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BindingDB Data by target


Target NameProtein/Small MoleculeOtherArticles
Ki
Data
IC50
Data
Kd
Data
EC50
Data
otherITC
Data
1 11-beta-Hydroxysteroid Dehydrogenase 1 (11-beta-HSD1) 16 40 0 0 0 0 0 2
2 11-beta-Hydroxysteroid Dehydrogenase 2 (11-beta-HSD2) 0 38 0 0 0 0 0 1
3 17-beta-Hydroxysteroid Dehydrogenase 1 (17-beta-HSD1) 2 3 0 0 1 0 0 1
4 17-beta-Hydroxysteroid Dehydrogenase 5 (17-beta-HSD5, AKR1C3) 5 3 0 0 0 0 0 2
5 2S-ScamLA 0 0 0 0 0 0 1 1
6 3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) 0 114 0 0 0 0 0 7
7 3S-ScamLA 0 0 0 0 0 0 1 1
8 Ab 3B44 0 0 0 0 0 8 0 1
9 Ab N1G9 0 0 0 0 0 4 0 1
10 ABL 0 44 63 0 0 0 0 5
11 Acetate Operon Repressor (C-IclR) 0 0 0 0 0 2 0 1
12 Acetate Operon Repressor (IclR) 0 0 0 0 0 2 0 1
13 Acetylcholinesterase (AChE) 54 749 0 0 0 0 0 38
14 Activated Protein C (APC) 1 0 0 0 0 0 0 1
15 Adenosine A3 Receptor 27 0 0 4 2 0 0 1
16 Adenosine Deaminase 5 0 0 0 0 0 0 1
17 Adenosine Kinase (AK) 0 8 0 0 0 0 0 1
18 Adenosine Receptor A1 59 0 0 0 10 0 0 3
19 Adenosine Receptor A2A 70 0 3 0 15 0 0 3
20 Aldehyde Reductase (ALR1) 0 40 0 0 0 0 0 1
21 Aldose Reductase (ALR2) 39 130 0 0 1 12 0 8
22 Aldosterone Synthase (CYP11B2) 4 83 0 0 11 0 0 6
23 alpha-Glucosidase (alpha-Glu) 0 14 0 0 0 0 0 1
24 alpha-Methylacyl-CoA Racemase 10 0 0 0 0 0 0 1
25 Alpha2 Adrenoreceptor 4 0 0 0 0 0 0 1
26 Androgen Receptor (AR) 232 91 0 132 0 0 0 14
27 Angiotensin-Converting Enzyme 33 6 0 0 0 0 0 3
28 Angiotensin-Converting Enzyme 2 23 13 0 0 0 0 0 2
29 Anthrax Lethal Factor (LF) 54 121 0 0 0 0 0 6
30 apocytochrome b562 0 0 0 0 0 1 0 1
31 apocytochrome b562(denatured) 0 0 0 0 0 1 0 1
32 Apoptosis Regulator Bcl-2 52 0 0 52 0 0 0 1
33 Apoptosis Regulator Bcl-xL 52 43 0 52 0 0 0 1
34 Aromatase (CYP19) 74 321 0 0 18 0 0 18
35 Aurora Kinase A (Aurora-A) 1 69 0 0 0 0 0 6
36 Aurora Kinase B (Aurora-B) 1 6 0 0 0 0 0 2
37 Aurora Kinase C (Aurora-C) 1 0 0 0 0 0 0 1
38 B-RAF 0 2 0 0 0 0 0 1
39 beta-Secretase (BACE-1) 51 213 0 0 3 0 0 24
40 beta-Secretase (BACE-2) 12 12 0 0 0 0 0 4
41 BirA Bifunctional Protein 0 0 0 0 0 16 0 2
42 Butyrylcholinesterase (BuChE) 37 421 0 0 0 0 0 28
43 c-Kit 0 94 21 0 0 0 0 7
44 CaM Kinase II 0 42 0 0 0 0 0 3
45 CAM-alpha-lactalbumin 0 0 0 0 0 0 4 1
46 CAM-BPTI 0 0 0 0 0 0 5 1
47 CAM-RNase A 0 0 0 0 0 0 4 1
48 cAMP-Dependent Protein Kinase (PKA) 5 455 0 0 0 0 0 33
49 Cannabinoid Receptor 1 91 0 0 0 0 0 0 2
50 Cannabinoid Receptor 2 91 0 0 54 0 0 0 2
51 Carbonic Anhydrase (hpCA) 47 0 0 0 0 0 0 1
52 Carbonic Anhydrase I 351 5 5 0 0 0 0 13
53 Carbonic Anhydrase II 432 79 28 0 0 0 0 23
54 Carbonic Anhydrase IV 179 24 0 0 0 0 0 8
55 Carbonic Anhydrase IX 200 5 0 0 0 0 0 10
56 Carbonic Anhydrase VA 88 0 0 0 0 0 0 3
