Receptor, alpha-2, beta-3, gamma-2 [3H]flunitrazepam 8
GABAA Receptor, alpha-3, beta-2, gamma-2 [3H]Ro15-1788 3
GABAA Receptor, alpha-3, beta-3, gamma-2 [3H]flunitrazepam 7
GABAA Receptor, alpha-4, beta-2, gamma-2 [3H]Ro15-4513 3
GABAA Receptor, alpha-4, beta-3, gamma-2 [3H]flunitrazepam 4
GABAA Receptor, alpha-5, beta-2, gamma-2 [3H]Ro15-1788 3
GABAA Receptor, alpha-5, beta-3, gamma-2 [3H]flunitrazepam 8
GABAA Receptor, alpha-6, beta-2, gamma-2 [3H]Ro15-4513 3
GABAA Receptor, alpha-6, beta-3, gamma-2 [3H]flunitrazepam 7
Galectin-1 fluorescein-tagged saccharide 14
Galectin-3 fluorescein-tagged saccharide 23
Galectin-7 fluorescein-tagged saccharide 12
Galectin-8 fluorescein-tagged saccharide 11
Galectin-9 fluorescein-tagged saccharide 12
gamma-Aminobutyric Acid Type B Receptor [3H]GABA 16
Gamma-Secretase beta-Amyloid Precursor Protein (APP) 98
GAR Tfase GAR 18
Gastric Inhibitory Polypeptide Receptor (GIPR) 125I-GIP 30
Geranylgeranyl Diphosphate Synthase (GGPPS) [14C]IPP 61
Geranylgeranyl Transferase (GGTase-I) Biotinylated Peptide Substrate 29
Ha-Ras-CVLL 28
K-ras(B) decapeptide 43
PGGT I peptide substrate 1
Ras-CVLL 1
Ghrelin Receptor (Growth Hormone Secretagogue Receptor Type 1) 125I-His9-ghrelin 118
Not Available 13
Glucagon Receptor 125I-Glucagon 30
Glucocerebrosidase (Acid beta-Glucosidase) 4-methylumbelliferyl beta-D-glucoside 18
resorufin-beta-D-glucopyranoside 59
Glucocorticoid Receptor (GR) dexamethasone 84
dexamethasone (tetramethyl-rhodamine conjugated ) 49
Glucokinase D-glucose 34
Glutamate Carboxypeptidase II (GCPII) N-acetylaspartylglutamate (NAAG) 42
Glutaminyl Cyclase Gln-AMC 90
Glycogen Phosphorylase (PYGL) glycogen 102
Glycogen Phosphorylase (PYGM) glucose-1-phosphate 73
Glycogen Synthase Kinase-3, alpha Biotinylated Peptide Substrate 171
GSK-3 Peptide Substrate 2
Glycogen Synthase Kinase-3, beta Biotinylated Peptide Substrate 182
GS-1 peptide 344
GSK-3 beta Substrate Peptide 30
GSK-3 Peptide Substrate 29
GSK-3 Substrate Peptide 24
Phospho-GS2 Substrate Peptide 1
Phosphor-Glycogen Synthase Peptide-2 3
GRB2 Grb2 SH2 Binding Substrate 15
HCV NS3 Helicase DNA Substrate 12
HCV NS3-NS4A Serine Proteinase NS3-NS4A Chromogenic Peptide Substrate 291
NS4B-5A 30
HCV NS5B Polymerase biotinylated oligo (rG13)/poly rC 165
poly(A)/oligo(U)18 43
HCV NS5B Polymerase Mutant (M414T) poly(A)/oligo(U)18 2
HCV NS5B Polymerase Mutant (M423K) poly(A)/oligo(U)18 2
HCV NS5B Polymerase Mutant (P495A) poly(A)/oligo(U)18 2
HCV NS5B Polymerase Mutant (R501E) poly(A)/oligo(U)18 2
Heat Shock 70kDa Protein 1 Fluorescein-12-ATP 33
