PMID

Data

Article Title

Organization

Discovery of high affinity inhibitors of Leishmania donovani N-myristoyltransferase.

Imperial College

Discovery of pyridyl-based inhibitors of Plasmodium falciparum N-myristoyltransferase.

Imperial College

Lead optimization of a pyrazole sulfonamide series of Trypanosoma brucei N-myristoyltransferase inhibitors: identification and evaluation of CNS penetrant compounds as potential treatments for stage 2 human African trypanosomiasis.

University Of Dundee

Structure-based design of potent and selective Leishmania N-myristoyltransferase inhibitors.

Imperial College

Discovery of novel and ligand-efficient inhibitors of Plasmodium falciparum and Plasmodium vivax N-myristoyltransferase.

Imperial College

Design and synthesis of inhibitors of Plasmodium falciparum N-myristoyltransferase, a promising target for antimalarial drug discovery.

Imperial College

Discovery of Plasmodium vivax N-myristoyltransferase inhibitors: screening, synthesis, and structural characterization of their binding mode.

Imperial College

Discovery of a novel class of orally active trypanocidal N-myristoyltransferase inhibitors.

University Of Dundee

Derivatives of aryl amines containing the cytotoxic 1,4-dioxo-2-butenyl pharmacophore.

Acadia University

 

A chiral recognition element with an unusual size constraint affects the potency and selectivity for peptidomimetic inhibitors of Candida albicans myristoyl-CoA:protein N-myristoyltransferase

TBA

A Molecular Hybridization Approach for the Design of Potent, Highly Selective, and Brain-Penetrant N-Myristoyltransferase Inhibitors.

University Of Dundee

Design and Synthesis of Brain Penetrant Trypanocidal N-Myristoyltransferase Inhibitors.

University Of Dundee