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32 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27964995 42 Synthesis and optimization of novela-phenylglycinamides as selective TRPM8 antagonists.EBI Kissei Pharmaceutical Co., Ltd.
27437071 8 N-(2-Alkyleneimino-3-phenylpropyl)acetamide Compounds and Their Use against Pain and Pruritus via Inhibition of TRPA1 Channels.EBI Temple University
26942860 101 Optimization of a Novel Quinazolinone-Based Series of Transient Receptor Potential A1 (TRPA1) Antagonists Demonstrating Potent in Vivo Activity.EBI Amgen, Inc.
26750258 67 TRPA1 channels as targets for resveratrol and related stilbenoids.EBI Sapienza Universit£ di Roma
26706172 21 a-Aryl pyrrolidine sulfonamides as TRPA1 antagonists.EBI Genentech
26263397 22 Structure-Activity Relationship Study on Isothiocyanates: Comparison of TRPA1-Activating Ability between Allyl Isothiocyanate and Specific Flavor Components of Wasabi, Horseradish, and White Mustard.EBI University of Shizuoka
24953819 49 Development of novel azabenzofuran TRPA1 antagonists as in vivo tools.EBI Amgen Inc.
24880903 24 Discovery of a series of aryl-N-(3-(alkylamino)-5-(trifluoromethyl)phenyl)benzamides as TRPA1 antagonists.EBI AstraZeneca
25455494 172 Effect of acyclic monoterpene alcohols and their derivatives on TRP channels.EBI Sapienza Universit£ di Roma
25455182 52 Identification of a novel 2-pyridyl-benzensulfonamide derivative, RQ-00203078, as a selective and orally active TRPM8 antagonist.EBI RaQualia Pharma Inc.
24884675 70 Discovery, optimization, and biological evaluation of 5-(2-(trifluoromethyl)phenyl)indazoles as a novel class of transient receptor potential A1 (TRPA1) antagonists.EBI Genomics Institute of the Novartis Research Foundation
24835202 68 Discovery of a 4-aryloxy-1H-pyrrolo[3,2-c]pyridine and a 1-aryloxyisoquinoline series of TRPA1 antagonists.EBI AstraZeneca
24484240 19 Activation and inhibition of thermosensitive TRP channels by voacangine, an alkaloid present in Voacanga africana, an African tree.EBI University of Shizuoka
23993334 70 3-Ylidenephthalides as a new class of transient receptor potential channel TRPA1 and TRPM8 modulators.EBI Sapienza Universit£ di Roma
23886683 54 The discovery of potent blockers of the canonical transient receptor channels, TRPC3 and TRPC6, based on an anilino-thiazole pharmacophore.EBI GlaxoSmithKline
23474898 161 Biaryl tetrazolyl ureas as inhibitors of endocannabinoid metabolism: modulation at the N-portion and distal phenyl ring.EBI Sapienza Universit£ di Roma
23121096 86 Ion channels as therapeutic targets: a drug discovery perspective.EBI Pfizer Inc.
22503249 149 Modulation of thermo-transient receptor potential (thermo-TRP) channels by thymol-based compounds.EBI Sapienza Universit£ di Roma
22868228 57 N-1-Alkyl-2-oxo-2-aryl amides as novel antagonists of the TRPA1 receptor.EBI AstraZeneca
20356305 151 Transient receptor potential ankyrin 1 (TRPA1) channel as emerging target for novel analgesics and anti-inflammatory agents.EBI Ferrara University
17237762 10 Noxious compounds activate TRPA1 ion channels through covalent modification of cysteines.EBI The Scripps Research Institute
22325155 20 7-Substituted-pyrrolo[3,2-d]pyrimidine-2,4-dione derivatives as antagonists of the transient receptor potential ankyrin 1 (TRPA1) channel: a promising approach for treating pain and inflammation.EBI University of Ferrara
22222037 77 Tricyclic 3,4-dihydropyrimidine-2-thione derivatives as potent TRPA1 antagonists.EBI Janssen Research& Development, Janssen Pharmaceutica N.V.
21741838 17 Design and pharmacological evaluation of PF-4840154, a non-electrophilic reference agonist of the TrpA1 channel.EBI Pfizer Inc.
20806939 52 Analogues of morphanthridine and the tear gas dibenz[b,f][1,4]oxazepine (CR) as extremely potent activators of the human transient receptor potential ankyrin 1 (TRPA1) channel.EBI Johnson& Johnson Pharmaceutical Research& Development
19875281 73 Synthesis and biological evaluation of piperazinyl carbamates and ureas as fatty acid amide hydrolase (FAAH) and transient receptor potential (TRP) channel dual ligands.EBI Sapienza Universit£ di Roma
19945872 12 Oxime derivatives related to AP18: Agonists and antagonists of the TRPA1 receptor.EBI Renovis, Inc.