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514 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
 1 Peptide argininol “inverse substrates” of anisic acid: Novel inhibitors of the trypsin-like serine proteinasesEBI TBA
 19 Rational design of selective thrombin inhibitorsEBI TBA
 15 Rational design, synthesis, and serine protease inhibitory activity of a novel P1-argininal derivative featuring a conformationally constrained P2–P3 bicyclic lactam moietyEBI TBA
 37 Synthesis and biological activity of P2–P4 azapeptidomimetic P1-argininal and P1-ketoargininamide derivatives: a novel class of serine protease inhibitorsEBI TBA
 32 Bisbenzamidine isoxazoline derivatives as factor Xa inhibitorsEBI TBA
 27 Rational design and synthesis of a novel, selective class of thrombin inhibitors: P1-argininal derivatives incorporating P3---P4 quaternary lactam dipeptide surrogatesEBI TBA
 44 Biaryl substituted alkylboronate esters as thrombin inhibitorsEBI TBA
 3 An efficient preparation of the potent and selective pseudopeptide thrombin inhibitor, inogatranEBI TBA
 25 Design and synthesis of a novel class of thrombin inhibitors incorporating heterocyclic dipeptide surrogatesEBI TBA
 14 RATIONAL DESIGN, SYNTHESIS, AND SERINE PROTEASE INHIBITORY ACTIVITY OF NOVEL P1-ARGININOYL HETEROCYCLESEBI TBA
 4 Synthesis, evaluation, and crystallographic analysis of L-371,912: A potent and selective active-site thrombin inhibitorEBI TBA
 78 Synthesis and evaluation of 2-aryl-4H-3,1-benzoxazin-4-ones as C1r serine protease inhibitorsEBI TBA
 22 Synthesis of conformationally-restricted boropeptide thrombin inhibitorsEBI TBA
 8 Design and synthesis of ring-constrained boropeptide thrombin inhibitorsEBI TBA
 24 Novel thrombin inhibitors that are based on a macrocyclic tripeptide motifEBI TBA
 61 (N-acyl-N-alkyl)glycyl borolysine analogs: A new class of potent thrombin inhibitorsEBI TBA
 15 O-benzyl hydroxyproline as a bioisostere for Phe-Pro: Novel dipeptide thrombin inhibitorsEBI TBA
 12 Tripeptidyl pyridinium methyl ketones as potent active site inhibitors of thrombinEBI TBA
 12 Derivatives of 5-amidine indole as inhibitors of thrombin catalytic activityEBI TBA
 13 Characterization of LY806303 as a potent and selective inhibitor of thrombinEBI TBA
 6 α-hydroxy- and α-ketoester functionalized thrombin inhibitorsEBI TBA