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 11-beta-Hydroxysteroid Dehydrogenase 1 (11-beta-HSD1) [ 191 ] HIV-1 Protease Mutant (L10I/L90M) [ 9 ]
 11-beta-Hydroxysteroid Dehydrogenase 2 (11-beta-HSD2) [ 34 ] HIV-1 Protease Mutant (L23I) [ 1 ]
 15-Lipoxygenase [ 115 ] HIV-1 Protease Mutant (L23V) [ 1 ]
 17-beta-Hydroxysteroid Dehydrogenase 1 (17-beta-HSD1) [ 44 ] HIV-1 Protease Mutant (L24I) [ 3 ]
 17-beta-Hydroxysteroid Dehydrogenase 2 (17-beta-HSD2) [ 16 ] HIV-1 Protease Mutant (L76M) [ 1 ]
 17-beta-Hydroxysteroid Dehydrogenase 5 (17-beta-HSD5, AKR1C3) [ 6 ] HIV-1 Protease Mutant (L90M) [ 2 ]
 20-alpha-Hydroxysteroid Dehydrogenase (AKR1C1) [ 1 ] HIV-1 Protease Mutant (M36I) [ 5 ]
 20-alpha-Hydroxysteroid Dehydrogenase (AKR1C1) Mutant (H222S) [ 1 ] HIV-1 Protease Mutant (M36I/A71V) [ 5 ]
 20-alpha-Hydroxysteroid Dehydrogenase (AKR1C1) Mutant (L306A) [ 1 ] HIV-1 Protease Mutant (M46I,L63P,A71V,V82F,I84V) [ 6 ]
 20-alpha-Hydroxysteroid Dehydrogenase (AKR1C1) Mutant (L308A) [ 1 ] HIV-1 Protease Mutant (M46I/I54V) [ 9 ]
 20-alpha-Hydroxysteroid Dehydrogenase (AKR1C1) Mutant (L54V) [ 1 ] HIV-1 Protease Mutant (V32I) [ 1 ]
 2C-methyl-D-erythritol-2,4-cyclodiphosphate synthase (IspF) [ 9 ] HIV-1 Protease Mutant (V82A) [ 5 ]
 3-alpha-Hydroxysteroid Dehydrogenase Type 1 (AKR1C4) [ 1 ] HIV-1 Protease Mutant (V82A/I84V) [ 9 ]
 3-alpha-Hydroxysteroid Dehydrogenase Type 3 (AKR1C2) [ 1 ] HIV-1 Protease Mutant (V82F/I84V) [ 4 ]
 3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) [ 133 ] HIV-1 Protease Mutant (V82I) [ 1 ]
 3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (A162V) [ 2 ] HIV-1 Protease Mutant K-60C [ 14 ]
 3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (E166D) [ 2 ] HIV-1 Protease Mutant M1 (L10I, G48V, I54V, L63P, V82A) [ 19 ]
 3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (L159M) [ 2 ] HIV-1 Protease Mutant M2 (D30N, L63P, N88D) [ 19 ]
 3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (T222A) [ 2 ] HIV-1 Protease Mutant M3 (L10I, L63P, A71V, G73S, I84V, L90M) [ 19 ]
 3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (V143T) [ 2 ] HIV-1 Protease Mutant Q-60C [ 10 ]
 3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (V143T/T222A) [ 2 ] HIV-1 Protease Mutant V-18C [ 25 ]
 5-Lipoxygenase [ 101 ] HIV-1 Protease Mutant V6 [ 4 ]
 Ab N1G9 [ 1 ] HIV-1 Protease Mutant V6(46) [ 4 ]
 Abhydrolase Domain-Containing Protein 6 [ 1 ] HIV-1 Protease Mutant V6(46/54/84) [ 4 ]
 ABL [ 51 ] HIV-1 Protease Mutant V6(46/84) [ 4 ]
 ABL Mutant (E255K) [ 7 ] HIV-1 Protease Mutant V6(54) [ 4 ]
 ABL Mutant (F359V) [ 7 ] HIV-1 Protease Mutant V6(54/84) [ 4 ]
 ABL Mutant (H396P) [ 7 ] HIV-1 Protease Mutant V6(84) [ 4 ]
 ABL Mutant (M351T) [ 7 ] HIV-1 Protease Mutant, A-1 [ 4 ]
 ABL Mutant (Q252H) [ 7 ] HIV-1 Protease Mutant, ANAM-11 [ 4 ]
 ABL Mutant (T315I) [ 26 ] HIV-1 Protease Mutant, MDR-HM [ 9 ]
 ABL Mutant (T315N) [ 7 ] HIV-1 Protease Mutant, MDR-QM [ 9 ]
 ABL Mutant (Y253F) [ 7 ] HIV-1 Protease Mutant, NAM-10 [ 4 ]
 Acetate Operon Repressor (C-IclR) [ 2 ] HIV-1 Reverse Transcriptase [ 1437 ]
 Acetate Operon Repressor (IclR) [ 2 ] HIV-1 Reverse Transcriptase Mutant (103N/181C) [ 36 ]
 Acetylcholinesterase (AChE) [ 836 ] HIV-1 Reverse Transcriptase Mutant (G190A) [ 9 ]
 Activated Protein C (APC) [ 1 ] HIV-1 Reverse Transcriptase Mutant (K103N) [ 92 ]
 Acyl Cholesterol Acyltransferase 1 (ACAT-1) [ 7 ] HIV-1 Reverse Transcriptase Mutant (K103N/Y181C) [ 11 ]
 ADAMTS-4 (Aggrecanase-1) [ 30 ] HIV-1 Reverse Transcriptase Mutant (L100I) [ 58 ]
 ADAMTS-5 (Aggrecanase-2) [ 65 ] HIV-1 Reverse Transcriptase Mutant (L100I/K103N) [ 3 ]
 Adenosine A3 Receptor [ 29 ] HIV-1 Reverse Transcriptase Mutant (P236L) [ 52 ]
 Adenosine Deaminase [ 56 ] HIV-1 Reverse Transcriptase Mutant (V106A) [ 12 ]
 Adenosine Kinase (AK) [ 8 ] HIV-1 Reverse Transcriptase Mutant (V179D) [ 5 ]
 Adenosine Phosphosulfate Reductase (APSR) [ 10 ] HIV-1 Reverse Transcriptase Mutant (Y181C) [ 317 ]
 Adenosine Receptor A1 [ 171 ] HIV-1 Reverse Transcriptase Mutant (Y181I) [ 5 ]