N6-(6-amino)hexyl-ATP-5-FAM 17
Not Available 8
Heat Shock Protein 90 (Hsp90) ATP 14
BODIPY-labeled Geldanamycin 9
cy3B-GM 268
Not Available 81
VER-00045864 25
VER-00051001 100
Heme Oxygenase 1 (HO-1) methemalbumin 44
Heme Oxygenase 2 (HO-2) methemalbumin 44
Hepsin Hepsin Chromogenic Substrate 6
hERG Potassium Channel 1 Not Available 10
[35S]-MK499 53
[3H]Astemizole 21
Histamine H1 Receptor [3H]Chlorpheniramine 18
[3H]mepyramine 5
[3H]pyrilamine 3
Histamine H2 Receptor tiotidine 1
[3H]tiotidine 5
Histamine H3 Receptor [3H]N-alpha-methyl histamine 104
Histamine H4 Receptor [3H]histamine 119
Histone Deacetylase (pfHDAC-1) pfHDAC-1 Substrate 23
Histone Deacetylase 1 (HDAC1) Ac-KGLGK(Ac)-AMC 14
acetyl-Gly-Ala-(N-acetyl-Lys)-AMC 5
Boc-Ac-Lys-AMC 1
Boc-Lys (Ac) -AMC 18
Carboxyfluorescein (FAM)-labeled acetylated peptide 18
Fluor de Lys-H4-AcK16 25
Fluor-de-Lys Fluorogenic Deacetylase Substrate 100
Fluorophore-conjugated substrate 3
[3H]acetyl-labeled histones 19
Histone Deacetylase 10 (HDAC10) acetyl-Gly-Ala-(N-acetyl-Lys)-AMC 1
Carboxyfluorescein (FAM)-labeled acetylated peptide 17
Histone Deacetylase 11 (HDAC11) Boc-Ac-Lys-AMC 1
Histone Deacetylase 2 (HDAC2) acetyl-Gly-Ala-(N-acetyl-Lys)-AMC 1
Boc-Ac-Lys-AMC 1
Boc-Lys (Ac) -AMC 18
Carboxyfluorescein (FAM)-labeled acetylated peptide 18
Fluor-de-Lys Fluorogenic Deacetylase Substrate 5
Histone Deacetylase 3 (HDAC3) acetyl-Gly-Ala-(N-acetyl-Lys)-AMC 1
Boc-Ac-Lys-AMC 1
Boc-Lys (Ac) -AMC 7
Carboxyfluorescein (FAM)-labeled acetylated peptide 17
Fluor-de-Lys Fluorogenic Deacetylase Substrate 62
Histone Deacetylase 4 (HDAC4) Ac-KGLGK(Ac)-AMC 8
Boc-Ac-Lys-AMC 1
Boc-L-Lys-MCA 48
[3H]acetyl-labeled histones 19
Histone Deacetylase 4 (HDAC4) Mutant (H976Y) Fluor-de-Lys Fluorogenic Deacetylase Substrate 48
Histone Deacetylase 5 (HDAC5) Boc-Ac-Lys-AMC 1
Boc-L-Lys-MCA 5
Histone Deacetylase 6 (HDAC6) Ac-KGLGK(Ac)-AMC 14
acetyl-Gly-Ala-(N-acetyl-Lys)-AMC 1
Boc-Ac-Lys-AMC 1
Carboxyfluorescein (FAM)-labeled acetylated peptide 18
Fluor-de-Lys Fluorogenic Deacetylase Substrate 47
Fluorophore-conjugated substrate 3
[3H]acetyl-labeled histones 19
Histone Deacetylase 7 (HDAC7) Boc-Ac-Lys-AMC 1
Boc-L-Lys-MCA 5
Histone Deacetylase 8 (HDAC8) acetyl-Gly-Ala-(N-acetyl-Lys)-AMC 1
Boc-Ac-Lys-AMC 1
Boc-Lys (Ac) -AMC 7
Carboxyfluorescein (FAM)-labeled acetylated peptide 18
Fluor de Lys-HDAC8 Fluorogenic Deacetylase Substrate 22
Fluorophore-conjugated substrate 3
Histone Lysine Demethylase Histone H3 fragment substrate 19
Histone-Arginine Methyltransferase CARM1 Histone H3 19
