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59 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27390066 99 Discovery of potent and selective inhibitors of human aminopeptidases ERAP1 and ERAP2 by screening libraries of phosphorus-containing amino acid and dipeptide analogues.EBI Wroclaw University of Technology
27100031 85 A structural insight into the P1S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases.EBI Wroclaw University of Technology
27039251 66 Design, synthesis and anti-HIV-1 evaluation of hydrazide-based peptidomimetics as selective gelatinase inhibitors.EBI Shandong University
26629857 44 Novel leucine ureido derivatives as aminopeptidase N inhibitors. Design, synthesis and activity evaluation.EBI Fudan University
26386821 15 Synthesis of chiral ND-322, ND-364 and ND-364 derivatives as selective inhibitors of human gelatinase.EBI Shandong University
25982416 43 Exploring S1 plasticity and probing S1' subsite of mammalian aminopeptidase N/CD13 with highly potent and selective aminobenzosuberone inhibitors.EBI Universit£ de Haute Alsace
25192493 57 Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and selective inhibitors of neutral aminopeptidases.EBI University of Athens
24755524 60 Design, synthesis and preliminary evaluation ofa-sulfonyl┐-(glycinyl-amino)proline peptidomimetics as matrix metalloproteinase inhibitors.EBI Shandong University
24055078 14 Synthesis of amino-hydroxy-benzocycloheptenones as potent, selective, non-peptidic dinuclear zinc metalloaminopeptidase inhibitors.EBI Universit£ de Haute Alsace
23860593 17 Novel▀-dicarbonyl derivatives as inhibitors of aminopeptidase N (APN).EBI Shandong University
23528299 4 Discovery of a synthetic Aminopeptidase N inhibitor LB-4b as a potential anticancer agent.EBI Shandong University
23510562 30 Novel indoline-2,3-dione derivatives as inhibitors of aminopeptidase N (APN).EBI Shandong University
23428964 9 Selective aminopeptidase-N (CD13) inhibitors with relevance to cancer chemotherapy.EBI Universit£ de Haute-Alsace
23453219 29 Novel leucine ureido derivatives as inhibitors of aminopeptidase N (APN).EBI Shandong University
23176597 14 Structure-activity relationships and blood distribution of antiplasmodial aminopeptidase-1 inhibitors.EBI INSERM
22796349 34 Rapid and efficient synthesis of a novel series of substituted aminobenzosuberone derivatives as potent, selective, non-peptidic neutral aminopeptidase inhibitors.EBI Universit£ de Haute Alsace
22901392 27 A novel aminopeptidase N inhibitor developed by virtual screening approach.EBI Shandong Academy of Sciences
22607877 38 Design, synthesis and biological evaluation of novel amino acid ureido derivatives as aminopeptidase N/CD13 inhibitors.EBI Shandong University
19339187 49 Novel aminopeptidase N inhibitors derived from antineoplaston AS2-5 (Part II).EBI Shandong University
19329328 42 Novel aminopeptidase N inhibitors derived from antineoplaston AS2-5 (Part I).EBI Shandong University
12801228 18 The most potent organophosphorus inhibitors of leucine aminopeptidase. Structure-based design, chemistry, and activity.EBI Wroclaw University of Technology
10753476 84 Phosphinic derivatives as new dual enkephalin-degrading enzyme inhibitors: synthesis, biological properties, and antinociceptive activities.EBI INSERM
10602705 82 Investigation of subsite preferences in aminopeptidase A (EC 3.4.11.7) led to the design of the first highly potent and selective inhibitors of this enzyme.EBI INSERM
1348542 23 Potent and systemically active aminopeptidase N inhibitors designed from active-site investigation.EBI INSERM
1347791 35 Analgesic dipeptide derivatives. 7. 3,7-Diamino-2-hydroxyheptanoic acid (DAHHA) containing dipeptide analogues of the analgesic compound H-Lys-Trp(Nps)-OMe.EBI Instituto de Qu£mica M£dica
3184126 46 Synthesis of sulfur-containing analogues of bestatin. Inhibition of aminopeptidases by alpha-thiolbestatin analogues.EBI University of Wisconsin
3897541 27 New bidentates as full inhibitors of enkephalin-degrading enzymes: synthesis and analgesic properties.EBI TBA
6142952 41 Inhibition of aminopeptidases by amastatin and bestatin derivatives. Effect of inhibitor structure on slow-binding processes.EBI TBA
10386926 29 Design of the first highly potent and selective aminopeptidase N (EC 3.4.11.2) inhibitor.EBI INSERM