 Adenosine Receptor A2A [ 165 ] HIV-1 Reverse Transcriptase Mutant (Y188L) [ 60 ]
 Adenosine Receptor A2B [ 7 ] HIV-1 Reverse Transcriptase RNase H [ 374 ]
 Adenosine Receptor A3 [ 7 ] HIV-1 Reverse Transcriptase RNase H Mutant (D67N/K70R/T215F/K219Q) [ 2 ]
 AICAR Tfase [ 19 ] HIV-1 Reverse Transcriptase RNase H Mutant (L100I/K103N) [ 2 ]
 Aldehyde Reductase (ALR1) [ 40 ] HIV-1 Reverse Transcriptase RNase H Mutant (V106A/Y181C) [ 2 ]
 Aldose Reductase (ALR2) [ 145 ] HIV-1 Reverse Transcriptase RNase H Mutant (Y181C) [ 2 ]
 Aldose Reductase (ALR2) Mutant (C298A) [ 2 ] HIV-1 Reverse Transcriptase RNase H Mutant (Y188L) [ 2 ]
 Aldose Reductase (ALR2) Mutant (C298A/W219Y) [ 12 ] HIV-2 Protease [ 22 ]
 Aldose Reductase (ALR2) Mutant (L300P) [ 2 ] HIV-2 Reverse Transcriptase [ 3 ]
 Aldosterone Synthase (CYP11B2) [ 108 ] HIV-2 Reverse Transcriptase RNase H [ 2 ]
 Alpha-1 Adrenergic Receptor [ 12 ] HMG-CoA Reductase [ 126 ]
 alpha-Amylase [ 20 ] Homoisocitrate Dehydrogenase (HICDH) [ 8 ]
 alpha-Carbonic Anhydrase [ 17 ] I-kappa-B Kinase 1 (IKK-alpha) [ 142 ]
 alpha-Chymotrypsin [ 1 ] I-kappa-B Kinase 2 (IKK-beta) [ 173 ]
 alpha-Glucosidase (alpha-Glu) [ 34 ] I-kappa-B Kinase 3 (IKK-epsilon) [ 40 ]
 alpha-Methylacyl-CoA Racemase [ 10 ] Immunophilin FKBP12 [ 79 ]
 Alpha2 Adrenoreceptor [ 4 ] IMP Cyclohydrolase (IMPCH) [ 3 ]
 Aminopeptidase M [ 46 ] Indoleamine 2,3-Dioxygenase [ 108 ]
 Androgen Receptor (AR) [ 307 ] Inosine Monophosphate Dehydrogenase Type 1 (IMPDH1) [ 14 ]
 Angiotensin-Converting Enzyme [ 39 ] Inosine Monophosphate Dehydrogenase Type 2 (IMPDH2) [ 39 ]
 Angiotensin-Converting Enzyme 2 [ 36 ] Insulin Receptor Tyrosine Kinase (IRK) [ 94 ]
 Anthrax Lethal Factor (LF) [ 240 ] Insulin Receptor-Related Protein (INSRR) [ 6 ]
 apocytochrome b562 [ 1 ] Insulin-like Growth Factor 1 Receptor (IGF-1R) [ 177 ]
 apocytochrome b562(denatured) [ 1 ] Integrin alpha1beta1 [ 5 ]
 Apoptosis Regulator Bcl-2 [ 62 ] Integrin alpha2beta1 [ 28 ]
 Apoptosis Regulator Bcl-xL [ 209 ] Integrin alpha4beta1 (VLA-4) [ 246 ]
 Apurinic-Apyrimidinic Endonuclease 1 (APE1) [ 47 ] Integrin alpha4beta7 [ 71 ]
 Aromatase (CYP19) [ 397 ] Integrin alpha5beta1 [ 5 ]
 Aryl Hydrocarbon Receptor (AhR) [ 25 ] Kallikrein [ 54 ]
 Asparaginyl Endopeptidase (AE) [ 31 ] Kappa Opioid Receptor [ 94 ]
 ATP Phosphoribosyltransferase [ 11 ] KIAA1363 [ 1 ]
 ATP-Binding Cassette Transporter ABCG2 [ 21 ] Kinesin Spindle Protein Eg5 [ 198 ]
 Aurora Kinase A (Aurora-A) [ 332 ] KIT(D816V) [ 23 ]
 Aurora Kinase B (Aurora-B) [ 97 ] KIT(V559D T670I) [ 18 ]
 Aurora Kinase C (Aurora-C) [ 19 ] Kynurenine Aminotransferase 1/Glutamine Transaminase K [ 2 ]
 AXL Receptor Tyrosine Kinase [ 16 ] Lactate Dehydrogenase [ 34 ]
 B-Raf Protein Kinase [ 71 ] Lck [ 232 ]
 B-Raf Protein Kinase Mutant (V599E) [ 1 ] Leucine Aminopeptidase [ 19 ]
 B-Raf Protein Kinase Mutant (V600E) [ 144 ] Leukotriene A4 Hydrolase [ 117 ]
 Bacterial Leucyl Aminopeptidase [ 19 ] Lipoxygenase-1 [ 8 ]
 Bacteriophage T4 DNA Ligase [ 6 ] Liver Receptor Homolog 1 [ 23 ]
 Beta-1 Adrenergic Receptor [ 25 ] Liver X Receptor alpha (LXR-alpha) [ 199 ]
 Beta-2 Adrenergic Receptor [ 38 ] Liver X Receptor beta (LXR-beta) [ 251 ]
 Beta-3 Adrenergic Receptor [ 25 ] Major Urinary Protein (MUP-1) [ 8 ]
 beta-Carbonic Anhydrase [ 37 ] Malate Dehydrogenase (pfMDH) [ 8 ]
 beta-Hydroxyacyl-Acyl Carrier Protein Dehydratase (FabZ) [ 53 ] Malate Dehydrogenase, cytoplasmic [ 7 ]
 beta-Ketoacyl-ACP Synthase III (FabH) [ 46 ] Malate Dehydrogenase, mitochondrial [ 9 ]
 beta-Secretase (BACE-1) [ 398 ] Mammalian Target of Rapamycin (mTOR) [ 91 ]
 beta-Secretase (BACE-2) [ 107 ] MAP Kinase Kinase 1 (MEK1) [ 1 ]
 Bfl-1 [ 206 ] MAP Kinase p38 alpha [ 482 ]
 Bfl-1  [ 44 ] MAP Kinase p38 alpha Mutant (G110A) [ 6 ]
 Biotin Carboxylase [ 14 ] MAP Kinase p38 alpha Mutant (G110D) [ 6 ]
 BirA Bifunctional Protein [ 4 ] MAP Kinase p38 beta [ 15 ]
 BirA Bifunctional Protein Mutant (V214A) [ 3 ] MAP Kinase-Interacting Protein Kinase (MNK1) [ 4 ]