HIV-1 Integrase Biotinylated Target DNA 144
DIG-tagged Target DNA 13
[3H]Target DNA 88
HIV-1 Protease Biotinylated HIV-1 Protease Peptide Substrate 84
Chromogenic peptide substrate 5
Chromogenic peptide substrate 74
Chromogenic Substrate 3
decapeptide substrate 46
fluorescence peptide substrate 1
Fluorescent peptide substrate 408
Fluorogenic Peptide Substrate 324
fluorogenic peptide substrate, SQNY/PIVQ 4
Fluorogenic substrate 13
Fluorogenic substrate Abz-NF-6* 11
HIV Peptide Substrate 2
HIV Protease Chromogenic Peptide Substrate 7
HIV Protease peptide substrate 304
HIV Protease substrate 268
HIV-1 Peptide Substrate 83
HIV-1 PR Substrate Peptide 11
HIV-1 Protease substrate 111
HIV-1 proteinase peptide substrate 18
Peptide substrate 721
[3H]GW0385 16
HIV-1 Protease AE HIV Protease Chromogenic Peptide Substrate 7
HIV-1 Protease AE Mutant (V82F) HIV Protease Chromogenic Peptide Substrate 7
HIV-1 Protease AE-P HIV Protease Chromogenic Peptide Substrate 7
HIV-1 Protease AE-P Mutant (F82V) HIV Protease Chromogenic Peptide Substrate 7
HIV-1 Protease B Subtype HIV Protease Chromogenic Peptide Substrate 7
HIV-1 Protease B Subtype Mutant (V82F) HIV Protease Chromogenic Peptide Substrate 7
HIV-1 Protease Mutant (A71V) Chromogenic peptide substrate 5
HIV-1 Protease Mutant (A71V/V82T/I84V) Chromogenic peptide substrate 1
HIV-1 Protease Mutant (D30N) Chromogenic peptide substrate 5
HIV Peptide Substrate 2
HIV-1 Protease Mutant (D30N/A71V) Chromogenic peptide substrate 5
HIV-1 Protease Mutant (D30N/M36I) Chromogenic peptide substrate 5
HIV-1 Protease Mutant (D30N/M36I/A71V) Chromogenic peptide substrate 5
HIV-1 Protease Mutant (G73S) Chromogenic Substrate 3
HIV-1 Protease Mutant (I47L) HIV-1 Protease substrate 1
HIV-1 Protease Mutant (I50L) HIV-1 Protease substrate 1
HIV-1 Protease Mutant (I50V) Chromogenic Substrate 3
fluorescence peptide substrate 1
HIV Peptide Substrate 2
[3H]GW0385 5
HIV-1 Protease Mutant (I84V) HIV Peptide Substrate 2
HIV-1 Protease substrate 1
HIV-1 Protease Mutant (L10I,L19Q,K20R,E35D,M36I, ..) fluorescence peptide substrate 1
[3H]GW0385 5
HIV-1 Protease Mutant (L23I) HIV-1 Protease substrate 1
HIV-1 Protease Mutant (L23V) HIV-1 Protease substrate 1
HIV-1 Protease Mutant (L24I) Chromogenic Substrate 3
HIV-1 Protease Mutant (L76M) HIV-1 Protease substrate 1
HIV-1 Protease Mutant (L90M) HIV Peptide Substrate 2
HIV-1 Protease Mutant (M36I) Chromogenic peptide substrate 5
HIV-1 Protease Mutant (M36I/A71V) Chromogenic peptide substrate 5
HIV-1 Protease Mutant (M46I,L63P,A71V,V82F,I84V) fluorescence peptide substrate 1
