| Target Name | Protein/Small Molecule | Other | Articles | UniProtKB/ Swiss-Prot/TrEMBL |
Ki Data | IC50 Data | Kd Data | EC50 Data | other | ITC Data |
| 1 |
11-beta-Hydroxysteroid Dehydrogenase 1 (11-beta-HSD1) |
58
|
190
|
0
|
45
|
10
|
0
|
0
|
8
|
8 |
| 2 |
11-beta-Hydroxysteroid Dehydrogenase 2 (11-beta-HSD2) |
0
|
53
|
0
|
0
|
0
|
0
|
0
|
3
|
3 |
| 3 |
15-Lipoxygenase |
0
|
115
|
0
|
0
|
0
|
0
|
0
|
3
|
1 |
| 4 |
17-beta-Hydroxysteroid Dehydrogenase 1 (17-beta-HSD1) |
2
|
28
|
0
|
0
|
15
|
0
|
0
|
2
|
3 |
| 5 |
17-beta-Hydroxysteroid Dehydrogenase 2 (17-beta-HSD2) |
0
|
16
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 6 |
17-beta-Hydroxysteroid Dehydrogenase 5 (17-beta-HSD5, AKR1C3) |
6
|
3
|
0
|
0
|
0
|
0
|
0
|
3
|
2 |
| 7 |
20-alpha-Hydroxysteroid Dehydrogenase (AKR1C1) |
5
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 8 |
2C-methyl-D-erythritol-2,4-cyclodiphosphate synthase (IspF) |
0
|
0
|
6
|
0
|
3
|
0
|
0
|
1
|
40 |
| 9 |
2S-ScamLA |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 10 |
3-alpha-Hydroxysteroid Dehydrogenase Type 1 (AKR1C4) |
1
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 11 |
3-alpha-Hydroxysteroid Dehydrogenase Type 3 (AKR1C2) |
1
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 12 |
3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) |
0
|
149
|
0
|
0
|
0
|
0
|
0
|
8
|
5 |
| 13 |
3S-ScamLA |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 14 |
5-Lipoxygenase |
0
|
87
|
0
|
54
|
7
|
0
|
0
|
4
|
3 |
| 15 |
Ab N1G9 |
0
|
0
|
0
|
0
|
0
|
4
|
0
|
1
|
3 |
| 16 |
Abhydrolase Domain-Containing Protein 6 |
0
|
1
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 17 |
ABL |
0
|
44
|
83
|
0
|
0
|
0
|
0
|
45
|
4 |
| 18 |
Acetate Operon Repressor (C-IclR) |
0
|
0
|
0
|
0
|
0
|
2
|
0
|
1
|
34 |
| 19 |
Acetate Operon Repressor (IclR) |
0
|
0
|
0
|
0
|
0
|
2
|
0
|
1
|
0
|
| 20 |
Acetylcholinesterase (AChE) |
200
|
808
|
0
|
0
|
0
|
0
|
0
|
44
|
8 |
| 21 |
Activated Protein C (APC) |
1
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
5 |
| 22 |
Acyl Cholesterol Acyltransferase 1 (ACAT-1) |
0
|
7
|
0
|
0
|
0
|
0
|
0
|
1
|
6 |
| 23 |
ADAMTS-4 (Aggrecanase-1) |
0
|
28
|
0
|
0
|
2
|
0
|
0
|
3
|
2 |
| 24 |
ADAMTS-5 (Aggrecanase-2) |
0
|
57
|
0
|
0
|
8
|
0
|
0
|
2
|
1 |
| 25 |
Adenosine A3 Receptor |
27
|
0
|
0
|
4
|
2
|
0
|
0
|
1
|
2 |
| 26 |
Adenosine Deaminase |
56
|
0
|
0
|
0
|
3
|
0
|
0
|
6
|
2 |
| 27 |
Adenosine Kinase (AK) |
0
|
8
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 28 |
Adenosine Phosphosulfate Reductase (APSR) |
0
|
0
|
10
|
0
|
0
|
0
|
0
|
1
|
8 |
| 29 |
Adenosine Receptor A1 |
164
|
0
|
0
|
0
|
10
|
0
|
0
|
6
|
2 |
| 30 |
Adenosine Receptor A2A |
168
|
0
|
3
|
0
|
15
|
0
|
0
|
5
|
10 |
| 31 |
Adenosine Receptor A2B |
7
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 32 |
Adenosine Receptor A3 |
7
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 33 |
AICAR Tfase |
14
|
6
|
0
|
0
|
0
|
0
|
0
|
3
|
3 |
| 34 |
Aldehyde Reductase (ALR1) |
0
|
40
|
0
|
0
|
0
|
0
|
0
|
1
|
3 |
| 35 |
Aldose Reductase (ALR2) |
39
|
130
|
0
|
0
|
1
|
12
|
0
|
8
|
0
|
| 36 |
Aldosterone Synthase (CYP11B2) |
4
|
99
|
0
|
0
|
11
|
0
|
0
|
7
|
2 |
| 37 |
Alpha-1 Adrenergic Receptor |
12
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 38 |
alpha-Amylase |
0
|
8
|
0
|
0
|
12
|
0
|
0
|
1
|
3 |