 BirA Bifunctional Protein Mutant (V219A) [ 3 ] MAP-Microtubule Affinity-Regulating Kinase 3 (MARK3) [ 1 ]
 BirA Bifunctional Protein Mutant (W223A) [ 3 ] MAP4K4 (HGK) [ 1 ]
 Bone Morphogenetic Protein Receptor type II (BMPR2) [ 6 ] MAPK-Activated Protein Kinase 2 (MK2) [ 150 ]
 Botulinum Neurotoxin Type A [ 128 ] MAPK-Activated Protein Kinase 3 (MK3) [ 4 ]
 Butyrylcholinesterase (BuChE) [ 579 ] MAPK-Activated Protein Kinase 5 (MK5) [ 4 ]
 C-Raf Protein Kinase [ 34 ] Matriptase [ 68 ]
 Calcium-Sensing Receptor (CaSR) [ 44 ] Matrix Metalloproteinase-1 (MMP-1) [ 188 ]
 Calpain-1 [ 21 ] Matrix Metalloproteinase-10 (MMP-10) [ 4 ]
 Calpain-2 [ 10 ] Matrix Metalloproteinase-12 (MMP-12) [ 68 ]
 CaM Kinase II [ 42 ] Matrix Metalloproteinase-13 (MMP-13) [ 212 ]
 cAMP-Dependent Protein Kinase (PKA) [ 422 ] Matrix Metalloproteinase-14 (MMP-14) [ 11 ]
 cAMP-Dependent Protein Kinase (PKA) Mutant PKAR1 (1) [ 5 ] Matrix Metalloproteinase-2 (MMP-2) [ 220 ]
 cAMP-Dependent Protein Kinase (PKA) Mutant PKAR1 (2) [ 5 ] Matrix Metalloproteinase-3 (MMP-3) [ 109 ]
 cAMP-Dependent Protein Kinase (PKA) Mutant PKAR1 (3) [ 5 ] Matrix Metalloproteinase-7 (MMP-7) [ 27 ]
 cAMP-Dependent Protein Kinase (PKA) Mutant PKAR1 (4) [ 5 ] Matrix Metalloproteinase-8 (MMP-8) [ 120 ]
 cAMP-Dependent Protein Kinase (PKA) Mutant PKAR2 (1) [ 5 ] Matrix Metalloproteinase-9 (MMP-9) [ 161 ]
 cAMP-Dependent Protein Kinase (PKA) Mutant PKAR2 (2) [ 1 ] Mcl-1 [ 10 ]
 cAMP-Dependent Protein Kinase (PKA) Mutant PKAR2 (3) [ 3 ] MEK Kinase 1 (MEKK1) [ 1 ]
 cAMP-Dependent Protein Kinase (PKA) Mutant PKAR3 [ 5 ] Melanin-Concentrating Hormone Receptor 1 (MCH1R) [ 21 ]
 cAMP-Dependent Protein Kinase (PKA) Mutant PKAR3 (1) [ 5 ] Methionine Aminopeptidase (MAP) [ 20 ]
 cAMP-Dependent Protein Kinase (PKA) Mutant PKAR4 [ 5 ] Methionine Aminopeptidase Type 1 (MetAP1) [ 14 ]
 cAMP-Dependent Protein Kinase (PKA) Mutant PKAR5 [ 5 ] Methionine Aminopeptidase Type 2 (MetAP2) [ 286 ]
 Cannabinoid Receptor 1 [ 160 ] Methylthioadenosine Nucleosidase(MTAN) [ 3 ]
 Cannabinoid Receptor 2 [ 130 ] Methylthioadenosine Phosphorylase (MTAP) [ 3 ]
 Carbonic Anhydrase (hpCA) [ 47 ] Mineralocorticoid Receptor (MR) [ 22 ]
 Carbonic Anhydrase (mtCA 1) [ 37 ] Mitogen- and Stress-Activated Protein Kinase 1 (MSK1) [ 15 ]
 Carbonic Anhydrase (mtCA 3) [ 37 ] Mitogen- and Stress-Activated Protein Kinase 2 (MSK2) [ 4 ]
 Carbonic Anhydrase 2 (Can2) [ 37 ] Mitogen-Activated Protein Kinase 1 [ 4 ]
 Carbonic Anhydrase I [ 393 ] Mitogen-Activated Protein Kinase 10 (JNK3) [ 94 ]
 Carbonic Anhydrase II [ 476 ] Mitogen-Activated Protein Kinase 8 (JNK1) [ 269 ]
 Carbonic Anhydrase II Mutant (F131V) [ 11 ] Mitogen-Activated Protein Kinase 9 (JNK2) [ 75 ]
 Carbonic Anhydrase III [ 47 ] Mitogen-Activated Protein Kinase 9 (JNK2) Mutant (C162S) [ 1 ]
 Carbonic Anhydrase IV [ 241 ] Mitogen-Activated Protein Kinase 9 (JNK2) Mutant (R127A) [ 1 ]
 Carbonic Anhydrase IX [ 233 ] Mixed Lineage Kinase 1 (MLK1) [ 36 ]
 Carbonic Anhydrase VA [ 129 ] Mixed Lineage Kinase 2 (MLK2) [ 8 ]
 Carbonic Anhydrase VB [ 94 ] Mixed Lineage Kinase 3 (MLK3) [ 36 ]
 Carbonic Anhydrase VI [ 78 ] MKP-3 [ 45 ]
 Carbonic Anhydrase VII [ 49 ] ML-IAP-BIR [ 32 ]
 Carbonic Anhydrase XII [ 63 ] Monoamine Oxidase Type A (MAO-A) [ 245 ]
 Carbonic Anhydrase XIII [ 48 ] Monoamine Oxidase Type B (MAO-B) [ 244 ]
 Carbonic Anhydrase XIV [ 50 ] Monoamine oxidase type B (MAO-B) Mutant (I199F) [ 5 ]
 Carbonic Anhydrase XV [ 73 ] Monocarboxylate Transporter 1 [ 42 ]
 Carboxylesterase 1 [ 143 ] Monoglyceride Lipase (MGL) [ 22 ]
 Carboxylesterase 2 (intestine, liver) [ 143 ] MPI protein  [ 462 ]
 Carboxypeptidase A (CPA) [ 15 ] MRCK alpha [ 5 ]
 Casein Kinase I [ 12 ] Mu Opioid Receptor [ 159 ]
 Casein Kinase II [ 41 ] MurD [ 37 ]
 Caspase-1 [ 135 ] Myosin Light-Chain Kinase [ 18 ]
 Caspase-2 [ 24 ] NAD-Dependent Deacetylase Sirtuin-1 [ 21 ]
 Caspase-3 [ 374 ] NAD-Dependent Deacetylase Sirtuin-2 [ 20 ]
 Caspase-3|IST-1 Complex [ 1 ] Neuraminidase A [ 246 ]
 Caspase-4 [ 17 ] Neuraminidase B [ 176 ]
 Caspase-5 [ 9 ] Neutral Endopeptidase [ 29 ]
