17 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Synthesis and biological evaluation of a series of N-alkylated imidazole alkanoic acids as mGAT3 selective GABA uptake inhibitors.
Ludwig-Maximilians-Universit£T M£Nchen
Conformationally Restricted GABA with Bicyclo[3.1.0]hexane Backbone as the First Highly Selective BGT-1 Inhibitor.
Hokkaido University
Design, synthesis and SAR studies of GABA uptake inhibitors derived from 2-substituted pyrrolidine-2-yl-acetic acids.
Ludwig-Maximilians-Universit£T M£Nchen
The lignan (-)-hinokinin displays modulatory effects on human monoamine and GABA transporter activities.
Drexel University College Of Medicine
Cyclopropane-based conformational restriction of GABA by a stereochemical diversity-oriented strategy: identification of an efficient lead for potent inhibitors of GABA transports.
Hokkaido University
Synthesis of N-substituted acyclicß-amino acids and their investigation as GABA uptake inhibitors.
Zentrum F£R Pharmaforschung
Aminomethyltetrazoles as potential inhibitors of the¿-aminobutyric acid transporters mGAT1-mGAT4: synthesis and biological evaluation.
Ludwig-Maximilians-University Munich
Design, synthesis, and biological evaluation of the N-diarylalkenyl-piperidinecarboxylic acid derivatives as GABA uptake inhibitors (I).
Fudan University
Development of imidazole alkanoic acids as mGAT3 selective GABA uptake inhibitors.
Ludwig-Maximilians-University Munich
Stereospecific synthesis and structure-activity relationships of unsymmetrical 4,4-diphenylbut-3-enyl derivatives of nipecotic acid as GAT-1 inhibitors.
Glaxosmithkline
Azetidine derivatives as novel gamma-aminobutyric acid uptake inhibitors: synthesis, biological evaluation, and structure-activity relationship.
Zentrum F£R Pharmaforschung
Screening oxime libraries by means of mass spectrometry (MS) binding assays: Identification of new highly potent inhibitors to optimized inhibitors ?-aminobutyric acid transporter 1.
Ludwig-Maximilians-University M£Nchen
Five-Membered N-Heterocyclic Scaffolds as Novel Amino Bioisosteres at ?-Aminobutyric Acid (GABA) Type A Receptors and GABA Transporters.
University Of Copenhagen
Novel Allosteric Ligands of ?-Aminobutyric Acid Transporter 1 (GAT1) by MS Based Screening of Pseudostatic Hydrazone Libraries.
Ludwig-Maximilians-Universit£T M£Nchen
Design, synthesis and evaluation of substituted triarylnipecotic acid derivatives as GABA uptake inhibitors: identification of a ligand with moderate affinity and selectivity for the cloned human GABA transporter GAT-3.
Synaptic Pharmaceutical