[3H]GW0385 5
HIV-1 Protease Mutant (V32I) HIV-1 Protease substrate 1
HIV-1 Protease Mutant (V82A) HIV Peptide Substrate 2
HIV Protease Chromogenic Peptide Substrate 3
HIV-1 Protease Mutant (V82I) HIV-1 Protease substrate 1
HIV-1 Protease Mutant K-60C HIV Protease Peptide Substrate 15
HIV-1 Protease Mutant M1 (L10I, G48V, I54V, L63P, V82A) HIV-1 Protease Substrate 19
HIV-1 Protease Mutant M2 (D30N, L63P, N88D) HIV-1 Protease Substrate 19
HIV-1 Protease Mutant M3 (L10I, L63P, A71V, G73S, I84V, L90M) HIV-1 Protease Substrate 19
HIV-1 Protease Mutant Q-60C HIV Protease Peptide Substrate 11
HIV-1 Protease Mutant V-18C HIV Protease Peptide Substrate 27
HIV-1 Protease Mutant V6 HIV Protease Chromogenic Peptide Substrate 4
HIV-1 Protease Mutant V6(46) HIV Protease Chromogenic Peptide Substrate 4
HIV-1 Protease Mutant V6(46/54/84) HIV Protease Chromogenic Peptide Substrate 4
HIV-1 Protease Mutant V6(46/84) HIV Protease Chromogenic Peptide Substrate 4
HIV-1 Protease Mutant V6(54) HIV Protease Chromogenic Peptide Substrate 4
HIV-1 Protease Mutant V6(54/84) HIV Protease Chromogenic Peptide Substrate 4
HIV-1 Protease Mutant V6(84) HIV Protease Chromogenic Peptide Substrate 4
HIV-1 Protease Mutant, A-1 fluorogenic peptide substrate, SQNY/PIVQ 4
HIV-1 Protease Mutant, ANAM-11 fluorogenic peptide substrate, SQNY/PIVQ 4
HIV-1 Protease Mutant, NAM-10 fluorogenic peptide substrate, SQNY/PIVQ 4
HIV-1 Reverse Transcriptase (poly)rA:(oligo)dT(12-18) 139
(poly)rC:(oligo)dG 224
(rC)n.(dG)12-18 149
poly r(A).oligo d(T)16 10
poly rC/biotin-dG15 36
poly(A)/oligo(dT) 26
Poly(C)-oligo(dG) 7
poly(rA)-oligo(dT) 5
poly(rA)-oligo(dT)(12-18) 11
poly(rA).oligo(dT)12-18 28
poly(rA)/oligo(dT) 14
poly(rA)600:oligo(dT)10 45
poly(rA):oligo(dT) template:primer 11
poly(rA):oligo(dT)(12-18) 33
poly(rC)-oligo(dG) 13
poly(rC)-oligo(dG)(12-18) 183
poly(rC)500:oligo(dG)10 103
Poly(rC):oligo(dG )Template:Primer 50
poly(rC):oligo(dG) 313
RNA template(1080) : deoxy-oligo primer(18) 83
RNA:Biotin-DNA template:primer 10
RNA:DNA template:primer 70
HIV-1 Reverse Transcriptase Mutant (103N/181C) poly rC/biotin-dG15 26
RNA:Biotin-DNA template:primer 10
HIV-1 Reverse Transcriptase Mutant (G190A) poly(rC)500:oligo(dG)10 9
HIV-1 Reverse Transcriptase Mutant (K103N) (poly)rC:(oligo)dG 8
(rC)n.(dG)12-18 22
poly r(A).oligo d(T)16 5
poly(rA)/oligo(dT) 5
poly(rC)-oligo(dG)(12-18) 4
poly(rC)500:oligo(dG)10 10
Poly(rC):oligo(dG )Template:Primer 50
HIV-1 Reverse Transcriptase Mutant (K103N/Y181C) poly rC/biotin-dG15 11
