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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
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Ki
IC50
Kd
EC50
ΔG°
ΔH°
-TΔS°
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Compound Name:
Exact
Starts With
Ends With
Contain
< Molecular Weight <
< KI <
nM
< IC50 <
nM
< ΔG° <
kcal/mole
AND
OR
0-9
&
(
A
B
C
D
E
F
G
H
I
J
K
L
M
N
O
P
Q
R
S
T
U
V
W
X
Y
Z
[
RAC-alpha serine/threonine-protein kinase
[
36
] [
3D
]
RAC-alpha serine/threonine-protein kinase (Akt)
[
36
] [
3D
]
RAD51-BRCA2 BRC repeat complex
[
2
] [
3D
]
RAF proto-oncogene serine/threonine-protein kinase
[
2
] [
3D
]
RAF proto-oncogene serine/threonine-protein kinase (c-Raf)(Y340D)(Y341D)
[
9
] [
3D
]
RAF serine/threonine protein kinase
[
9
] [
3D
]
RAF-1
[
1
] [
3D
]
RAMP1
[
1
] [
3D
]
Rap guanine nucleotide exchange factor 3
[
13
] [
3D
]
Rap guanine nucleotide exchange factor 4
[
13
] [
3D
]
RAR-related orphan receptor C (RORc)
[
132
] [
3D
]
RAS guanyl releasing protein 1
[
132
] [
3D
]
RAS guanyl releasing protein 3
[
52
] [
3D
]
RAS guanyl-releasing protein 1
[
52
] [
3D
]
ras protein
[
196
] [
3D
]
Ras-related C3 botulinum toxin substrate 1
[
196
] [
3D
]
Ras-related C3 botulinum toxin substrate 1/T-lymphoma invasion and metastasis-inducing protein 1
[
18
] [
3D
]
Ras-related protein Rab-2A.
[
18
] [
3D
]
Ras-related protein Rab-7L1
[
1
] [
3D
]
Ras-related protein Rap-1A
[
1
] [
3D
]
Receptor protein-tyrosine kinase erbB-2
[
13
] [
3D
]
Receptor tyrosine-protein kinase erbB-4 (HER4)
[
13
] [
3D
]
Receptor-histidine kinase AgrC
[
13
] [
3D
]
Receptor-interacting serine/threonine-protein kinase 1
[
13
] [
3D
]
Receptor-interacting serine/threonine-protein kinase 2
[
1
] [
3D
]
Receptor-interacting serine/threonine-protein kinase 3
[
1
] [
3D
]
Receptor-interacting serine/threonine-protein kinase 4
[
73
] [
3D
]
Receptor-type tyrosine-protein kinase FLT3
[
73
] [
3D
]
Receptor-type tyrosine-protein kinase FLT3 (FLT3)
[
1
] [
3D
]
Receptor-type tyrosine-protein kinase FLT3 (K663Q)
[
1
] [
3D
]
Receptor-type tyrosine-protein kinase FLT3 (R834Q)
[
1
] [
3D
]
Receptor-type tyrosine-protein phosphatase beta (PTPβ)
[
1
] [
3D
]
Receptor-type tyrosine-protein phosphatase epsilon (PTPε)
[
34
] [
3D
]
Receptor-type tyrosine-protein phosphatase F (LAR)
[
34
] [
3D
]
Receptor-type tyrosine-protein phosphatase gamma (PTPγ)
[
38
] [
3D
]
Receptor-type tyrosine-protein phosphatase mu (PTPμ)
[
38
] [
3D
]
Receptor-type tyrosine-protein phosphatase R
[
1
] [
3D
]
Receptor-type tyrosine-protein phosphatase S
[
1
] [
3D
]
RecName: Full=Zinc finger protein mex-5
[
1670
] [
3D
]
Redox-regulatory protein FAM213A
[
1
] [
3D
]
regulator of G-protein signaling 4
[
192
] [
3D
]
Regulator of G-protein signaling 4 (RGS4)
[
192
] [
3D
]
Regulator of G-protein signaling 8
[
235
] [
3D
]
regulator of G-protein signalling 16
[
235
] [
3D
]
Regulatory protein E2
[
2
] [
3D
]
Relaxin receptor 1
[
2
] [
3D
]
Relaxin-3 receptor 1
[
12
] [
3D
]
Relaxin-3 receptor 2
[
12
] [
3D
]
Renal dipeptidase
[
193
] [
3D
]
Renal Outer Medullary Potassium (ROMK)
[
193
] [
3D
]
