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Compound Name:

Compounds Sorted by Binding Data per Compound

1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29
30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 78 79 80 81
82 83 84 85 86 87 88 89 90 91 92 93 94 95 96 97 98 99 100 101 102 103 104 105
106 107 108 109 110 111 112 113 114 115 116 117 118 119 120 121 122 123 124
125 127 128 129 130 132 133 134 135 136 137 138 139 140 141 143 144 145 146
147 148 149 150 151 153 154 155 156 159 160 161 163 164 165 168 170 171 173
174 176 178 179 183 184 186 188 189 190 191 192 193 196 198 199 200 203 204
205 206 207 208 209 210 216 220 224 226 227 229 232 237 238 241 243 248 252
253 259 261 270 274 276 277 285 291 303 304 313 318 323 325 328 333 335 337
339 341 353 360 361 365 389 393 398 401 413 433 442 444 445 446 447 448 451
453 454 455 457 458 460 463 465 467 473 477 478 482 484 499 504 505 506 517
521 525 543 549 551 554 591 606 663 691 708 796 804 821 825 833 842 847 854
855 861 873 879 883 887 913 914 925 926 938 947 1010 1027 1050 1052 1081 1082
1099 1115 1130 1133 1206 1262 1543 1639 1903 2029
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Enz. Inhib. Data
ITC Data
Binding Targets
Alternate Compound Names
5 Ki 5 IC50
  • Beta-secretase 1
  • Cytochrome P450 3A
  • US8541427, 15
  • US8541427, 206
  • US8541427, 44
  • US8541427, 45
8 Ki 2 IC50
  • Caspase-1
  • Caspase-2
  • Caspase-3
  • Caspase-4
  • Caspase-6
  • Caspase-7
  • Caspase-8
  • Caspase-9
  • 5-(pyrrolidine-1-sulfonyl)-2,3-dihydro-1H-indole-2,3-dione
  • 5-[1-(Pyrrolidinyl)sulfonyl]isatin
  • Isatin Sulfonamide 20
8 Ki 2 IC50
  • Caspase-1
  • Caspase-2
  • Caspase-3
  • Caspase-4
  • Caspase-6
  • Caspase-7
  • Caspase-8
  • Caspase-9
  • (S)-5-{1-[2-(Anilinomethyl)pyrrolidinyl]sulfonyl}isatin
  • 5-{[(2S)-2-[(phenylamino)methyl]pyrrolidine-1-]sulfonyl}-2,3-dihydro-1H-indole-2,3-dione
  • Isatin Sulfonamide 26
10 IC50
  • JAK1 (aa 850-1154)
  • JAK2 (aa 808-1132)
  • JAK3 (aa 781-1124)
  • Non-receptor tyrosine-protein kinase TYK2
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • US10206907, Compound 234
  • US8563545, 11
7 Ki 3 EC50
  • Beta-2 adrenergic receptor
  • Muscarinic acetylcholine receptor M3
  • US8551978, I-85
  • US8816088, I-85
  • US9394275, I-86
  • US9572802, Compound I-87
  • US9682957, I-85
10 IC50
  • Cytochrome P450 1A
  • Cytochrome P450 2B6
  • Cytochrome P450 2C19
  • Cytochrome P450 2C9
  • Cytochrome P450 2D6 (2D6)
  • Cytochrome P450 3A
  • Sodium/glucose cotransporter 1 (SGLT1)
  • Sodium/glucose cotransporter 2
  • US8575114, I-12
8 Ki 2 IC50
  • 5-hydroxytryptamine receptor 1A
  • Acetylcholinesterase
  • Adrenergic alpha1B
  • Alpha-1A adrenergic receptor
  • Alpha-1D adrenergic receptor
  • Carboxylic ester hydrolase
  • Bivalent 4-Aminoquinoline 9f
  • N,N-di-4-Quinolyl-1,7-diaminoheptane dihydrochloride
  • N-[7-(quinolin-4-ylamino)heptyl]quinolin-4-amine dihydrochloride
1 Ki 9 IC50
  • Acetylcholinesterase
  • Acetylcholinesterase and butyrylcholinesterase (AChE and BChE)
  • Carboxylic ester hydrolase
  • Rhodesain
  • Trypanothione reductase
  • Bis-THA inhibitor 1c
  • Bis-THA inhibitor 8
  • CHEMBL424707
  • N-[9-(1,2,3,4-tetrahydroacridin-9-ylamino)nonyl]-1,2,3,4-tetrahydroacridin-9-amine
9 IC50 0 Other
  • ATP-binding cassette sub-family G member 2
  • CYP3A-M
  • Cytochrome P450 1A
  • Cytochrome P450 2C19
  • Cytochrome P450 2C8
  • Cytochrome P450 2C9
  • Cytochrome P450 2D6 (2D6)
  • P-glycoprotein 1
  • US9695174, I-1
10 IC50
  • Acetylcholinesterase
  • Cholinesterases
  • 3-{[methyl({3-[(9-oxo-9H-xanthen-3-yl)oxy]propyl})amino]methyl}phenyl N-methylcarbamate