 Caspase-6 [ 71 ] Neutrophil Elastase (NE) [ 56 ]
 Caspase-7 [ 123 ] Niacin Receptor GPR109A [ 18 ]
 Caspase-8 [ 124 ] Nitric Oxide Synthase, brain [ 49 ]
 Caspase-9 [ 8 ] Nitric Oxide Synthase, brain Mutant (D597N) [ 3 ]
 Cathepsin B [ 171 ] Nitric Oxide Synthase, brain Mutant (D597N/M336V) [ 4 ]
 Cathepsin B  [ 56 ] Nitric Oxide Synthase, endothelial [ 51 ]
 Cathepsin B-Like Cysteine Protease (TbcatB) [ 56 ] Nitric Oxide Synthase, endothelial Mutant (N368D) [ 3 ]
 Cathepsin D [ 277 ] Nitric Oxide Synthase, inducible [ 55 ]
 Cathepsin K [ 488 ] NK1 Receptor [ 15 ]
 Cathepsin L [ 436 ] Nociceptin Receptor (ORL1 Receptor) [ 168 ]
 Cathepsin L2 [ 24 ] Norepinephrine Transporter (NET) [ 56 ]
 Cathepsin S [ 458 ] Orotidine Monophosphate Decarboxylase (ODCase) [ 9 ]
 Cathepsin V [ 2 ] Outer Membrane Phospholipase A [ 1 ]
 Cdc7 Kinase [ 99 ] Outer Membrane Phospholipase A (sulfonylated) [ 1 ]
 Cell Division Cycle 2-Like 1(CDC2L1) [ 7 ] p53-Binding Protein HDMX [ 25 ]
 Cell Division Cycle 2-Like 2 (CDC2L2) [ 7 ] p53-Binding Protein MDM2 [ 170 ]
 Cell Division Cycle 2-Like 6 (CDK11) [ 11 ] Papain [ 48 ]
 cGMP-Dependent Protein Kinase [ 23 ] PDGFR-beta [ 626 ]
 Checkpoint Kinase (Chk1) [ 198 ] Pepsin [ 26 ]
 Checkpoint Kinase (Chk2) [ 14 ] Peptide Deformylase [ 3 ]
 Chicken erythrocyte chromatin [ 2 ] Peripheral-Type Benzodiazepine Receptor [ 10 ]
 Chitinase [ 5 ] Peroxisome Proliferator-Activated Receptor alpha [ 265 ]
 Chitinase Mutant (A217G) [ 3 ] Peroxisome Proliferator-Activated Receptor delta [ 224 ]
 Chitinase Mutant (D175A) [ 3 ] Peroxisome Proliferator-Activated Receptor gamma [ 258 ]
 Chitinase Mutant (D246A) [ 1 ] Phenylethanolamine N-Methyltransferase (PNMT) [ 29 ]
 Chitinase Mutant (E177A) [ 1 ] Phosphodiesterase Type 1 (PDE1B) [ 10 ]
 Chitinase Mutant (E322A) [ 3 ] Phosphodiesterase Type 10 (PDE10A) [ 59 ]
 Chitinase Mutant (M243A) [ 3 ] Phosphodiesterase Type 11 (PDE11A) [ 10 ]
 Chitinase Mutant (R301K) [ 3 ] Phosphodiesterase Type 2 (PDE2A) [ 10 ]
 Chitinase Mutant (T138A) [ 3 ] Phosphodiesterase Type 3 (PDE3A) [ 69 ]
 Chitinase Mutant (Y245F) [ 2 ] Phosphodiesterase Type 3 (PDE3B) [ 80 ]
 Cholecystokinin-1 Receptor [ 17 ] Phosphodiesterase Type 4 (PDE4A) [ 142 ]
 Cholecystokinin-2 Receptor [ 17 ] Phosphodiesterase Type 4 (PDE4B) [ 80 ]
 Chymase [ 1 ] Phosphodiesterase Type 4 (PDE4C) [ 2 ]
 Chymotrypsin [ 28 ] Phosphodiesterase Type 4 (PDE4D) [ 79 ]
 cIAP-1 BIR3 [ 10 ] Phosphodiesterase Type 5 (PDE5) [ 26 ]
 cIAP-2 BIR3 [ 10 ] Phosphodiesterase Type 5 (PDE5A) [ 12 ]
 cIAP1-BIR3 [ 5 ] Phosphodiesterase Type 5 (PDE5A) Mutant (661-681 deletion) [ 3 ]
 cIAP2-BIR3 [ 3 ] Phosphodiesterase Type 5 (PDE5A) Mutant (663-678 deletion) [ 3 ]
 CLK1 [ 16 ] Phosphodiesterase Type 6 (PDE6) [ 7 ]
 CLK4 [ 13 ] Phosphodiesterase Type 7 (PDE7B) [ 10 ]
 Collagenase (ChC) [ 184 ] Phosphodiesterase Type 8 (PDE8A) [ 10 ]
 Conantokin-G [ 3 ] Phosphodiesterase Type 9 (PDE9A) [ 10 ]
 Conantokin-T [ 3 ] Phosphoinositide 3-Kinase (PI3K), alpha [ 133 ]
 Corticotropin-releasing Factor Receptor 1 [ 134 ] Phosphoinositide 3-Kinase (PI3K), alpha Mutant (E545K) [ 1 ]
 cPLA2 C2 [ 1 ] Phosphoinositide 3-Kinase (PI3K), alpha Mutant (H1047R) [ 1 ]
 Cyclin-Dependent Kinase 1 (CDK1) [ 953 ] Phosphoinositide 3-Kinase (PI3K), beta [ 11 ]
 Cyclin-Dependent Kinase 2 (CDK2) [ 1652 ] Phosphoinositide 3-Kinase (PI3K), C2beta [ 6 ]
 Cyclin-Dependent Kinase 2 (CDK2) Mutant (F82H) [ 1 ] Phosphoinositide 3-Kinase (PI3K), delta [ 7 ]
 Cyclin-Dependent Kinase 2 (CDK2) Mutant (F82H/L83V/H84D) [ 2 ] Phosphoinositide 3-Kinase (PI3K), gamma [ 66 ]
 Cyclin-Dependent Kinase 2 (CDK2) Mutant (F82H/L83V/H84D/K89T) [ 2 ] Phosphoinositide 3-Kinase (PI3K), Vps34 [ 1 ]
 Cyclin-Dependent Kinase 2 (CDK2) Mutant (K89T) [ 2 ] Phospholipase A2, major isoenzyme [ 21 ]
 Cyclin-Dependent Kinase 2 (CDK2) Mutant (L83V/H84D) [ 1 ] Phospholipase A2, membrane associated [ 32 ]
 Cyclin-Dependent Kinase 4 (CDK4) [ 957 ] Phosphorylase Kinase [ 13 ]
 Cyclin-Dependent Kinase 5 (CDK5) [ 298 ] PIM-1 Kinase [ 179 ]