HIV-1 Reverse Transcriptase Mutant (L100I) (rC)n.(dG)12-18 47
poly(rA)-oligo(dT) 5
poly(rA)/oligo(dT) 4
poly(rC)-oligo(dG)(12-18) 5
HIV-1 Reverse Transcriptase Mutant (L100I/K103N) poly(rA).oligo(dT)12-18 3
HIV-1 Reverse Transcriptase Mutant (P236L) poly(rA)600:oligo(dT)10 43
poly(rC)500:oligo(dG)10 10
HIV-1 Reverse Transcriptase Mutant (V106A) poly(rA)/oligo(dT) 3
poly(rC)500:oligo(dG)10 9
HIV-1 Reverse Transcriptase Mutant (V179D) poly(rA)/oligo(dT) 5
HIV-1 Reverse Transcriptase Mutant (Y181C) (poly)rC:(oligo)dG 7
(rC)n.(dG)12-18 69
poly r(A).oligo d(T)16 4
poly(rA)-oligo(dT) 5
poly(rA).oligo(dT)12-18 3
poly(rA)600:oligo(dT)10 40
poly(rC)-oligo(dG)(12-18) 10
poly(rC)500:oligo(dG)10 93
Poly(rC):oligo(dG )Template:Primer 46
poly(rC):oligo(dG) 63
HIV-1 Reverse Transcriptase Mutant (Y181I) poly(rA)/oligo(dT) 5
HIV-1 Reverse Transcriptase Mutant (Y188L) poly(rA)/oligo(dT) 3
poly(rC)500:oligo(dG)10 59
HIV-1 Reverse Transcriptase RNase H RNA/DNA hybrid 374
HIV-1 Reverse Transcriptase RNase H Mutant (D67N/K70R/T215F/K219Q) RNA/DNA hybrid 2
HIV-1 Reverse Transcriptase RNase H Mutant (L100I/K103N) RNA/DNA hybrid 2
HIV-1 Reverse Transcriptase RNase H Mutant (V106A/Y181C) RNA/DNA hybrid 2
HIV-1 Reverse Transcriptase RNase H Mutant (Y181C) RNA/DNA hybrid 2
HIV-1 Reverse Transcriptase RNase H Mutant (Y188L) RNA/DNA hybrid 2
HIV-2 Protease decapeptide substrate 7
HIV Protease Peptide Substrate 13
HIV-1 Protease substrate 1
Peptide Substrate 1
HIV-2 Reverse Transcriptase poly(rC)-oligo(dG)(12-18) 3
HIV-2 Reverse Transcriptase RNase H RNA/DNA hybrid 2
HMG-CoA Reductase HMG-CoA 107
Homoisocitrate Dehydrogenase (HICDH) Homoisocitrate 12
I-kappa-B Kinase 1 (IKK-alpha) I-kappa-B-alpha 142
I-kappa-B Kinase 2 (IKK-beta) Biotinylated I-kappa-B-alpha Peptide Substrate 22
I-kappa-B-alpha 151
I-kappa-B Kinase 3 (IKK-epsilon) I-kappa-B-alpha 40
Immunophilin FKBP12 N-succinyl Ala-Leu-Pro-Phe p-nitroanilide 79
IMP Cyclohydrolase (IMPCH) FAICAR 3
Indoleamine 2,3-Dioxygenase L-tryptophan 108
Inosine Monophosphate Dehydrogenase Type 1 (IMPDH1) IMP 14
Inosine Monophosphate Dehydrogenase Type 2 (IMPDH2) IMP 40
Insulin Receptor Tyrosine Kinase (IRK) Insulin Kinase Peptide Substrate 5
peptide 1150 1
Peptide Substrate 8
poly Glu4: Tyr 77
polyGlu4Tyr 4
Insulin Receptor-Related Protein (INSRR) biotinylated affinity ligand 6
Insulin-like Growth Factor 1 Receptor (IGF-1R) biotinylated gastrin substrate 2
Biotinylated substrate peptide 160
Peptide Substrate 8
poly (Glu/Tyr) 10
Integrin alpha1beta1 Collagen IV 5
Integrin alpha2beta1 Collagen I 33