  • CHEMBL340427
  • Xanthostigmine
  • aminoalkoxyheteroaryl deriv. 8
4 Ki 5 IC50 1 EC50
  • Cytochrome P450 2C9
  • Cytochrome P450 2D6 (2D6)
  • Cytochrome P450 3A
  • Nuclear receptor subfamily 1 group I member 2
  • Orexin receptor type 1
  • Orexin receptor type 2
  • US8592457, 7-5
1 Ki 9 IC50
  • Acetylcholinesterase
  • Bile salt export pump
  • Cholinesterases
  • Neuronal acetylcholine receptor subunit alpha-4
  • 1,3a,8-trimethyl-1H,2H,3H,3aH,8H,8aH-pyrrolo[2,3-b]indol-5-yl N-methylcarbamate
  • CHEMBL11773
  • Eserine
  • Physostigmine
10 IC50
  • 11-beta-hydroxysteroid dehydrogenase 1
  • Cytochrome P450 2C19
  • Cytochrome P450 2C9
  • Cytochrome P450 3A
  • US8575157, 194
  • US8592410, Comparator 6
  • US8598163, 64
10 IC50
  • 11-beta-hydroxysteroid dehydrogenase 1
  • Cytochrome P450 2C19
  • Cytochrome P450 2C9
  • Cytochrome P450 3A
  • US8575157, 199
  • US8592410, Comparator 11
  • US8598163, 69
10 IC50
  • 11-beta-hydroxysteroid dehydrogenase 1
  • Cytochrome P450 2C19
  • Cytochrome P450 2C9
  • Cytochrome P450 3A
  • US8575157, 202
  • US8592410, Comparator 14
  • US8598163, 72
10 IC50
  • 11-beta-hydroxysteroid dehydrogenase 1
  • Cytochrome P450 2C19
  • Cytochrome P450 2C9
  • Cytochrome P450 3A
  • US8575157, 203
  • US8592410, Comparator 15
  • US8598163, 73
10 Ki
  • Coagulation factor X
  • Coagulation factor XI
  • Complement C1r subcomponent
  • Complement C1s
  • Factor XIIa
  • Plasma kallikrein
  • Plasminogen
  • Tissue-type plasminogen activator
  • Transcription initiation factor IIA
  • Vitamin K-dependent protein C
  • US8598206, Table 6, 15
10 Ki
  • Coagulation factor X
  • Coagulation factor XI
  • Complement C1r subcomponent
  • Complement C1s
  • Factor XIIa
  • Plasma kallikrein
  • Plasminogen
  • Transcription initiation factor IIA
  • Vitamin K-dependent protein C
  • US8598206, Table 6, 24
10 Ki
  • Coagulation factor X
  • Coagulation factor XI
  • Complement C1r subcomponent
  • Complement C1s
  • Factor XIIa
  • Plasma kallikrein
  • Plasminogen
  • Tissue-type plasminogen activator
  • Transcription initiation factor IIA
  • Vitamin K-dependent protein C
  • US8598206, Table 6, 3
10 IC50
  • Apoptosis regulator Bcl-2
  • BCL-W
  • Bcl-2-like protein 1
  • Induced myeloid leukemia cell differentiation protein Mcl-1
  • Isoform Bcl-X(L)
  • 2-(8-(2-(Benzothiazol-2-yl)hydrazono)-5,6,7,8-tetrahydronaphthalen-2-yl)thiazole-4-carboxylic acid (Compound 4)
  • CHEMBL2398260
6 IC50 4 Kd
  • Apoptosis regulator Bcl-2
  • BCL-W
  • Induced myeloid leukemia cell differentiation protein Mcl-1
  • Isoform Bcl-X(L)
  • WEHI-539
5 Ki 2 IC50 3 Kd
  • Adrenergic receptor alpha-2
  • Cytochrome P450 130
  • Cytochrome P450 130 (G243A)
  • Cytochrome P450 142 (CYP142)
  • Lysyl oxidase homolog 2
  • Phenylethanolamine N-methyltransferase
  • Trypsin-1
  • Urease
  • Benzenemethanamine
  • CHEMBL522
  • benzylamine
  • phenylmethanamine
7 Ki 3 IC50
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Monoamine Oxidase Type B (MAO-B)
  • Monoamine oxidase type B (MAO-B) Mutant (I199F)
  • Neuraminidase A
  • Uridine-5'-diphosphoglucuronosyltransferase 1A1
  • (2E,6E)-3,7,11-trimethyldodeca-2,6,10-trien-1-ol
  • trans,trans-Farnesol
10 Ki
  • Carbonic anhydrase
  • Carbonic anhydrase 1
  • Carbonic anhydrase 2
  • Carbonic anhydrase 9
  • Carbonic anhydrase V
  • Carbonic anhydrases; II & IX
  • CHEMBL386049
  • N-(4-sulfamoylphenyl)-2-sulfanylbenzamide
  • reduced monomeric thio of compound 5a
  • reduced thio H5a
7 Ki 3 IC50
  • Cathepsin G
  • Chymotrypsin
  • Kallikrein 14
  • Kallikrein 5
  • Kallikrein 7
  • Prothrombin
  • Trypsin-1
  • US9695194, 5
10 Ki