Renal sodium-dependent phosphate transport protein 1
[
1
] [
3D
]
Renin
[
1
] [
3D
]
Replicase polyprotein 1a
[
6
] [
3D
]
Replication protein A 70 kDa DNA-binding subunit
[
6
] [
3D
]
Replication protein E1
[
51
] [
3D
]
Replicative DNA helicase
[
51
] [
3D
]
REST corepressor 1
[
15
] [
3D
]
RET Mutant (M918T)
[
15
] [
3D
]
Ret proto-oncogene
[
2
] [
3D
]
Retina-specific amine oxidase, copper containing
[
2
] [
3D
]
Retinal dehydrogenase 2
[
4
] [
3D
]
Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta
[
4
] [
3D
]
Retinoic acid receptor alpha
[
43
] [
3D
]
Retinoic acid receptor alpha/Retinoid X receptor alpha
[
43
] [
3D
]
Retinoic acid receptor beta
[
20
] [
3D
]
Retinoic acid receptor gamma
[
20
] [
3D
]
Retinoic acid receptor RXR-alpha
[
5
] [
3D
]
Retinoic acid receptor RXR-alpha/gamma
[
5
] [
3D
]
Retinoic acid receptor RXR-alpha/oxysterols receptor LXR-alpha
[
15
] [
3D
]
Retinoic acid receptor RXR-alpha/oxysterols receptor LXR-beta
[
15
] [
3D
]
Retinoic acid receptor RXR-alpha/Retinoic acid receptor beta
[
44
] [
3D
]
Retinoic Acid Receptor, alpha
[
44
] [
3D
]
Retinoic Acid Receptor, beta
[
10
] [
3D
]
Retinoic Acid Receptor, gamma
[
10
] [
3D
]
Retinoic Acid Receptors Gamma / Alpha
[
2
] [
3D
]
Retinoic acid-related nuclear receptor gamma t (RORγt)
[
2
] [
3D
]
Retinoic acid-related nuclear receptor gamma t (RORγt)
[
44
] [
3D
]
Retinoid receptor
[
44
] [
3D
]
Retinoid X receptor
[
2
] [
3D
]
Retinoid X receptor alpha
[
2
] [
3D
]
Retinoid X receptor alpha (F313I/L436F)
[
1
] [
3D
]
Retinoid X receptor alpha (F313I/L436V)
[
1
] [
3D
]
Retinoid X receptor beta
[
97
] [
3D
]
Retinoid X receptor gamma
[
97
] [
3D
]
Retinoid X receptor gamma/retinoic acid receptor alpha
[
345
] [
3D
]
Retinoid-related orphan receptor gamma (RORγ-LBD)
[
345
] [
3D
]
Retinoid-related orphan receptor-gamma (RORgT)
[
157
] [
3D
]
Retinol-binding protein 4 (RBP4)
[
157
] [
3D
]
Reverse transcriptase
[
304
] [
3D
]
Reverse Transcriptase (HIV-1 K103N RT)
[
304
] [
3D
]
Reverse transcriptase (HIV-1 RT)(1-350)
[
4
] [
3D
]
Reverse transcriptase protein
[
4
] [
3D
]
RGS7
[
192
] [
3D
]
Rhizopuspepsin
[
192
] [
3D
]
Rho Kinase 1
[
6
] [
3D
]
Rho kinase 2 (ROCKII)
[
6
] [
3D
]
Rho Transcription Termination Factor
[
2
] [
3D
]
Rho-associated protein kinase
[
2
] [
3D
]
Rho-associated protein kinase 1 (ROCK I)
[
4
] [
3D
]
Rho-associated protein kinase 1 (ROCK1)
[
4
] [
3D
]
Rho-associated protein kinase 2 (ROCK II)
[
6
] [
3D
]
Rho-associated protein kinase 2 (ROCK2)
[
6
] [
3D
]
Rho-associated protein kinase 2/Rho-kinase (ROCK I)
[
90
] [
3D
]
Rho-GTPase-activating protein 3
[
90
] [
3D
]
Rho-kinase (ROCK II)
[
12
] [
3D
]
Rho/Rac guanine nucleotide exchange factor
[
12
] [
3D
]
Rhodesain
[
172
] [
3D
]
Rhodopsin
[
172
] [
3D
]
Rhodopsin kinase
[
108
] [
3D
]
Rhomboid protease (AaROM)
[
108
] [
3D
]
Rhomboid protease (AfROM)
[
2
] [
3D
]
Rhomboid protease (BsYqgP)
[
2
] [
3D
]
Rhomboid protease (EcGlpG)
[
2
] [
3D
]
Rhomboid protease (HiGlpG)
[
2
] [
3D
]
Rhomboid protease (MmRHBDL1)
[
2
] [
3D
]
Rhomboid protease (MmRHBDL3)
[
2
] [
3D
]
Rhomboid protease (PhROM)
[
2
] [
3D
]