Integrin alpha4beta1 (VLA-4) biotinylated CS-1 peptide 61
Eu-Labeled Human VCAM-1/Fc Chimera 42
Tritiated 3H Standard Compound A 44
VCAM-1 101
Integrin alpha4beta7 MAdCAM-1 71
Integrin alpha5beta1 Fibronectin 5
Kallikrein benzyloxycarbonyl-Phe-Arg-7-amino-4-methylcoumarin 27
Pefachrome FVIIa 27
Kappa Opioid Receptor [3H]-diprenorphine 90
[3H]U69593 5
KIAA1363 FP-rhodamine 1
Kinesin Spindle Protein Eg5 ATP 198
KIT(D816V) biotinylated affinity ligand 23
KIT(V559D T670I) biotinylated affinity ligand 19
Kynurenine Aminotransferase 1/Glutamine Transaminase K Kynurenine 2
Lactate Dehydrogenase Lactate 52
Pyruvate 16
Lck biotinylated gastrin substrate 60
Biotinylated peptide substrate 54
Enolase 78
Gastrin Peptide Substrate 35
N-biotinyl peptide substrate 1
Not Specified 1
poly-Glu-Ala-Tyr 16
Leucine Aminopeptidase L-Leucine-para-nitroanilide 19
Leukotriene A4 Hydrolase Alanine para-nitroanilide 75
Leukotriene A4 42
Lipoxygenase-1 Sodium linoleate 8
Liver Receptor Homolog 1 Biotinylated TIF2 Peptide 23
Liver X Receptor alpha (LXR-alpha) biotinylated SRC-1 peptide 85
GW3965 4
Not Available 18
T0901317 39
[3H]T0901317 76
Liver X Receptor beta (LXR-beta) biotinylated SRC-1 peptide 137
GW3965 4
Not Available 18
T0901317 39
[3H]T0901317 74
Malate Dehydrogenase (pfMDH) Oxaloacetic acid 8
Malate Dehydrogenase, cytoplasmic Oxaloacetic acid 7
Malate Dehydrogenase, mitochondrial Oxaloacetic acid 9
Mammalian Target of Rapamycin (mTOR) GFP-4EBP 1
S6K1 91
MAP Kinase Kinase 1 (MEK1) biotin-MBP protein 1
MAP Kinase p38 alpha ATF-2-GST 129
biotinylated ATF2 substrate 28
biotinylated GST-ATF2 56
biotinylated-ATF2 60
Epidermal Growth Factor Receptor Peptide (EGFRP) 12
myelin basic protein 136
Not Available 28
Rhodamine-green Labelled Fluoroligand 33
SKF 86002 12
Substrate Peptide T669 5
MAP Kinase p38 alpha Mutant (G110A) biotinylated GST-ATF2 6
MAP Kinase p38 alpha Mutant (G110D) biotinylated GST-ATF2 6
MAP Kinase p38 beta biotinylated GST-ATF2 15
MAP Kinase-Interacting Protein Kinase (MNK1) MBP 4
MAP-Microtubule Affinity-Regulating Kinase 3 (MARK3) CHKtide Substrate 1
MAP4K4 (HGK) Substrate Peptide SerThr 07 1
MAPK-Activated Protein Kinase 2 (MK2) Biotinylated GST-LSP1 102
HSP27 Peptide 31
Hsp27 Substrate Peptide 17
MAPK-Activated Protein Kinase 3 (MK3) Peptide Substrate 4
MAPK-Activated Protein Kinase 5 (MK5) Peptide Substrate 4
Matriptase Pefachrome tPA 54
t-Boc-Gln-Ala-Arg-AMC 14
Matrix Metalloproteinase-1 (MMP-1) Fluorescence-quenched peptide substrate 1
Fluorogenic Peptide Substrate 10
MMP Fluorogenic Peptide Substrate 27