  • 72 kDa type IV collagenase
  • Carbonic Anhydrase IV
  • Carbonic anhydrase 1
  • Carbonic anhydrase 2
  • Collagenase (ChC)
  • Interstitial collagenase
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Hydroxamate 7
  • N-hydroxy-2-[(1,1,2,2,3,3,4,4,4-nonafluorobutane)sulfonamido]acetamide
10 Ki
  • 72 kDa type IV collagenase
  • Carbonic Anhydrase IV
  • Carbonic anhydrase 1
  • Carbonic anhydrase 2
  • Collagenase (ChC)
  • Interstitial collagenase
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Hydroxamate 13
  • N-hydroxy-2-[(1,1,2,2,3,3,4,4,4-nonafluorobutane)sulfonamido]propanamide
  • N-n-Perfluorobutylsulfonyl-alanine hydroxamate
9 Ki 1 IC50
  • 72 kDa type IV collagenase
  • Carbonic Anhydrase IV
  • Carbonic anhydrase 1
  • Carbonic anhydrase 2
  • Collagenase (ChC)
  • Interstitial collagenase
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Hydroxamate 15
  • N-hydroxy-2-[(4-methoxybenzene)sulfonamido]propanamide
10 Ki
  • 72 kDa type IV collagenase
  • Carbonic Anhydrase IV
  • Carbonic anhydrase 1
  • Carbonic anhydrase 2
  • Collagenase (ChC)
  • Interstitial collagenase
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Hydroxamate 19
  • N-hydroxy-3-methyl-2-[(1,1,2,2,3,3,4,4,4-nonafluorobutane)sulfonamido]butanamide
10 Ki
  • 72 kDa type IV collagenase
  • Carbonic Anhydrase IV
  • Carbonic anhydrase 1
  • Carbonic anhydrase 2
  • Collagenase (ChC)
  • Interstitial collagenase
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Hydroxamate 25
  • N-hydroxy-4-methyl-2-[(1,1,2,2,3,3,4,4,4-nonafluorobutane)sulfonamido]pentanamide
10 Ki
  • 72 kDa type IV collagenase
  • Carbonic Anhydrase IV
  • Carbonic anhydrase 1
  • Carbonic anhydrase 2
  • Collagenase (ChC)
  • Interstitial collagenase
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Hydroxamate 27
  • N-hydroxy-2-[(4-methoxybenzene)sulfonamido]-4-methylpentanamide
2 Ki 8 IC50
  • Dipeptidyl peptidase 2 (DPP II)
  • Dipeptidyl peptidase 4
  • Dipeptidyl peptidase 9
  • Dipeptidyl peptidase VIII
  • Potassium voltage-gated channel subfamily H member 2
  • CHEMBL22310
  • N-{4-[(1S)-1-amino-2-[(3S)-3-fluoropyrrolidin-1-yl]-2-oxoethyl]cyclohexyl}-2,4-difluorobenzene-1-sulfonamide
  • difluorobenzenesulfonamide 1
10 IC50
  • Beta-secretase 1
  • Beta-secretase 2
  • IDH1 R132H
  • US10035794, Example 34
  • US10683287, Example 34
  • US8637508, 34
10 IC50
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
  • US8653092, 61
10 IC50
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
  • US8653092, 68
10 IC50
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
  • US8653092, 83
6 Ki 4 IC50
  • 72 kDa type IV collagenase
  • Collagenase 3
  • Interstitial collagenase
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Stromelysin-1
  • CHEMBL256157
  • N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride
  • N-hydroxy-4-{[(4-phenoxybenzene)sulfonyl]methyl}-1-(prop-2-yn-1-yl)piperidine-4-carboxamide hydrochloride
  • beta-sulfone 7e
10 Ki
  • 72 kDa type IV collagenase
  • Collagenase 3
  • Interstitial collagenase
  • Matrix metalloproteinase 10
  • Matrix metalloproteinase 14
  • Matrix metalloproteinase-12 (MMP12)
  • Matrix metalloproteinase-7 (MMP7)
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Stromelysin-1
  • US8691753, 3
10 Ki
  • 72 kDa type IV collagenase
  • Collagenase 3
  • Interstitial collagenase
  • Matrix metalloproteinase 10
  • Matrix metalloproteinase 14
  • Matrix metalloproteinase-12 (MMP12)
  • Matrix metalloproteinase-7 (MMP7)
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Stromelysin-1
  • US8691753, 14
10 Ki
  • 72 kDa type IV collagenase
  • Collagenase 3
  • Interstitial collagenase
