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22 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
26862980 37 Tweaking Subtype Selectivity and Agonist Efficacy at (S)-2-Amino-3-(3-hydroxy-5-methyl-isoxazol-4-yl)propionic acid (AMPA) Receptors in a Small Series of BnTetAMPA Analogues.EBI University of Copenhagen
26653877 47 Studies on Aryl-Substituted Phenylalanines: Synthesis, Activity, and Different Binding Modes at AMPA Receptors.EBI University of Copenhagen
24824658 8 Structure-activity relationship studies of N-methylated and N-hydroxylated spider polyamine toxins as inhibitors of ionotropic glutamate receptors.EBI University of Copenhagen
23320429 48 Structure-activity relationship studies of argiotoxins: selective and potent inhibitors of ionotropic glutamate receptors.EBI University of Copenhagen
23092360 19 General synthesis ofß-alanine-containing spider polyamine toxins and discovery of nephila polyamine toxins 1 and 8 as highly potent inhibitors of ionotropic glutamate receptors.EBI University of Copenhagen
21188966 2 Solid-phase synthesis and biological evaluation of Joro spider toxin-4 from Nephila clavata.EBI University of Copenhagen
19588945 55 The glutamate receptor GluR5 agonist (S)-2-amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic acid and the 8-methyl analogue: synthesis, molecular pharmacology, and biostructural characterization.EBI University of Copenhagen
18811139 126 1H-cyclopentapyrimidine-2,4(1H,3H)-dione-related ionotropic glutamate receptors ligands. structure-activity relationships and identification of potent and Selective iGluR5 modulators.EBI European Research Centre for Drug Discovery and Development (NatSynDrugs)
18338843 57 Synthesis and pharmacological characterization at glutamate receptors of the four enantiopure isomers of tricholomic acid.EBI Universit£ degli Studi di Milano
9357531 58 Synthesis of willardiine and 6-azawillardiine analogs: pharmacological characterization on cloned homomeric human AMPA and kainate receptor subtypes.EBI University of Bristol
1977908 10 (R)-4-oxo-5-phosphononorvaline: a new competitive glutamate antagonist at the NMDA receptor complex.EBI Merrell Dow Research Institute
21923187 5 A new phenylalanine derivative acts as an antagonist at the AMPA receptor GluA2 and introduces partial domain closure: synthesis, resolution, pharmacology, and crystal structure.EBI University of Copenhagen
21067182 37 Biostructural and Pharmacological Studies of Bicyclic Analogues of the 3-Isoxazolol Glutamate Receptor Agonist Ibotenic AcidEBI TBA
20684595 374 Quinazolin-4-one derivatives: A novel class of noncompetitive NR2C/D subunit-selective N-methyl-D-aspartate receptor antagonists.EBI Emory University
20096591 84 Developing a complete pharmacology for AMPA receptors: a perspective on subtype-selective ligands.EBI University of California
 10 Synthesis and biology of the rigidified glutamate analogue, trans-2-carboxyazetidine-3-acetic acid (t-CAA)EBI TBA
17455929 36 A tetrazolyl-substituted subtype-selective AMPA receptor agonist.EBI University of Copenhagen
16942015 43 Uncompetitive antagonism of AMPA receptors: Mechanistic insights from studies of polyamine toxin derivatives.EBI The Danish University of Pharmaceutical Sciences
15615543 56 Bioisosteric modifications of 2-arylureidobenzoic acids: selective noncompetitive antagonists for the homomeric kainate receptor subtype GluR5.EBI The Danish University of Pharmaceutical Sciences
12747796 39 Design, synthesis, and pharmacology of a highly subtype-selective GluR1/2 agonist, (RS)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)propionic acid (Cl-HIBO).EBI The Danish University of Pharmaceutical Sciences
7629789 8 Synthesis, resolution, and biological evaluation of the four stereoisomers of 4-methylglutamic acid: selective probes of kainate receptors.EBI Symphony Pharmaceuticals, Inc.