MMP Substrate Peptide 3
MMP Thioester Substrate 91
NFF-2 Substrate 53
OmniMMP Substrate 2
Unknown 1
Wammp-5 2
Matrix Metalloproteinase-10 (MMP-10) Fluorescence-quenched peptide substrate 1
MMP Substrate Peptide 3
Matrix Metalloproteinase-12 (MMP-12) Fluorescence-quenched peptide substrate 6
MMP Fluorogenic Substrate 32
MMP Substrate Peptide 20
Not Available 5
OmniMMP Substrate 2
Wammp-5 4
Matrix Metalloproteinase-13 (MMP-13) 5-FAM/QXL 520 Peptide Substrate 23
Fluorescence-quenched peptide substrate 1
Fluorogenic Peptide Substrate 10
MMP Fluorogenic Peptide Substrate 27
MMP Fluorogenic Substrate 36
MMP Substrate Peptide 3
MMP-13 Fluorogenic Peptide Substrate 2
MMP-13 Substrate 64
Wammp-5 51
Matrix Metalloproteinase-14 (MMP-14) OmniMMP Substrate 2
Wammp-5 9
Matrix Metalloproteinase-2 (MMP-2) 5-FAM/QXL520 27
Fluorogenic Peptide Substrate 10
MMP Fluorogenic Peptide Substrate 34
MMP Substrate Peptide 19
MMP Thioester Substrate 91
OmniMMP Substrate 2
Unknown 1
Wammp-5 39
Matrix Metalloproteinase-3 (MMP-3) MMP Fluorogenic Peptide Substrate 7
MMP Substrate Peptide 19
MMP-3 Fluorogenic Peptide Substrate 19
NFF-2 Substrate 4
Substance P 62
Matrix Metalloproteinase-7 (MMP-7) Fluorescence-quenched peptide substrate 1
MMP Substrate Peptide 19
OmniMMP Substrate 2
Wammp-5 7
Matrix Metalloproteinase-8 (MMP-8) Fluorescence-quenched peptide substrate 1
MMP Fluorogenic Peptide Substrate 18
MMP Substrate Peptide 3
MMP Thioester Substrate 91
OmniMMP Substrate 2
Wammp-5 7
Matrix Metalloproteinase-9 (MMP-9) 5-FAM/QXL520 27
Fluorogenic Peptide Substrate 10
MMP Fluorogenic Peptide Substrate 19
MMP Substrate Peptide 3
MMP Thioester Substrate 91
NFF-2 Substrate 4
OmniMMP Substrate 2
Unknown 1
Wammp-5 8
Mcl-1 FITC-conjugated-Bim BH3 Peptide 10
MEK Kinase 1 (MEKK1) MBP 1
Melanin-Concentrating Hormone Receptor 1 (MCH1R) [125I]-MCH 21
Methionine Aminopeptidase (MAP) Met-Gly-Met-Met 14
Met-Pro-pNA 6
Methionine Aminopeptidase Type 1 (MetAP1) Met-Pro-pNA 5
Octapeptide substrate 9
Methionine Aminopeptidase Type 2 (MetAP2) Met-AMC 124
Met-Pro-pNA 5
Octapeptide substrate 159
Methylthioadenosine Nucleosidase(MTAN) MTA 6
Methylthioadenosine Phosphorylase (MTAP) MTA 3
Mineralocorticoid Receptor (MR) Aldosterone 11
dexamethasone 8
dexamethasone (tetramethyl-rhodamine conjugated ) 3
Mitogen- and Stress-Activated Protein Kinase 1 (MSK1) Crosstide 11
Peptide Substrate 4
Mitogen- and Stress-Activated Protein Kinase 2 (MSK2) Peptide Substrate 4
Mitogen-Activated Protein Kinase 1 Myelin basic protein 4