| 39 |
alpha-Carbonic Anhydrase |
17
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 40 |
alpha-Chymotrypsin |
1
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 41 |
alpha-Glucosidase (alpha-Glu) |
0
|
35
|
0
|
0
|
0
|
0
|
0
|
2
|
4 |
| 42 |
alpha-Methylacyl-CoA Racemase |
10
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 43 |
Alpha2 Adrenoreceptor |
4
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 44 |
Aminopeptidase M |
6
|
13
|
0
|
0
|
27
|
0
|
0
|
2
|
1 |
| 45 |
Androgen Receptor (AR) |
254
|
126
|
0
|
173
|
0
|
0
|
0
|
18
|
2 |
| 46 |
Angiotensin-Converting Enzyme |
33
|
6
|
0
|
0
|
0
|
0
|
0
|
3
|
5 |
| 47 |
Angiotensin-Converting Enzyme 2 |
23
|
13
|
0
|
0
|
0
|
0
|
0
|
2
|
2 |
| 48 |
Anthrax Lethal Factor (LF) |
54
|
214
|
0
|
0
|
0
|
0
|
0
|
8
|
10 |
| 49 |
apocytochrome b562 |
0
|
0
|
0
|
0
|
0
|
2
|
0
|
1
|
9 |
| 50 |
Apoptosis Regulator Bcl-2 |
52
|
10
|
0
|
52
|
0
|
0
|
0
|
2
|
3 |
| 51 |
Apoptosis Regulator Bcl-xL |
92
|
72
|
6
|
130
|
10
|
0
|
0
|
6
|
6 |
| 52 |
Apurinic-Apyrimidinic Endonuclease 1 (APE1) |
2
|
39
|
0
|
0
|
8
|
0
|
0
|
2
|
2 |
| 53 |
Aromatase (CYP19) |
74
|
393
|
0
|
0
|
20
|
0
|
0
|
21
|
3 |
| 54 |
Aryl Hydrocarbon Receptor (AhR) |
25
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 55 |
Asparaginyl Endopeptidase (AE) |
0
|
86
|
0
|
0
|
3
|
0
|
0
|
1
|
3 |
| 56 |
ATP Phosphoribosyltransferase |
0
|
7
|
0
|
0
|
4
|
0
|
0
|
1
|
10 |
| 57 |
ATP-Binding Cassette Transporter ABCG2 |
0
|
19
|
0
|
0
|
2
|
0
|
0
|
2
|
1 |
| 58 |
Aurora Kinase A (Aurora-A) |
60
|
268
|
11
|
0
|
1
|
0
|
0
|
58
|
10 |
| 59 |
Aurora Kinase B (Aurora-B) |
38
|
48
|
13
|
0
|
1
|
0
|
0
|
49
|
1 |
| 60 |
Aurora Kinase C (Aurora-C) |
1
|
0
|
18
|
0
|
0
|
0
|
0
|
41
|
2 |
| 61 |
AXL Receptor Tyrosine Kinase |
0
|
0
|
16
|
0
|
0
|
0
|
0
|
40
|
0
|
| 62 |
B-Raf Protein Kinase |
3
|
201
|
17
|
12
|
0
|
0
|
0
|
9
|
5 |
| 63 |
Bacterial Leucyl Aminopeptidase |
4
|
15
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 64 |
Bacteriophage T4 DNA Ligase |
0
|
7
|
0
|
0
|
0
|
0
|
0
|
2
|
1 |
| 65 |
Bak |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 66 |
Beta-1 Adrenergic Receptor |
0
|
0
|
25
|
0
|
0
|
0
|
0
|
1
|
4 |
| 67 |
Beta-2 Adrenergic Receptor |
13
|
6
|
25
|
6
|
0
|
0
|
0
|
3
|
1 |
| 68 |
Beta-3 Adrenergic Receptor |
0
|
0
|
25
|
0
|
0
|
0
|
0
|
1
|
1 |
| 69 |
beta-Carbonic Anhydrase |
37
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 70 |
beta-Hydroxyacyl-Acyl Carrier Protein Dehydratase (FabZ) |
0
|
16
|
0
|
0
|
37
|
0
|
0
|
1
|
1 |
| 71 |
beta-Ketoacyl-ACP Synthase III (FabH) |
0
|
58
|
0
|
0
|
0
|
0
|
0
|
1
|
22 |
| 72 |
beta-Secretase (BACE-1) |
53
|
371
|
0
|
0
|
4
|
0
|
0
|
33
|
8 |
| 73 |
beta-Secretase (BACE-2) |
12
|
112
|
0
|
0
|
0
|
0
|
0
|
9
|
4 |
| 74 |
Bfl-1 |
0
|
8
|
0
|
198
|
0
|
0
|
0
|
2
|
3 |
| 75 |
Bfl-1 |
0
|
44
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 76 |
Bid (34-mer) |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 77 |
Bim |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 78 |
Biotin Carboxylase |
0
|
14
|
0
|
0
|
0
|
0
|
0
|
1
|
18 |
| 79 |
BirA Bifunctional Protein |
0
|
0
|
0
|
0
|
0
|
16
|
0
|
2
|
5 |
| 80 |
Bmf |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 81 |
Bone Morphogenetic Protein Receptor type II (BMPR2) |
0
|
0
|
6
|
0
|
0
|
0
|
0
|
40
|
4 |
| 82 |