 Cyclin-Dependent Kinase 6 (CDK6) [ 8 ] PIM-2 Kinase [ 142 ]
 Cyclin-Dependent Kinase 7 (CDK7) [ 41 ] PIM-3 Kinase [ 2 ]
 Cyclin-Dependent Kinase 8 (CDK8) [ 8 ] Plasma Kallikrein [ 4 ]
 Cyclin-Dependent Kinase 9 (CDK9) [ 19 ] Plasmepsin I [ 92 ]
 Cyclooxygenase-1 [ 71 ] Plasmepsin II [ 107 ]
 Cyclooxygenase-2 [ 69 ] Plasmepsin IV [ 11 ]
 Cytochrome P450 1A2 [ 1 ] Plasmin [ 140 ]
 Cytochrome P450 2A6 [ 31 ] PLD alpha C2 [ 1 ]
 Cytochrome P450 2B4 [ 2 ] PLD beta C2 [ 1 ]
 Cytochrome P450 2B4 Mutant (F206A) [ 2 ] Polo-Like Kinase 1 [ 136 ]
 Cytochrome P450 2C19 [ 8 ] Polo-Like Kinase 2 [ 29 ]
 Cytochrome P450 2C9 [ 29 ] Polo-Like Kinase 3 [ 45 ]
 Cytochrome P450 2D6 [ 8 ] Polo-Like Kinase 4 [ 21 ]
 Cytochrome P450 2E1 [ 9 ] Poly (ADP-ribose) Polymerase-1 (PARP-1) [ 216 ]
 Cytochrome P450 3A1 [ 11 ] Poly (ADP-ribose) Polymerase-2 (PARP-2) [ 35 ]
 Cytochrome P450 3A4 [ 91 ] PPIase Pin1 [ 15 ]
 Cytochrome P450 51(CYP51) [ 25 ] Pregnane X Receptor [ 12 ]
 Cytochrome P450 51(CYP51) Mutant (F78L) [ 2 ] Progesterone Receptor (PR) [ 73 ]
 Cytochrome P450 Reductase (CPR) [ 4 ] Prokineticin Receptor 1 (PKR1) [ 3 ]
 D-Amino Acid Oxidase (DAAO) [ 47 ] Prokineticin Receptor 2 (PKR2) [ 3 ]
 D-Aspartate Oxidase (DDO) [ 23 ] Prostacyclin (IP) Receptor [ 17 ]
 Delta Opioid Receptor [ 139 ] Prostaglandin D Synthase [ 16 ]
 Dengue Virus 1 (DENV1) NS2B-NS3 Protease [ 10 ] Prostaglandin D2 Receptor CRTH2 [ 69 ]
 Dengue Virus 2 (DENV2) NS2B-NS3 Protease [ 15 ] Prostanoid EP1 Receptor [ 19 ]
 Dengue Virus 3 (DENV3) NS2B-NS3 Protease [ 10 ] Prostanoid EP2 Receptor [ 19 ]
 Dengue Virus 4 (DENV4) NS2B-NS3 Protease [ 10 ] Prostanoid EP3 Receptor [ 19 ]
 Diacyl Glycerolacyltransferase 1 (DGAT-1) [ 21 ] Prostanoid EP4 Receptor [ 19 ]
 Diacyl Glycerolacyltransferase 2 (DGAT-2) [ 2 ] Protein Farnesyltransferase (PFT) [ 203 ]
 Dihydrofolate Reductase (DHFR) [ 202 ] Protein kinase B (Akt 1) [ 461 ]
 Dihydrofolate Reductase (DHFR) Mutant (F98Y) [ 2 ] Protein kinase B (Akt 2) [ 157 ]
 Dihydrofolate Reductase (DHFR) Mutant (I100L) [ 2 ] Protein kinase B (Akt 3) [ 68 ]
 Dihydrofolate Reductase-Thymidylate Synthase (DHFR-TS) [ 21 ] Protein Kinase C [ 153 ]
 Dihydrofolate Reductase-Thymidylate Synthase (DHFR-TS) Mutant KICB1 [ 3 ] Protein Kinase C, alpha [ 132 ]
 Dihydrofolate Reductase-Thymidylate Synthase (DHFR-TS) Mutant SP21 [ 19 ] Protein Kinase C, beta I [ 48 ]
 Dihydrofolate Reductase-Thymidylate Synthase (DHFR-TS) Mutant V1/S [ 3 ] Protein Kinase C, beta II [ 87 ]
 Dihydroorotate Dehydrogenase (DHODH) [ 132 ] Protein Kinase C, delta [ 109 ]
 Dihydroorotate Dehydrogenase (DHODH) Mutant (H185A) [ 13 ] Protein Kinase C, epsilon [ 93 ]
 Dihydroorotate Dehydrogenase (DHODH) Mutant (R265A) [ 13 ] Protein Kinase C, eta [ 61 ]
 Dipeptidyl Peptidase II (DPP-II) (QPP) [ 51 ] Protein Kinase C, gamma [ 44 ]
 Dipeptidyl Peptidase IV (DPP-IV) [ 721 ] Protein Kinase C, theta [ 91 ]
 Dipeptidyl Peptidase VII (DPP-VII) (QPP) [ 321 ] Protein Kinase C, zeta [ 44 ]
 DNA Gyrase [ 30 ] Protein Kinase D1  [ 30 ]
 DNA Ligase (MtuLigA) [ 6 ] Protein Kinase YpkA [ 4 ]
 DNA Ligase I [ 4 ] Protein Tyrosine Phosphatase CD45 [ 1 ]
 DNA Polymerase alpha [ 12 ] Protein Tyrosine Phosphatase LAR [ 1 ]
 DNA Polymerase beta [ 10 ] Protein Tyrosine Phosphatase PTPA [ 1 ]
 DNA Polymerase gamma [ 2 ] Protein Tyrosine Phosphatase PTPB [ 5 ]
 DNA polymerase IIIC [ 2 ] Protein Tyrosine Phosphatase TC-PTP [ 1 ]
 DNA polymerase IIIE [ 2 ] Protein Tyrosine Phosphatase VHR [ 1 ]
 DNA Topoisomerase IV [ 27 ] Protein-Tyrosine Phosphatase 1B (PTP1B) [ 280 ]
 DNA(calf thymus) [ 2 ] Protein-Tyrosine Phosphatase 1B (PTP1B) Mutant (G117E) [ 1 ]
 Dopamine Receptor D2 [ 39 ] Protein-Tyrosine Phosphatase 1B (PTP1B) Mutant (L119V) [ 2 ]
 Dopamine Transporter (DAT) [ 64 ] Protein-Tyrosine Phosphatase 1B (PTP1B) Mutant (M114V) [ 1 ]
 DPP8 [ 389 ] Protein-Tyrosine Phosphatase 1B (PTP1B) Mutant (V113I) [ 1 ]
 DPP9 [ 273 ] Protein-Tyrosine Phosphatase 1B (PTP1B) Mutant (V113L/M114V) [ 1 ]