  • Matrix metalloproteinase 10
  • Matrix metalloproteinase 14
  • Matrix metalloproteinase-12 (MMP12)
  • Matrix metalloproteinase-7 (MMP7)
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Stromelysin-1
  • US8691753, 40
10 Ki
  • 72 kDa type IV collagenase
  • Collagenase 3
  • Interstitial collagenase
  • Matrix metalloproteinase 10
  • Matrix metalloproteinase 14
  • Matrix metalloproteinase-12 (MMP12)
  • Matrix metalloproteinase-7 (MMP7)
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Stromelysin-1
  • US8691753, 80
10 Ki
  • 72 kDa type IV collagenase
  • Collagenase 3
  • Interstitial collagenase
  • Matrix metalloproteinase 10
  • Matrix metalloproteinase 14
  • Matrix metalloproteinase-12 (MMP12)
  • Matrix metalloproteinase-7 (MMP7)
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Stromelysin-1
  • US8691753, 99
10 Ki
  • 72 kDa type IV collagenase
  • Collagenase 3
  • Interstitial collagenase
  • Matrix metalloproteinase 10
  • Matrix metalloproteinase 14
  • Matrix metalloproteinase-12 (MMP12)
  • Matrix metalloproteinase-7 (MMP7)
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Stromelysin-1
  • US8691753, 101
10 Ki
  • 72 kDa type IV collagenase
  • Collagenase 3
  • Interstitial collagenase
  • Matrix metalloproteinase 10
  • Matrix metalloproteinase 14
  • Matrix metalloproteinase-12 (MMP12)
  • Matrix metalloproteinase-7 (MMP7)
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Stromelysin-1
  • US8691753, 103
10 Ki
  • 72 kDa type IV collagenase
  • Collagenase 3
  • Interstitial collagenase
  • Matrix metalloproteinase 10
  • Matrix metalloproteinase 14
  • Matrix metalloproteinase-12 (MMP12)
  • Matrix metalloproteinase-7 (MMP7)
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Stromelysin-1
  • US8691753, 106
10 Ki
  • 72 kDa type IV collagenase
  • Collagenase 3
  • Interstitial collagenase
  • Matrix metalloproteinase 10
  • Matrix metalloproteinase 14
  • Matrix metalloproteinase-12 (MMP12)
  • Matrix metalloproteinase-7 (MMP7)
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Stromelysin-1
  • US8691753, 95 bis
2 Ki 8 IC50
  • Dipeptidyl peptidase 2 (DPP II)
  • Dipeptidyl peptidase 4
  • Dipeptidyl peptidase VIII
  • (2S)-2-amino-2-cyclohexyl-1-(pyrrolidin-1-yl)ethan-1-one
  • (S)-2-Amino-2-cyclohexyl-1-pyrrolidin-1-yl-ethanone
  • (S)-2-amino-2-cyclohexyl-1-(pyrrolidin-1-yl)ethanone
  • CHEMBL278393
  • isoquinoline derivative 14
10 IC50
  • CDK2/CycE
  • Cyclin-Dependent Kinase 1 (CDK1)
  • Cyclin-Dependent Kinase 4 (CDK4)
  • Cyclin-Dependent Kinase 7 (CDK7)
  • Cyclin-Dependent Kinase 9 (CDK9)
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Cyclin-dependent kinase 4
  • Cyclin-dependent kinase 7
  • Cyclin-dependent kinase 9
  • AAP1742
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 1
  • US10758542, Example 1
  • US8791123, 1
  • US9782415, Example 1
  • US9796724, Example 1
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 2
  • US10758542, Example 2
  • US8791123, 2
  • US9782415, Example 2
  • US9796724, Example 2
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 3
  • US10758542, Example 3
  • US8791123, 3
  • US9782415, Example 3
  • US9796724, Example 3
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 4
  • US10758542, Example 4
  • US8791123, 4
  • US9782415, Example 4
  • US9796724, Example 4
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 5
  • US10758542, Example 5
  • US8791123, 5
  • US9782415, Example 5
  • US9796724, Example 5
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 6
  • US10758542, Example 6
  • US8791123, 6
  • US9782415, Example 6
  • US9796724, Example 6