22206607 9 Novel potent 2,5-pyrrolidinedione peptidomimetics as aminopeptidase N inhibitors. Design, synthesis and activity evaluation.EBI Central South University
21911297 40 Design, synthesis and biological evaluation of novel 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid derivatives as aminopeptidase N/CD13 inhibitors.EBI Shan Dong University
21843945 36 A novel amino-benzosuberone derivative is a picomolar inhibitor of mammalian aminopeptidase N/CD13.EBI Universit£ de Haute Alsace
21802307 64 Novel aminopeptidase N (APN/CD13) inhibitors derived from chloramphenicol amine.EBI Shandong University
18458130 8 Chemical target validation studies of aminopeptidase in malaria parasites using alpha-aminoalkylphosphonate and phosphonopeptide inhibitors.EBI Trinity College
21194957 27 Design, synthesis and biological evaluation of novel L-lysine ureido derivatives as aminopeptidase N inhibitors.EBI Shandong University
20637634 48 Novel aminopeptidase N (APN/CD13) inhibitors derived from 3-phenylalanyl-N'-substituted-2,6-piperidinedione.EBI Shandong University
20347318 49 New aromatic monoesters of alpha-aminoaralkylphosphonic acids as inhibitors of aminopeptidase N/CD13.EBI Wroclaw University of Technology
19969464 56 Design, synthesis and primary activity assay of bi- or tri-peptide analogues with the scaffold l-arginine as amino-peptidase N/CD13 inhibitors.EBI Shandong University
19782572 62 Design, synthesis, and preliminary studies of the activity of novel derivatives of N-cinnamoyl-L-aspartic acid as inhibitors of aminopeptidase N/CD13.EBI Shandong University
19683842 27 Novel cyclic-imide peptidomimetics as aminopeptidase N inhibitors. Design, chemistry and activity evaluation. Part I.EBI Shandong University
19454370 52 Design, synthesis and primary activity evaluation of L-arginine derivatives as amino-peptidase N/CD13 inhibitors.EBI Shandong University
19423354 26 Design and synthesis of novel chloramphenicol amine derivatives as potent aminopeptidase N (APN/CD13) inhibitors.EBI Shandong University
19299146 33 Design, synthesis and SAR studies of tripeptide analogs with the scaffold 3-phenylpropane-1,2-diamine as aminopeptidase N/CD13 inhibitors.EBI Shandong University
18996018 42 Novel 3-phenylpropane-1,2-diamine derivates as inhibitors of aminopeptidase N (APN).EBI Shandong University
18571419 24 Novel aminopeptidase N inhibitors derived from 1,3,4-thiadiazole scaffold.EBI ShanDong University
18524593 12 First synthesis of alpha-aminoalkyl-(N-substituted)thiocarbamoyl-phosphinates: inhibitors of aminopeptidase N (APN/CD13) with the new zinc-binding group.EBI Wroc£?aw University of Technology
17433673 44 Novel 3-galloylamido-N'-substituted-2,6-piperidinedione-N-acetamide peptidomimetics as metalloproteinase inhibitors.EBI Shandong University
17326615 49 Novel selective inhibitors of the zinc plasmodial aminopeptidase PfA-M1 as potential antimalarial agents.EBI Inserm
17070058 15 A library of novel hydroxamic acids targeting the metallo-protease family: design, parallel synthesis and screening.EBI University of Lille 2
12930151 1 Synthesis and biological evaluation of novel flavone-8-acetic acid derivatives as reversible inhibitors of aminopeptidase N/CD13.EBI INSERM
7915326 28 Differential inhibition of aminopeptidase A and aminopeptidase N by new beta-amino thiols.EBI INSERM
2738884 27 New kelatorphan-related inhibitors of enkephalin metabolism: improved antinociceptive properties.EBI INSERM
22545941 14 Design, synthesis and biological evaluation of novel L-isoserine tripeptide derivatives as aminopeptidase N inhibitors.BDB Shandong University
22380779 35 Design, synthesis and preliminary activity evaluation of novel 3-amino-2-hydroxyl-3-phenylpropanoic acid derivatives as aminopeptidase N/CD13 inhibitors.BDB Shan Dong University
21770859 26 Synthesis of a novel series of L-isoserine derivatives as aminopeptidase N inhibitors.BDB Shan Dong University
27113097 7 Design, synthesis, and biological characterization of tamibarotene analogs as anticancer agents.BDB Shandong University
16844380 76 Synthesis and structure activity relationships of novel non-peptidic metallo-aminopeptidase inhibitors.BDB ENSCMu
17850059 195 N-benzoylpyrazoles are novel small-molecule inhibitors of human neutrophil elastase.BDB Montana State University