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17 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27721153 18 Design, synthesis and biological evaluation of new phthalimide and saccharin derivatives with alicyclic amines targeting cholinesterases, beta-secretase and amyloid beta aggregation.EBI Jagiellonian University Medical College
28043778 3 Neuritogenic activity of bi-functional bis-tryptoline triazole.EBI Chiang Mai University
27816517 14 Discovery of furo[2,3-d][1,3]thiazinamines as beta amyloid cleaving enzyme-1 (BACE1) inhibitors.EBI Bristol-Myers Squibb
27104967 1 Pregnane-10,2-carbolactones from a Hawaiian Marine Sponge in the Genus Myrmekioderma.EBI University of Hawaii at Manoa
24704031 69 The evolution of amidine-based brain penetrant BACE1 inhibitors.EBI Janssen Research and Development
14684336 20 P3 cap modified Phe*-Ala series BACE inhibitors.EBI Lilly Research Laboratories
14684335 21 Phe*-Ala-based pentapeptide mimetics are BACE inhibitors: P2 and P3 SAR.EBI Lilly Research Laboratories
14643321 31 Design and synthesis of statine-containing BACE inhibitors.EBI Eli Lilly and Company
15177452 13 Synthesis and SAR of bis-statine based peptides as BACE 1 inhibitors.EBI Wyeth Research
15006396 4 KMI-358 and KMI-370, highly potent and small-sized BACE1 inhibitors containing phenylnorstatine.EBI Kyoto Pharmaceutical University
14741251 12 Rational design and synthesis of selective BACE-1 inhibitors.EBI Merck Research Laboratories
14643307 1 KMI-008, a novel beta-secretase inhibitor containing a hydroxymethylcarbonyl isostere as a transition-state mimic: design and synthesis of substrate-based octapeptides.EBI Kyoto Pharmaceutical University
14592472 15 Green tea catechins as a BACE1 (beta-secretase) inhibitor.EBI Kyungpook National University
19195886 22 Structure-based design and synthesis of macrocyclic peptidomimetic beta-secretase (BACE-1) inhibitors.BDB Novartis
16451048 7 Aminoethylenes: a tetrahedral intermediate isostere yielding potent inhibitors of the aspartyl protease BACE-1.BDB Sunesis
16854060 58 Structure-based design and synthesis of macroheterocyclic peptidomimetic inhibitors of the aspartic protease beta-site amyloid precursor protein cleaving enzyme (BACE).BDB Universite de Montreal at Succursale Centre-Ville
16078837 34 Structure-based design, synthesis, and memapsin 2 (BACE) inhibitory activity of carbocyclic and heterocyclic peptidomimetics.BDB Universite de Montreal at Succursale Centre-Ville