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 7
  • US10758542, Example 7
  • US8791123, 7
  • US9782415, Example 7
  • US9796724, Example 7
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 8
  • US10758542, Example 8
  • US8791123, 8
  • US9782415, Example 8
  • US9796724, Example 8
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 9
  • US10758542, Example 9
  • US8791123, 9
  • US9782415, Example 9
  • US9796724, Example 9
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 10
  • US10758542, Example 10
  • US8791123, 10
  • US9782415, Example 10
  • US9796724, Example 10
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 13
  • US10758542, Example 13
  • US8791123, 13
  • US9782415, Example 13
  • US9796724, Example 13
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 14
  • US10758542, Example 14
  • US8791123, 14
  • US9782415, Example 14
  • US9796724, Example 14
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 15
  • US10758542, Example 15
  • US8791123, 15
  • US9782415, Example 15
  • US9796724, Example 15
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 16
  • US10758542, Example 16
  • US8791123, 16
  • US9782415, Example 16
  • US9796724, Example 16
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 18
  • US10758542, Example 18
  • US8791123, 18
  • US9782415, Example 18
  • US9796724, Example 18
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 19
  • US10758542, Example 19
  • US8791123, 19
  • US9782415, Example 19
  • US9796724, Example 19
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 20
  • US10758542, Example 20
  • US8791123, 20
  • US9782415, Example 20
  • US9796724, Example 20
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 21
  • US10758542, Example 21
  • US8791123, 21
  • US9782415, Example 21
  • US9796724, Example 21
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 22
  • US10758542, Example 22
  • US8791123, 22
  • US9782415, Example 22
  • US9796724, Example 22
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 23
  • US10758542, Example 23
  • US8791123, 23
  • US9782415, Example 23
  • US9796724, Example 23
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 24
  • US10758542, Example 24
  • US8791123, 24
  • US9782415, Example 24
  • US9796724, Example 24
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 26
  • US10758542, Example 26
  • US8791123, 26
  • US9782415, Example 26
  • US9796724, Example 26
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 27
  • US10758542, Example 27
  • US8791123, 27
  • US9782415, Example 27
  • US9796724, Example 27
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 28
  • US10758542, Example 28
  • US8791123, 28
  • US9782415, Example 28
  • US9796724, Example 28
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 29
  • US10758542, Example 29
  • US8791123, 29
  • US9782415, Example 29
  • US9796724, Example 29
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 31
  • US10758542, Example 31
  • US8791123, 31
  • US9782415, Example 31
  • US9796724, Example 31
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 32
  • US10758542, Example 32
  • US8791123, 32
  • US9782415, Example 32
  • US9796724, Example 32
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 35
  • US10758542, Example 35
  • US8791123, 35
  • US9782415, Example 35
  • US9796724, Example 35
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 36
  • US10758542, Example 36
  • US8791123, 36
  • US9782415, Example 36
  • US9796724, Example 36
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 37
  • US10758542, Example 37
  • US8791123, 37
  • US9782415, Example 37
  • US9796724, Example 37
