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12 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27031670 16 Monoacidic Inhibitors of the Kelch-like ECH-Associated Protein 1: Nuclear Factor Erythroid 2-Related Factor 2 (KEAP1:NRF2) Protein-Protein Interaction with High Cell Potency Identified by Fragment-Based Discovery.EBI Astex Pharmaceuticals
26502061 6 Targeting Mitogen-Activated Protein Kinase-Activated Protein Kinase 2 (MAPKAPK2, MK2): Medicinal Chemistry Efforts To Lead Small Molecule Inhibitors to Clinical Trials.EBI Universit£ di Siena
21965623 170 In vitro inhibition of the bile salt export pump correlates with risk of cholestatic drug-induced liver injury in humans.EBI AstraZeneca
25310383 50 Potent nonimmunosuppressive cyclophilin inhibitors with improved pharmaceutical properties and decreased transporter inhibition.EBI Novartis Institutes for Biomedical Research
12739759 25 Fluorescent substrates of sister-P-glycoprotein (BSEP) evaluated as markers of active transport and inhibition: evidence for contingent unequal binding sites.EBI Schering-Plough Research Institute
11557132 5 Troglitazone-induced intrahepatic cholestasis by an interference with the hepatobiliary export of bile acids in male and female rats. Correlation with the gender difference in troglitazone sulfate formation and the inhibition of the canalicular bile salt export pump (Bsep) by troglitazone and troglEBI F. Hoffmann-La Roche Ltd.
10648470 4 Drug- and estrogen-induced cholestasis through inhibition of the hepatocellular bile salt export pump (Bsep) of rat liver.EBI University Hospital
11248200 4 Characterization of bile acid transport mediated by multidrug resistance associated protein 2 and bile salt export pump.EBI The University of Tokyo
28135235 71 An allosteric PRC2 inhibitor targeting the H3K27me3 binding pocket of EED.BDB Novartis Institutes for BioMedical Research
15901796 21 Bile salt export pump (BSEP/ABCB11) can transport a nonbile acid substrate, pravastatin.BDB University of Tokyo