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24 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
28319392 216 Scaffold Repurposing of Nucleosides (Adenosine Receptor Agonists): Enhanced Activity at the Human Dopamine and Norepinephrine Sodium Symporters.EBI National Institute of Diabetes and Digestive and Kidney Diseases
28435536 60 Norbenzomorphan Scaffold: Chemical Tool for Modulating Sigma Receptor-Subtype Selectivity.EBI The University of Texas at Austin
30103189 21 Pyridine bioisosteres of potent GluN2B subunit containing NMDA receptor antagonists with benzo[7]annulene scaffold.EBI Institut f£r Pharmazeutische und Medizinische Chemie der Westf£lischen Wilhelms-Universit£t M£nster
30025348 149 Neurogenic and neuroprotective donepezil-flavonoid hybrids with sigma-1 affinity and inhibition of key enzymes in Alzheimer's disease.EBI Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
30223122 64 Identification of dual Sigma1 receptor modulators/acetylcholinesterase inhibitors with antioxidant and neurotrophic properties, as neuroprotective agents.EBI University of Pavia
30143421 27 New piperidine-based derivatives as sigma receptor ligands. Synthesis and pharmacological evaluation.EBI University of Trieste
29289890 22 Hydroxymethyl bioisosteres of phenolic GluN2B-selective NMDA receptor antagonists: Design, synthesis and pharmacological evaluation.EBI Institut f£r Pharmazeutische und Medizinische Chemie der Universit£t M£nster
29287249 13 Multifunctional thiosemicarbazones and deconstructed analogues as a strategy to study the involvement of metal chelation, Sigma-2 (?EBI Universit£ degli Studi di Bari ALDO MORO
29039662 62 Quest for Novel Chemical Entities through Incorporation of Silicon in Drug Scaffolds.EBI CSIR-National Chemical Laboratory
29482951 10 Synthesis of 3-aza[4.4.3]propellanes with high ?EBI Institut f£r Pharmazeutische und Medizinische Chemie der Westf£lischen Wilhelms-Universit£t M£nster
29505935 13 Indole in the target-based design of anticancer agents: A versatile scaffold with diverse mechanisms.EBI Mazandaran University of Medical Sciences
28704758 50 Deconstruction - reconstruction approach to analyze the essential structural elements of tetrahydro-3-benzazepine-based antagonists of GluN2B subunit containing NMDA receptors.EBI Institut f£r Pharmazeutische und Medizinische Chemie der Westf£lischen Wilhelms-Universit£t M£nster
29254894 18 2-Methyltetrahydro-3-benzazepin-1-ols - The missing link in SAR of GluN2B selective NMDA receptor antagonists.EBI Institut f£r Pharmazeutische und Medizinische Chemie der Westf£lischen Wilhelms-Universit£t M£nster
30350997 111 Synthesis, Receptor Affinity, and Antiallodynic Activity of Spirocyclic ? Receptor Ligands with Exocyclic Amino Moiety.EBI Universit£t M£nster
29656199 148 Investigating isoindoline, tetrahydroisoquinoline, and tetrahydrobenzazepine scaffolds for their sigma receptor binding properties.EBI University of Texas at Austin
29438891 50 Synthesis and pharmacological evaluation of 6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline derivatives as sigma-2 receptor ligands.EBI Guangdong Medical University
29969030 24 Contilisant, a Tetratarget Small Molecule for Alzheimer's Disease Therapy Combining Cholinesterase, Monoamine Oxidase Inhibition, and H3R Antagonism with S1R Agonism Profile.EBI IQOG, CSIC
28764962 90 Chiral-pool synthesis of 1,2,4-trisubstituted 1,4-diazepanes as novel?EBI Institut f£r Pharmazeutische und Medizinische Chemie der Universit£t M£nster
28347632 18 Do spiroindolines have the potential to replace vesamicol as lead compound for the development of radioligands targeting the vesicular acetylcholine transporter?EBI Helmholtz-Zentrum Dresden-Rossendorf
28320613 19 Synthesis of conformationally restricted 1,3-dioxanes to analyze the bioactive conformation of 1,3-dioxane-based?EBI Institut f£r Pharmazeutische und Medizinische Chemie der Westf£lischen Wilhelms-Universit£t M£nster
28501431 27 Lipase-catalyzed kinetic resolution as key step in the synthesis of enantiomerically pure? ligands with 2-benzopyran structure.EBI Universit£t M£nster
28495085 17 Reevaluation of fenpropimorph as a? receptor ligand: Structure-affinity relationship studies at human?EBI Virginia Commonwealth University
16242653 33 A proteome-wide CDK/CRK-specific kinase inhibitor promotes tumor cell death in the absence of cell cycle progression.BDB GPC Biotech, Inc.
16807364 18 Inhibition of the enzymatic activity of heme oxygenases by azole-based antifungal drugs.BDB Queen's University