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 40
  • US10758542, Example 40
  • US8791123, 40
  • US9782415, Example 40
  • US9796724, Example 40
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 41
  • US10758542, Example 41
  • US8791123, 41
  • US9782415, Example 41
  • US9796724, Example 41
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 42
  • US10758542, Example 42
  • US8791123, 42
  • US9782415, Example 42
  • US9796724, Example 42
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 43
  • US10758542, Example 43
  • US8791123, 43
  • US9782415, Example 43
  • US9796724, Example 43
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 53
  • US10758542, Example 53
  • US8791123, 53
  • US9782415, Example 53
  • US9796724, Example 53
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 58
  • US10758542, Example 58
  • US8791123, 58
  • US9782415, Example 58
  • US9796724, Example 58
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 59
  • US10758542, Example 59
  • US8791123, 59
  • US9782415, Example 59
  • US9796724, Example 59
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 60
  • US10758542, Example 60
  • US8791123, 60
  • US9782415, Example 60
  • US9796724, Example 60
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 61
  • US10758542, Example 61
  • US8791123, 61
  • US9782415, Example 61
  • US9796724, Example 61
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 62
  • US10758542, Example 62
  • US8791123, 62
  • US9782415, Example 62
  • US9796724, Example 62
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 63
  • US10758542, Example 63
  • US8791123, 63
  • US9782415, Example 63
  • US9796724, Example 63
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 64
  • US10758542, Example 64
  • US8791123, 64
  • US9782415, Example 64
  • US9796724, Example 64
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 65
  • US10758542, Example 65
  • US8791123, 65
  • US9782415, Example 65
  • US9796724, Example 65
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 66
  • US10758542, Example 66
  • US8791123, 66
  • US9782415, Example 66
  • US9796724, Example 66
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 67
  • US10758542, Example 67
  • US8791123, 67
  • US9782415, Example 67
  • US9796724, Example 67
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 68
  • US10758542, Example 68
  • US8791123, 68
  • US9782415, Example 68
  • US9796724, Example 68
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 71
  • US10758542, Example 71
  • US8791123, 71
  • US9782415, Example 71
  • US9796724, Example 71
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 72
  • US10758542, Example 72
  • US8791123, 72
  • US9782415, Example 72
  • US9796724, Example 72
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 73
  • US10758542, Example 73
  • US8791123, 73
  • US9782415, Example 73
  • US9796724, Example 73
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 74
  • US10758542, Example 74
  • US8791123, 74
  • US9782415, Example 74
  • US9796724, Example 74
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 75
  • US10758542, Example 75
  • US8791123, 75
  • US9782415, Example 75
  • US9796724, Example 75
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 76
  • US10758542, Example 76
  • US8791123, 76
  • US9782415, Example 76
  • US9796724, Example 76
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 77
  • US10758542, Example 77
  • US8791123, 77
  • US9782415, Example 77
  • US9796724, Example 77
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 78
  • US10758542, Example 78
  • US8791123, 78
  • US9782415, Example 78