57 Carbonic Anhydrase VB 42 0 0 0 0 0 0 2
58 Carbonic Anhydrase VII 8 0 0 0 0 0 0 1
59 Carbonic Anhydrase XII 8 0 0 0 0 0 0 1
60 Carbonic Anhydrase XIII 6 0 0 0 0 0 0 1
61 Carbonic Anhydrase XIV 8 0 0 0 0 0 0 1
62 Carboxypeptidase A (CPA) 7 8 0 0 0 0 0 2
63 Casein Kinase I 0 12 0 0 0 0 0 3
64 Casein Kinase II 13 7 0 0 0 0 0 5
65 Caspase-1 47 77 0 0 0 0 0 9
66 Caspase-2 17 7 0 0 0 0 0 3
67 Caspase-3 101 249 0 0 0 9 0 15
68 Caspase-3|IST-1 Complex 7 0 0 0 0 9 0 1
69 Caspase-4 17 0 0 0 0 0 0 2
70 Caspase-5 9 0 0 0 0 0 0 1
71 Caspase-6 17 36 0 0 0 0 0 4
72 Caspase-7 18 94 0 0 0 0 0 7
73 Caspase-8 19 93 0 0 0 0 0 7
74 Caspase-9 8 0 0 0 0 0 0 1
75 Cathepsin B 25 123 0 6 1 0 0 10
76 Cathepsin D 104 52 0 0 0 0 0 10
77 Cathepsin K 267 226 0 27 1 0 0 20
78 Cathepsin L 269 142 0 6 0 0 0 19
79 Cathepsin S 257 150 0 13 0 0 0 18
80 Cathepsin V 2 0 0 0 0 0 0 1
81 cFMS Tyrosine Kinase 0 21 0 0 0 0 0 3
82 cGMP-Dependent Protein Kinase 0 23 0 0 0 0 0 2
83 Checkpoint Kinase (Chk1) 6 178 0 0 0 0 0 10
84 Chitinase 3 10 25 0 0 0 0 2
85 Cholecystokinin-1 Receptor 12 0 1 3 4 0 0 1
86 Cholecystokinin-2 Receptor 16 0 1 13 0 0 0 1
87 Chymase 2 0 0 0 0 0 0 1
88 Chymotrypsin 2 0 0 0 0 0 0 1
89 cIAP1-BIR3 3 0 0 0 0 0 0 1
90 cIAP2-BIR3 3 0 0 0 0 0 0 1
91 Collagenase (ChC) 187 0 0 0 0 0 0 3
92 Conantokin-G 0 0 0 0 0 6 0 1
93 Conantokin-T 0 0 0 0 0 4 0 1
94 Corticotropin-releasing Factor Receptor 1 0 61 0 0 0 0 0 3
95 cPLA2 C2 0 0 0 0 0 1 0 1
96 CSF1-R 0 4 0 0 0 0 0 1
97 Cyclin-Dependent Kinase 1 (CDK1) 32 854 0 0 61 0 0 56
98 Cyclin-Dependent Kinase 2 (CDK2) 81 1502 0 0 65 0 0 70
99 Cyclin-Dependent Kinase 4 (CDK4) 74 966 0 0 2 0 0 48
100 Cyclin-Dependent Kinase 5 (CDK5) 0 294 0 0 0 0 0 16
101 Cyclin-Dependent Kinase 6 (CDK6) 0 8 0 0 0 0 0 2
102 Cyclin-Dependent Kinase 7 (CDK7) 1 24 0 0 0 0 0 4
103 Cyclin-Dependent Kinase 9 (CDK9) 1 6 0 0 0 0 0 3
104 Cytochrome P450 1A2 0 1 0 0 0 0 0 1
105 Cytochrome P450 2A6 30 1 0 0 0 0 0 2
106 Cytochrome P450 2B4 0 0 0 0 0 4 0 1
107 Cytochrome P450 2C19 0 1 0 0 0 0 0 1
108 Cytochrome P450 2C9 0 21 0 0 1 0 0 2
109 Cytochrome P450 2D6 0 1 0 0 0 0 0 1
110 Cytochrome P450 3A4 30 22 0 0 0 0 0 3
111 Cytochrome P450 Reductase (CPR) 0 0 0 0 0 5 0 1
112 D1.3 Fv 0 0 0 0 0 0 6 2
113 D1.3 mAb 0 0 0 0 0 0 2 2
114 D11.15 Fab 0 0 0 0 0 0 2 1
115 D11.15 Fv 0 0 0 0 0 0 1 1
116 D11.15 mAb 0 0 0 0 0 0 2 1
117 D44.1 Fab 0 0 0 0 0 0 3 1
118 D44.1 mAb 0 0 0 0 0 0 4 1
119 Delta Opioid Receptor 71 0 3 43 0 0 0 6
120 Diacyl Glycerolacyltransferase I (DGAT-1) 0 25 0 0 0 0 0 1
121 Dihydrofolate Reductase (DHFR) 26 416 0 6 1 0 0 16
122 Dihydrofolate Reductase-Thymidylate Synthase (DHFR-TS) 46 47 0 0 0 0 0 2
123 Dihydroorotate Dehydrogenase (DHODH) 37 118 0 0 0 0 0 7
124 Dipeptidyl Peptidase IV (DPP-IV) 254 492 0 0 2 0 0 30