Mitogen-Activated Protein Kinase 10 (JNK3) biotinylated GST-ATF2 10
biotinylated-ATF2 47
EGF receptor peptide 29
fluorescently labelled inhibitor 4
Rhodamine-green Labelled Fluoroligand 4
Mitogen-Activated Protein Kinase 8 (JNK1) ATF2 45
Biotin-GST-c-JUN 34
Biotin-labeled pepJIP1 45
biotinylated GST-ATF2 6
biotinylated-ATF2 43
GST-ATF2 149
Mitogen-Activated Protein Kinase 9 (JNK2) biotinylated affinity ligand 5
biotinylated GST-ATF2 6
GST-ATF2 69
Mixed Lineage Kinase 1 (MLK1) Myelin basic protein 37
Mixed Lineage Kinase 2 (MLK2) Myelin basic protein 8
Mixed Lineage Kinase 3 (MLK3) Myelin basic protein 37
MKP-3 3-O-methylfluorescein phosphate (OMFP) 45
ML-IAP-BIR AVP-diPhe-FAM 32
Monoamine Oxidase Type A (MAO-A) 5-hydroxy tryptamine creatinine disulfate 79
kinuramine 34
Kynuramine 59
p-Tyramine 79
Monoamine Oxidase Type B (MAO-B) benzylamine 21
kinuramine 34
Kynuramine 38
MMTP 16
p-Tyramine 79
phenylethylamine 78
Monoamine oxidase type B (MAO-B) Mutant (I199F) benzylamine 5
Monocarboxylate Transporter 1 [125I]-pyrrolo[3,4-d]pyridazin-1-one 8
[3H]-pyrrolo[3,4-d]pyrimidine-2,4(3H,6H)-dione 35
Monoglyceride Lipase (MGL) 2-arachidonoylglycerol (2-AG) 21
FP-rhodamine 1
MPI protein Mannose-6-phosphate 462
MRCK alpha S6-peptide 5
Mu Opioid Receptor [3H]-diprenorphine 106
[3H]DAMGO 56
MurD D-[14C]Glu 37
Myosin Light-Chain Kinase Myosin Light-Chain 18
NAD-Dependent Deacetylase Sirtuin-1 Fluor de Lys-SIRT1 21
NAD-Dependent Deacetylase Sirtuin-2 Fluor de Lys-SIRT2 20
Neuraminidase A neuraminidase substrate 270
Neuraminidase B neuraminidase substrate 181
Neutral Endopeptidase DGPA 29
Neutrophil Elastase (NE) N-methylsuccinyl-Ala-Ala-Pro-Val-7-amino-4-methylcoumarin 33
Suc-Ala-Pro-Ala-MCA 23
Niacin Receptor GPR109A [5, 6-3H]-niacin 18
Nitric Oxide Synthase, brain L-arginine 24
Not Available 30
Nitric Oxide Synthase, brain Mutant (D597N) L-arginine 3
Nitric Oxide Synthase, brain Mutant (D597N/M336V) L-arginine 4
Nitric Oxide Synthase, endothelial L-arginine 24
Not Available 32
Nitric Oxide Synthase, endothelial Mutant (N368D) L-arginine 3
Nitric Oxide Synthase, inducible L-arginine 14
Not Available 41
NK1 Receptor Substance P 23
Nociceptin Receptor (ORL1 Receptor) leucyl-[3H]nociceptin 21
[125I]-nociceptin 89
[125I]Tyr14-Nociceptin 58
Norepinephrine Transporter (NET) [125I]RTI-55 29
[3H]NE 6
[3H]Nisoxetine 40
Orotidine Monophosphate Decarboxylase (ODCase) OMP 23
p53-Binding Protein HDMX p53 Peptide 25
p53-Binding Protein MDM2 6-FAM labeled octapeptide 20
biotinylated IP3 peptide 45
biotinylated p53-derived peptide 9
Fl 9mer 55
GST-p53 1