 Dual Specificity Protein Phosphatase 1 [ 164 ] Protein-Tyrosine Phosphatase SHP-1 [ 22 ]
 DYRK1A [ 3 ] Protein-Tyrosine Phosphatase SHP-2 [ 51 ]
 EGF-R Tyrosine Kinase [ 1076 ] Pteridine Reductase 1 (PTR1) [ 11 ]
 EGF-R Tyrosine Kinase Mutant (G719C) [ 20 ] Purine Nucleoside Phosphorylase (PNP) [ 6 ]
 EGF-R Tyrosine Kinase Mutant (G719S) [ 2 ] Quinone Reductase 1 [ 29 ]
 EGF-R Tyrosine Kinase Mutant (L858R) [ 2 ] Quinone Reductase 2 (QR2) [ 25 ]
 EGF-R Tyrosine Kinase Mutant (L858R/T790M) [ 2 ] RAF-1 [ 1 ]
 EGF-R Tyrosine Kinase Mutant (T790M) [ 6 ] Receptor Tyrosine Kinase TrkA [ 44 ]
 Endothelin-Converting Enzyme 1 [ 29 ] Receptor Tyrosine Kinase TrkB [ 2 ]
 Enoyl-ACP Reductase (FabI) [ 83 ] Renin [ 225 ]
 Enoyl-ACP Reductase (FabI) Mutant (F203L) [ 3 ] Retinoic Acid Receptor, alpha [ 10 ]
 Enoyl-ACP Reductase (FabK) [ 5 ] Retinoic Acid Receptor, beta [ 10 ]
 Enoyl-ACP Reductase (InhA) [ 108 ] Retinoic Acid Receptor, gamma [ 10 ]
 Enoyl-ACP Reductase (PfENR) [ 28 ] Rho Transcription Termination Factor [ 2 ]
 Epoxide Hydrolase B (EHB) [ 20 ] Rho-kinase (ROCK I) [ 70 ]
 Equilibrative Nucleoside Transporter 1 (ENT1) [ 80 ] Rho-kinase (ROCK II) [ 20 ]
 ErbB-2 (HER2) Tyrosine Kinase [ 142 ] Ribonuclease H [ 2 ]
 ErbB-4 (HER4) Tyrosine Kinase [ 9 ] Ribonuclease H1 [ 8 ]
 ERK-2 [ 72 ] Ribosomal S6 Kinase 1 (RSK-1) [ 9 ]
 ERK-8 [ 9 ] Ribosomal S6 Kinase 2 (RSK-2) [ 1 ]
 Estrogen Receptor (ER-alpha) [ 208 ] Ribosomal S6 Kinase 3 (RSK-3) [ 1 ]
 Estrogen Receptor (ER-beta) [ 169 ] Ribosomal S6 Kinase 4 (RSK-4) [ 1 ]
 Estrogen-Related Receptor, alpha [ 2 ] RNA(23-mer) [ 1 ]
 Estrogen-Related Receptor, alpha Mutant (C325S) [ 1 ] Runt-Related Transcription Factor 1 Isoform AML1C [ 115 ]
 Estrogen-Related Receptor, gamma [ 29 ] Runt-Related Transcription Factor 1 Isoform AML1C  [ 101 ]
 Factor IXa (fIXa) [ 90 ] S-Adenosylmethionine Decarboxylase (AdoMetDC) [ 34 ]
 Factor VIIa (fVIIa) [ 323 ] Sarco/endoplasmic Reticulum Ca2+ ATPase 1 [ 30 ]
 Factor Xa (fXa) [ 1172 ] SARS Coronavirus 3C-like Protease [ 84 ]
 Factor XIa (fXIa) [ 413 ] SARS Coronavirus Coronavirus Papain-Like Protease [ 24 ]
 Factor XIIa (fXIIa) [ 123 ] Serine Hydroxymethyltransferase [ 5 ]
 FAD-Binding Domain [ 1 ] Serotonin Receptor 1A [ 157 ]
 Falcipain-2 [ 30 ] Serotonin Receptor 1A  [ 346 ]
 Farnesoid X-Activated Receptor [ 54 ] Serotonin Receptor 1B [ 3 ]
 Farnesyl Diphosphate Synthase (FPPS) [ 6 ] Serotonin Receptor 1D [ 3 ]
 Fatty Acid Amide Hydrolase [ 236 ] Serotonin Receptor 1E [ 126 ]
 Fatty Acid Synthase [ 46 ] Serotonin Receptor 2A [ 58 ]
 FGFR-1 Tyrosine Kinase [ 534 ] Serotonin Receptor 2B [ 5 ]
 FGFR-2 Tyrosine Kinase [ 9 ] Serotonin Receptor 2C [ 5 ]
 Fibroblast Activation Protein (FAP) [ 18 ] Serotonin Receptor 4 [ 8 ]
 Formyl Peptide Receptor-Like 1 [ 18 ] Serotonin Receptor 6 [ 107 ]
 G-protein Coupled Receptor 40 [ 52 ] Serotonin Receptor 7 [ 64 ]
 G-protein Coupled Receptor 54 [ 12 ] Serotonin Transporter (SERT) [ 71 ]
 GABAA Receptor Mutant, alpha-1 (A160C), beta-2, gamma-2 [ 3 ] Sodium-Dependent Glucose Cotransporter 1 (SGLT1) [ 5 ]
 GABAA Receptor Mutant, alpha-1 (D97C), beta-2, gamma-2 [ 1 ] Sodium-Dependent Glucose Cotransporter 2 (SGLT2) [ 5 ]
 GABAA Receptor Mutant, alpha-1 (F99C), beta-2, gamma-2 [ 3 ] Sortase A (SrtA) [ 85 ]
 GABAA Receptor Mutant, alpha-1 (G157C), beta-2, gamma-2 [ 3 ] Sphingosine 1-Phosphate Receptor 1 [ 32 ]
 GABAA Receptor Mutant, alpha-1 (G200C), beta-2, gamma-2 [ 3 ] Sphingosine 1-Phosphate Receptor 2 [ 4 ]
 GABAA Receptor Mutant, alpha-1 (S204C), beta-2, gamma-2 [ 3 ] Sphingosine 1-Phosphate Receptor 3 [ 32 ]
 GABAA Receptor Mutant, alpha-1 (S205C), beta-2, gamma-2 [ 3 ] Sphingosine 1-Phosphate Receptor 4 [ 23 ]
 GABAA Receptor Mutant, alpha-1 (T162C), beta-2, gamma-2 [ 3 ] Sphingosine 1-Phosphate Receptor 5 [ 31 ]
 GABAA Receptor Mutant, alpha-1 (T206C), beta-2, gamma-2 [ 3 ] Src [ 958 ]
 GABAA Receptor Mutant, alpha-1 (V202C), beta-2, gamma-2 [ 3 ] Src Mutant (S345C) [ 4 ]
 GABAA Receptor Mutant, alpha-1 (V211C), beta-2, gamma-2 [ 3 ] Src Mutant (S345C/T338M) [ 4 ]