Rhomboid protease (PsAarA)
[
2
] [
3D
]
Rhomboid protease (TmROM)
[
4
] [
3D
]
Rhomboid protease (VcROM)
[
4
] [
3D
]
Riboflavin-binding protein
[
5
] [
3D
]
Ribokinase
[
5
] [
3D
]
Ribonuclease H
[
10
] [
3D
]
Ribonuclease H1
[
10
] [
3D
]
Ribonucleoside-diphosphate reductase large chain
[
63
] [
3D
]
Ribonucleoside-diphosphate reductase M1 chain
[
63
] [
3D
]
Ribonucleoside-diphosphate reductase M1 chain/Ribonucleoside-diphosphate reductase M2 chain/Ribonucleotide reductase
[
1
] [
3D
]
Ribonucleoside-diphosphate reductase M1 chain/Ribonucleotide reductase
[
1
] [
3D
]
Ribonucleoside-diphosphate reductase M1/M2 chain
[
75
] [
3D
]
Ribonucleoside-diphosphate reductase RR1
[
75
] [
3D
]
Ribonucleoside-diphosphate reductase subunit alpha
[
7
] [
3D
]
Ribose-5-phosphate isomerase B
[
7
] [
3D
]
Ribose-phosphate pyrophosphokinase I
[
4
] [
3D
]
Ribosomal protein S6 kinase (P70S6K)
[
4
] [
3D
]
Ribosomal protein S6 kinase 2/S6K1
[
5
] [
3D
]
Ribosomal protein S6 kinase alpha 1
[
5
] [
3D
]
Ribosomal protein S6 kinase alpha 2
[
324
] [
3D
]
Ribosomal protein S6 kinase alpha 3
[
324
] [
3D
]
Ribosomal protein S6 kinase alpha 4
[
92
] [
3D
]
Ribosomal protein S6 kinase alpha 5
[
92
] [
3D
]
Ribosomal protein S6 kinase alpha 6
[
86
] [
3D
]
Ribosomal protein S6 kinase alpha-3
[
86
] [
3D
]
Ribosomal S6 Kinase 1 (RSK-1)
[
1
] [
3D
]
Ribosomal S6 kinase 2 (RSK-2)
[
1
] [
3D
]
Ribosomal S6 kinase 2 (RSK-2)(C436V)
[
19
] [
3D
]
Ribosyldihydronicotinamide dehydrogenase [quinone]
[
19
] [
3D
]
Ricin
[
67
] [
3D
]
RmtA
[
67
] [
3D
]
RNA polymerase (NS5B)
[
164
] [
3D
]
RNA polymerase beta subunit (EC 2.7.7.6)
[
164
] [
3D
]
RNA polymerase sigma factor SigB (σB)
[
4
] [
3D
]
RNA polymerase subunit beta (β-RNAP)
[
4
] [
3D
]
RNA polymerase subunit beta ([D516V]β-RNAP)
[
2
] [
3D
]
RNA polymerase subunit beta ([H526D]β-RNAP)
[
2
] [
3D
]
RNA polymerase subunit beta ([S531L]β-RNAP)
[
2
] [
3D
]
RNA(23-mer)
[
2
] [
3D
]
RNA-directed RNA polymerase (NS5B)
[
130
] [
3D
]
RNA-directed RNA polymerase (NS5B) (S282T)
[
130
] [
3D
]
RNA-directed RNA polymerase (NS5B)(C316Y)
[
1
] [
3D
]
RNA-directed RNA polymerase (NS5B)(L392I)
[
1
] [
3D
]
RNA-directed RNA polymerase (NS5B)(M414T)
[
1
] [
3D
]
RNA-directed RNA polymerase (NS5B)(M423T)
[
1
] [
3D
]
RNA-directed RNA polymerase (NS5B)(P495L)
[
1
] [
3D
]
RNA-directed RNA polymerase (NS5B)(S282T)
[
1
] [
3D
]
RNA-directed RNA polymerase (NS5B)(V494A)
[
1
] [
3D
]
RNAse A
[
1
] [
3D
]
RNase L
[
88
] [
3D
]
ROCK Complex
[
88
] [
3D
]
RocR
[
4
] [
3D
]
Rod cGMP-specific 3',5'-cyclic phosphodiesterase alpha/beta
[
4
] [
3D
]
Rod cGMP-specific 3',5'-cyclic phosphodiesterase subunit alpha
[
5
] [
3D
]
Rous sarcoma virus integrase
[
5
] [
3D
]
RPL19A
[
105
] [
3D
]
RPS6KA2(Kin.Dom.2 - C-terminal)
[
105
] [
3D
]
RPS6KA4(Kin.Dom.1 - N-terminal)
[
10
] [
3D
]
rRNA adenine N-6-methyltransferase
[
10
] [
3D
]
Runt-Related Transcription Factor 1 Isoform AML1C
[
114
] [
3D
]
RuvB-like 1
[
114
] [
3D
]
RXR alpha/PPAR gamma
[
480
] [
3D
]
RYamide receptor
[
480
] [
3D
]
Ryanodine receptor 1
[
44
] [
3D
]
Ryanodine receptor 2
[
44
] [
3D
]
Ryanodine receptor 44F
[
1
] [
3D
]