  • US9796724, Example 78
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 85
  • US10758542, Example 85
  • US8791123, 85
  • US9782415, Example 85
  • US9796724, Example 85
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 86
  • US10758542, Example 86
  • US8791123, 86
  • US9782415, Example 86
  • US9796724, Example 86
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 87
  • US10758542, Example 87
  • US8791123, 87
  • US9782415, Example 87
  • US9796724, Example 87
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 88
  • US10758542, Example 88
  • US8791123, 88
  • US9782415, Example 88
  • US9796724, Example 88
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 89
  • US10758542, Example 89
  • US8791123, 89
  • US9782415, Example 89
  • US9796724, Example 89
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 90
  • US10758542, Example 90
  • US8791123, 90
  • US9782415, Example 90
  • US9796724, Example 90
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 92
  • US10758542, Example 92
  • US8791123, 92
  • US9782415, Example 92
  • US9796724, Example 92
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 94
  • US10758542, Example 94
  • US8791123, 94
  • US9782415, Example 94
  • US9796724, Example 94
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 95
  • US10758542, Example 95
  • US8791123, 95
  • US9782415, Example 95
  • US9796724, Example 95
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 96
  • US10758542, Example 96
  • US8791123, 96
  • US9782415, Example 96
  • US9796724, Example 96
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 97
  • US10758542, Example 97
  • US8791123, 97
  • US9782415, Example 97
  • US9796724, Example 97
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 102
  • US10758542, Example 102
  • US8791123, 102
  • US9782415, Example 102
  • US9796724, Example 102
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 103
  • US10758542, Example 103
  • US8791123, 103
  • US9782415, Example 103
  • US9796724, Example 103
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 104
  • US10758542, Example 104
  • US8791123, 104
  • US9782415, Example 104
  • US9796724, Example 104
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 105
  • US10758542, Example 105
  • US8791123, 105
  • US9782415, Example 105
  • US9796724, Example 105
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 107
  • US10758542, Example 107
  • US8791123, 107
  • US9782415, Example 107
  • US9796724, Example 107
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 108
  • US10758542, Example 108
  • US8791123, 108
  • US9782415, Example 108
  • US9796724, Example 108
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 109
  • US10758542, Example 109
  • US8791123, 109
  • US9782415, Example 109
  • US9796724, Example 109
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 110
  • US10758542, Example 110
  • US8791123, 110
  • US9782415, Example 110
  • US9796724, Example 110
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 111
  • US10758542, Example 111
  • US8791123, 111
  • US9782415, Example 111
  • US9796724, Example 111
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 112
  • US10758542, Example 112
  • US8791123, 112
  • US9782415, Example 112
  • US9796724, Example 112
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 113
  • US10758542, Example 113
  • US8791123, 113
  • US9782415, Example 113
  • US9796724, Example 113
10 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 115
  • US10758542, Example 115
  • US8791123, 115
  • US9782415, Example 115
  • US9796724, Example 115
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