 GABAA Receptor Mutant, alpha-1 (Y209C), beta-2, gamma-2 [ 1 ] Src Mutant (T338M) [ 9 ]
 GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (A79C) [ 3 ] STE20-Like Kinase MST2 [ 1 ]
 GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (Chimera) [ 3 ] Steroid 11-beta-Hydroxylase (CYP11B1) [ 97 ]
 GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (D56C) [ 3 ] Steroid 17-alpha-Monooxygenase (CYP17) [ 106 ]
 GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (F77C) [ 1 ] Steroid Sulfatase (STS) [ 38 ]
 GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (L140C) [ 3 ] Steroidogenic Factor 1 [ 47 ]
 GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (M130C) [ 3 ] Streptavadin(N23A) [ 1 ]
 GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (R132C) [ 3 ] Streptavadin(N23E) [ 1 ]
 GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (R144C) [ 3 ] Streptavadin(S27A) [ 1 ]
 GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (R185C) [ 3 ] Streptavadin(W108F) [ 1 ]
 GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (R194C) [ 3 ] Streptavadin(W120F) [ 1 ]
 GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (T126C) [ 3 ] Streptavadin(W79F) [ 1 ]
 GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (T142C) [ 3 ] Streptavadin(Y43A) [ 1 ]
 GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (T81C) [ 3 ] Streptavidin [ 1 ]
 GABAA Receptor, alpha-1, beta-2, gamma-2 [ 3 ] Streptavidin (Y43F) [ 1 ]
 GABAA Receptor, alpha-1, beta-3, gamma-2 [ 8 ] T-Cell Protein-Tyrosine Phosphatase (TCPTP) [ 53 ]
 GABAA Receptor, alpha-2, beta-2, gamma-2 [ 3 ] T-Cell Protein-Tyrosine Phosphatase (TCPTP) Mutant (V121L) [ 2 ]
 GABAA Receptor, alpha-2, beta-3, gamma-2 [ 8 ] t-Plasminogen Activator (tPA) [ 66 ]
 GABAA Receptor, alpha-3, beta-2, gamma-2 [ 3 ] Tankyrase-1 [ 1 ]
 GABAA Receptor, alpha-3, beta-3, gamma-2 [ 7 ] TGF-beta Receptor Type-1 [ 43 ]
 GABAA Receptor, alpha-4, beta-2, gamma-2 [ 3 ] TGR5 [ 9 ]
 GABAA Receptor, alpha-4, beta-3, gamma-2 [ 4 ] Thrombin [ 1297 ]
 GABAA Receptor, alpha-5, beta-2, gamma-2 [ 3 ] Thromboxane A2 Synthase (P450 TxA2) [ 20 ]
 GABAA Receptor, alpha-5, beta-3, gamma-2 [ 8 ] Thymidine Kinase [ 30 ]
 GABAA Receptor, alpha-6, beta-2, gamma-2 [ 3 ] Thymidine Kinase (TK.dT) [ 1 ]
 GABAA Receptor, alpha-6, beta-3, gamma-2 [ 7 ] Thymidine Phosphorylase (TP) [ 50 ]
 Galectin-1 [ 14 ] Thymidylate Synthase (TS) [ 68 ]
 Galectin-3 [ 23 ] Thyroid Hormone Receptor (TR-alpha) [ 150 ]
 Galectin-7 [ 12 ] Thyroid Hormone Receptor (TR-beta) [ 145 ]
 Galectin-8 [ 11 ] Tie-2 [ 216 ]
 Galectin-9 [ 12 ] TNF-alpha-Converting Enzyme [ 157 ]
 gamma-Aminobutyric Acid Type B Receptor [ 16 ] Transcription Factor STAT1 [ 11 ]
 Gamma-Secretase [ 94 ] Transcription Factor STAT1:STAT3 Dimer [ 2 ]
 GAR Tfase [ 13 ] Transcription Factor STAT3 [ 92 ]
 Gastric Inhibitory Polypeptide Receptor (GIPR) [ 30 ] Transcriptional Regulator TtgR [ 11 ]
 Geranylgeranyl Diphosphate Synthase (GGPPS) [ 61 ] Transcriptional Regulator TtgR Mutant R176G [ 2 ]
 Geranylgeranyl Transferase (GGTase-I) [ 99 ] Transcriptional Regulator TtgR-DNA [ 4 ]
 Ghrelin Receptor (Growth Hormone Secretagogue Receptor Type 1) [ 130 ] Triacylglycerol Hydrolase [ 46 ]
 Glucagon Receptor [ 30 ] tRNA synthetase (AspRS) [ 3 ]
 Glucocerebrosidase (Acid beta-Glucosidase) [ 74 ] tRNA synthetase (GlnRS) [ 2 ]
 Glucocorticoid Receptor (GR) [ 117 ] tRNA synthetase (GluRS) [ 4 ]
 Glucokinase [ 34 ] tRNA synthetase (GlyRS) [ 6 ]
 Glutamate Carboxypeptidase II (GCPII) [ 38 ] tRNA synthetase (IleRS) [ 21 ]
 Glutaminyl Cyclase [ 86 ] tRNA synthetase (PheRS) [ 45 ]
 Glycogen Phosphorylase (PYGL) [ 101 ] tRNA synthetase (TyrRS) [ 4 ]
 Glycogen Phosphorylase (PYGM) [ 73 ] Trypanothione Reductase (TryR) [ 19 ]
 Glycogen Synthase Kinase-3, alpha [ 172 ] Trypsin [ 377 ]
 Glycogen Synthase Kinase-3, beta [ 609 ] Tryptase [ 44 ]
 Glyoxylate Regulatory Protein (C-AllR) [ 1 ] Tumor Progression Loci-2 Kinase (COT) [ 87 ]
 GRB2 [ 15 ] Tyrosine Kinase ACK1 [ 10 ]
 H1/H5-depleted chromatin [ 2 ] Tyrosine Kinase ALK [ 15 ]