125 Dipeptidyl Peptidase VII (DPP-VII) (QPP) 0 381 0 0 0 0 0 14
126 DNA 0 0 0 0 0 0 3 1
127 DNA (D12CA) 0 0 0 0 0 0 1 1
128 DNA (D12CC) 0 0 0 0 0 0 1 1
129 DNA (D12CG) 0 0 0 0 0 0 1 1
130 DNA (D12CT) 0 0 0 0 0 0 1 1
131 DNA (D9AA) 0 0 0 0 0 0 1 1
132 DNA (D9AC) 0 0 0 0 0 0 1 1
133 DNA (D9AG) 0 0 0 0 0 0 1 1
134 DNA (D9AT) 0 0 0 0 0 0 5 1
135 DNA Gyrase 0 5 0 0 0 4 0 2
136 DNA Polymerase alpha 2 0 0 0 0 0 0 1
137 DNA Polymerase gamma 2 0 0 0 0 0 0 1
138 DNA polymerase IIIC 2 0 0 0 0 0 0 1
139 DNA polymerase IIIE 4 0 0 0 0 0 0 1
140 DNA Topoisomerase IV 0 5 0 0 0 0 0 1
141 DNA(calf thymus) 0 0 0 0 0 2 0 1
142 Dopamine Receptor D2 24 0 1 0 0 0 0 1
143 DPP8 38 362 0 0 0 0 0 20
144 DPP9 30 245 0 0 0 0 0 13
145 DYRK1A 0 3 0 0 0 0 0 1
146 EGF-R Tyrosine Kinase 39 1053 0 0 2 0 0 38
147 Endothelin-Converting Enzyme 1 29 0 0 0 0 0 0 1
148 Enoyl-ACP Reductase (FabI) 0 161 0 0 0 22 0 5
149 Enoyl-ACP Reductase (FabK) 0 5 0 0 0 0 0 1
150 Enoyl-ACP Reductase (InhA) 6 70 0 0 3 0 0 2
151 ERK-2 33 12 0 0 0 0 0 4
152 Estrogen Receptor (ER-alpha) 43 129 0 99 14 0 0 13
153 Estrogen Receptor (ER-beta) 43 138 0 116 4 0 0 13
154 F9.13.7 Fab 0 0 0 0 0 0 4 1
155 F9.13.7 mAb 0 0 0 0 0 0 4 1
156 Factor IXa (fIXa) 92 0 0 0 0 0 0 6
157 Factor VIIa (fVIIa) 145 108 0 0 0 0 0 13
158 Factor Xa (fXa) 977 62 0 0 0 0 0 47
159 Factor XIa (fXIa) 3 31 0 0 0 0 0 2
160 FAD-Binding Domain 0 0 0 0 0 1 0 1
161 Falcipain-2 0 10 0 0 0 0 0 1
162 Farnesoid X-Activated Receptor 0 0 0 23 0 0 0 2
163 Farnesyl Diphosphate Synthase (FPPS) 0 0 0 0 0 11 0 1
164 ferricytochrome c peroxidase (CcP) 0 0 0 0 0 0 13 1
165 FGFR-1 Tyrosine Kinase 0 549 0 0 8 0 0 21
166 FGFR-2 Tyrosine Kinase 0 10 0 0 0 0 0 3
167 Fibroblast Activation Protein (FAP) 0 18 0 0 0 0 0 1
168 FLT3 1 44 0 0 0 0 0 5
169 Formyl Peptide Receptor-Like 1 0 0 0 18 0 0 0 1
170 Galectin-1 0 0 14 0 0 0 0 1
171 Galectin-3 0 0 23 0 0 0 0 2
172 Galectin-7 0 0 12 0 0 0 0 1
173 Galectin-8 0 0 11 0 0 0 0 1
174 Galectin-9 0 0 12 0 0 0 0 1
175 Geranylgeranyl Transferase (GGTase-I) 0 101 0 0 1 0 0 7
176 Ghrelin Receptor (Growth Hormone Secretagogue Receptor Type 1) 0 111 17 95 0 0 0 4
177 Glucocerebrosidase (Acid beta-Glucosidase) 30 76 0 0 0 0 0 4
178 Glucocorticoid Receptor (GR) 13 127 0 66 0 0 0 7
179 Glutamate Carboxypeptidase II (GCPII) 0 42 0 0 0 0 0 4
180 Glutaminyl Cyclase 90 0 0 0 0 0 0 3
181 Glycogen Synthase Kinase-3 19 726 0 0 0 0 0 32
182 Glyoxylate Regulatory Protein (C-AllR) 0 0 0 0 0 1 0 1
183 GRB2 0 15 0 0 0 0 0 1
184 Grb2-SH2 0 0 0 0 0 0 10 1
185 Guanylyl Cyclase C receptor mAb 0 0 0 0 0 0 22 1
186 HCV NS3-NS4A Serine Proteinase 215 0 0 0 0 0 0 10
187 Heat Shock Protein 90 (Hsp90) 0 119 0 136 0 0 0 9
188 Hepsin 6 0 0 0 0 0 0 1
189 HER-2 (erbB-2) 0 84 0 0 0 0 0