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Targets Binding with 2401 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
Abelson murine leukemia viral oncogene homolog 1
Ki:
832
IC50:
2161
Kd:
1576
EC50:
100
323
23
2D
3D
TSV
Abl
IC50:
111
6
15
2D
3D
TSV
ABL1
Ki:
825
IC50:
2017
Kd:
1548
EC50:
100
315
9
2D
3D
TSV
c-ABL
Ki:
832
IC50:
2050
Kd:
1632
EC50:
100
318
9
2D
3D
TSV
Cereblon/BCR/ABL
Ki:
825
IC50:
2017
Kd:
1548
EC50:
100
315
9
2D
3D
TSV
JTK7
Ki:
825
IC50:
2017
Kd:
1548
EC50:
100
315
9
2D
3D
TSV
Mitogen-activated protein kinase 10/Receptor-interacting serine/threonine-protein kinase 1
Ki:
155
IC50:
2881
Kd:
372
EC50:
83
159
14
2D
3D
TSV
p150
Ki:
832
IC50:
2161
Kd:
1632
EC50:
100
323
23
2D
3D
TSV
Proto-oncogene c-Abl
Ki:
832
IC50:
2050
Kd:
1569
EC50:
100
317
9
2D
3D
TSV
Proto-oncogene tyrosine-protein kinase ABL1
Ki:
832
IC50:
2050
Kd:
1576
EC50:
100
318
9
2D
3D
TSV
Tyrosine-protein kinase (ABL)
Ki:
825
IC50:
2017
Kd:
1548
EC50:
100
315
9
2D
3D
TSV
tyrosine-protein kinase ABL1 isoform a
Ki:
825
IC50:
2017
Kd:
1548
EC50:
100
315
9
2D
3D
TSV
V-abl Abelson murine leukemia viral oncogene homolog 1
Ki:
825
IC50:
2017
Kd:
1548
EC50:
100
315
9
2D
3D
TSV
VHL/BCR-ABL1
Ki:
825
IC50:
2017
Kd:
1548
EC50:
100
315
9
2D
3D
TSV