 HCV NS3 Helicase [ 12 ] Tyrosine Kinase Axl [ 4 ]
 HCV NS3-NS4A Serine Proteinase [ 319 ] Tyrosine Kinase BMX [ 1 ]
 HCV NS5B Polymerase [ 156 ] Tyrosine Kinase BRK [ 2 ]
 HCV NS5B Polymerase Mutant (M414T) [ 2 ] Tyrosine Kinase BTK [ 1 ]
 HCV NS5B Polymerase Mutant (M423K) [ 2 ] Tyrosine Kinase c-Kit [ 120 ]
 HCV NS5B Polymerase Mutant (P495A) [ 2 ] Tyrosine Kinase c-Kit Mutant (N822K) [ 7 ]
 HCV NS5B Polymerase Mutant (R501E) [ 2 ] Tyrosine Kinase c-Kit Mutant (V559D) [ 28 ]
 Heat Shock 70kDa Protein 1 [ 50 ] Tyrosine Kinase c-Kit Mutant (V559D, V654A) [ 17 ]
 Heat Shock Protein 90 (Hsp90) [ 488 ] Tyrosine Kinase c-Kit Mutant (V559D/T670I) [ 7 ]
 Heme Oxygenase 1 (HO-1) [ 44 ] Tyrosine Kinase c-Met [ 109 ]
 Heme Oxygenase 2 (HO-2) [ 44 ] Tyrosine Kinase c-Met Mutant (D1228H) [ 1 ]
 Hepsin [ 6 ] Tyrosine Kinase c-Met Mutant (H1094R) [ 1 ]
 hERG Potassium Channel 1 [ 84 ] Tyrosine Kinase c-Met Mutant (M1250T) [ 1 ]
 Histamine H1 Receptor [ 23 ] Tyrosine Kinase c-Met Mutant (V1092I) [ 1 ]
 Histamine H2 Receptor [ 5 ] Tyrosine Kinase c-Met Mutant (Y1230H) [ 1 ]
 Histamine H3 Receptor [ 68 ] Tyrosine Kinase c-Ret [ 15 ]
 Histamine H4 Receptor [ 91 ] Tyrosine Kinase CSF1-R [ 89 ]
 Histone Deacetylase (pfHDAC-1) [ 23 ] Tyrosine Kinase CSF1-R Mutant (FGFR KID Chimera) [ 6 ]
 Histone Deacetylase 1 (HDAC1) [ 191 ] Tyrosine Kinase CSF1-R Mutant (Tie2 KID Chimera) [ 6 ]
 Histone Deacetylase 10 (HDAC10) [ 18 ] Tyrosine Kinase CSK [ 1 ]
 Histone Deacetylase 11 (HDAC11) [ 1 ] Tyrosine Kinase DDR1 [ 24 ]
 Histone Deacetylase 2 (HDAC2) [ 41 ] Tyrosine Kinase DDR2 [ 13 ]
 Histone Deacetylase 3 (HDAC3) [ 83 ] Tyrosine Kinase EPHA3 [ 14 ]
 Histone Deacetylase 4 (HDAC4) [ 72 ] Tyrosine Kinase EPHA6 [ 16 ]
 Histone Deacetylase 4 (HDAC4) Mutant (H976Y) [ 46 ] Tyrosine Kinase EPHA7 [ 10 ]
 Histone Deacetylase 5 (HDAC5) [ 6 ] Tyrosine Kinase EPHB3 [ 3 ]
 Histone Deacetylase 6 (HDAC6) [ 95 ] Tyrosine Kinase EPHB4 [ 8 ]
 Histone Deacetylase 7 (HDAC7) [ 6 ] Tyrosine Kinase FAK [ 3 ]
 Histone Deacetylase 8 (HDAC8) [ 49 ] Tyrosine Kinase FLT3 [ 70 ]
 Histone Lysine Demethylase [ 19 ] Tyrosine Kinase FLT3 Mutant (D835H) [ 23 ]
 Histone-Arginine Methyltransferase CARM1 [ 19 ] Tyrosine Kinase FLT3 Mutant (D835Y) [ 20 ]
 HIV-1 Integrase [ 238 ] Tyrosine Kinase FLT3 Mutant (N841I) [ 22 ]
 HIV-1 Nef [ 5 ] Tyrosine Kinase FLT3-ITD [ 19 ]
 HIV-1 Protease [ 2381 ] Tyrosine Kinase FRK [ 23 ]
 HIV-1 Protease A Subtype [ 5 ] Tyrosine Kinase FYN [ 1 ]
 HIV-1 Protease A Subtype Mutant (V82F/I84V) [ 5 ] Tyrosine Kinase JAK2 [ 1 ]
 HIV-1 Protease AE [ 7 ] Tyrosine Kinase JAK3 [ 41 ]
 HIV-1 Protease AE Mutant (V82F) [ 7 ] Tyrosine Kinase Syk [ 60 ]
 HIV-1 Protease AE-P [ 7 ] Tyrosine Kinase TrkA [ 5 ]
 HIV-1 Protease AE-P Mutant (F82V) [ 7 ] Tyrosine Kinase ZAP-70 [ 80 ]
 HIV-1 Protease B Subtype [ 8 ] Tyrosine-protein kinase ITK [ 77 ]
 HIV-1 Protease B Subtype Mutant (V82F) [ 7 ] Tyrosine-Specific Protein Kinase [ 6 ]
 HIV-1 Protease B Subtype Mutant (V82F/I84V) [ 5 ] Ubiquitin C-terminal Hydrolase L3 (UCH-L3) [ 10 ]
 HIV-1 Protease C Subtype [ 5 ] UDP-3-O-Acyl-GlcNAc Deacetylase (LpxC) [ 14 ]
 HIV-1 Protease C Subtype Mutant (V82F/I84V) [ 5 ] Urea Amidohydrolase [ 11 ]
 HIV-1 Protease Mutant (A71V) [ 5 ] Urokinase (uPA) [ 195 ]
 HIV-1 Protease Mutant (A71V/V82T/I84V) [ 1 ] Urokinase (uPA) Mutant (S190A) [ 14 ]
 HIV-1 Protease Mutant (D30N) [ 6 ] v-Src SH2 Domain [ 4 ]
 HIV-1 Protease Mutant (D30N/A71V) [ 5 ] Vanilloid Receptor 1 (TRPV1, VR1) [ 355 ]
 HIV-1 Protease Mutant (D30N/M36I) [ 5 ] Vasopressin V1a Receptor [ 44 ]
 HIV-1 Protease Mutant (D30N/M36I/A71V) [ 5 ] Vasopressin V2 Receptor [ 59 ]
 HIV-1 Protease Mutant (G73S) [ 3 ] VEGFR-1 (Flt-1) [ 195 ]
 HIV-1 Protease Mutant (I47L) [ 1 ] VEGFR-2 (KDR) [ 1115 ]
 HIV-1 Protease Mutant (I50L) [ 1 ] VEGFR-3 (FLT4) [ 19 ]
 HIV-1 Protease Mutant (I50V) [ 10 ] West Nile Virus (WNV) NS2B-NS3 Protease [ 36 ]
 HIV-1 Protease Mutant (I84V) [ 2 ] XIAP-BIR3 [ 173 ]
 HIV-1 Protease Mutant (L10I,L19Q,K20R,E35D,M36I, ..) [ 6 ] XIAP-Linker-BIR2-BIR3 [ 40 ]