Botulinum Neurotoxin Type A |
0
|
123
|
0
|
0
|
10
|
0
|
0
|
7
|
4 |
| 83 |
Butyrylcholinesterase (BuChE) |
180
|
451
|
0
|
0
|
0
|
0
|
0
|
33
|
5 |
| 84 |
C-Raf Protein Kinase |
0
|
34
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 85 |
Calcium-Sensing Receptor (CaSR) |
0
|
44
|
0
|
0
|
0
|
0
|
0
|
1
|
5 |
| 86 |
Calpain-1 |
11
|
10
|
0
|
0
|
0
|
0
|
0
|
2
|
10 |
| 87 |
Calpain-2 |
0
|
10
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 88 |
CaM Kinase II |
0
|
42
|
0
|
0
|
0
|
0
|
0
|
3
|
6 |
| 89 |
CAM-alpha-lactalbumin |
0
|
0
|
0
|
0
|
0
|
4
|
0
|
1
|
1 |
| 90 |
CAM-BPTI |
0
|
0
|
0
|
0
|
0
|
5
|
0
|
1
|
1 |
| 91 |
CAM-RNase A |
0
|
0
|
0
|
0
|
0
|
4
|
0
|
1
|
2 |
| 92 |
cAMP-Dependent Protein Kinase (PKA) |
5
|
423
|
27
|
0
|
0
|
0
|
0
|
35
|
5 |
| 93 |
cAMP-Dependent Protein Kinase (PKA) PKAR1 (1) |
0
|
5
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 94 |
cAMP-Dependent Protein Kinase (PKA) PKAR1 (2) |
0
|
5
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 95 |
cAMP-Dependent Protein Kinase (PKA) PKAR1 (3) |
0
|
5
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 96 |
cAMP-Dependent Protein Kinase (PKA) PKAR1 (4) |
0
|
5
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 97 |
cAMP-Dependent Protein Kinase (PKA) PKAR2 (1) |
0
|
5
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 98 |
cAMP-Dependent Protein Kinase (PKA) PKAR2 (2) |
0
|
1
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 99 |
cAMP-Dependent Protein Kinase (PKA) PKAR2 (3) |
0
|
3
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 100 |
cAMP-Dependent Protein Kinase (PKA) PKAR3 |
0
|
5
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 101 |
cAMP-Dependent Protein Kinase (PKA) PKAR3 (1) |
0
|
5
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 102 |
cAMP-Dependent Protein Kinase (PKA) PKAR4 |
0
|
5
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 103 |
cAMP-Dependent Protein Kinase (PKA) PKAR5 |
0
|
5
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 104 |
Cannabinoid Receptor 1 |
153
|
19
|
0
|
13
|
0
|
0
|
0
|
7
|
9 |
| 105 |
Cannabinoid Receptor 2 |
127
|
0
|
0
|
54
|
5
|
0
|
0
|
5
|
2 |
| 106 |
Carbonic Anhydrase (hpCA) |
47
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 107 |
Carbonic Anhydrase (mtCA 1) |
37
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
10 |
| 108 |
Carbonic Anhydrase (mtCA 3) |
37
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
10 |
| 109 |
Carbonic Anhydrase 2 (Can2) |
37
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 110 |
Carbonic Anhydrase I |
449
|
5
|
5
|
0
|
0
|
0
|
0
|
23
|
1 |
| 111 |
Carbonic Anhydrase II |
530
|
79
|
28
|
0
|
0
|
0
|
0
|
33
|
2 |
| 112 |
Carbonic Anhydrase III |
49
|
0
|
0
|
0
|
0
|
0
|
0
|
6
|
1 |
| 113 |
Carbonic Anhydrase IV |
243
|
24
|
0
|
0
|
0
|
0
|
0
|
15
|
3 |
| 114 |
Carbonic Anhydrase IX |
260
|
5
|
0
|
0
|
0
|
0
|
0
|
18
|
1 |
| 115 |
Carbonic Anhydrase VA |
149
|
0
|
0
|
0
|
0
|
0
|
0
|
10
|
3 |
| 116 |
Carbonic Anhydrase VB |
103
|
0
|
0
|
0
|
0
|
0
|
0
|
9
|
4 |
| 117 |
Carbonic Anhydrase VI |
85
|
0
|
0
|
0
|
0
|
0
|
0
|
7
|
3 |
| 118 |
Carbonic Anhydrase VII |
52
|
0
|
0
|
0
|
0
|
0
|
0
|
7
|
2 |
| 119 |
Carbonic Anhydrase XII |
69
|
0
|
0
|
0
|
0
|
0
|
0
|
8
|
1 |
| 120 |
Carbonic Anhydrase XIII |
51
|
0
|
0
|
0
|
0
|
0
|
0
|
7
|
1 |
| 121 |
Carbonic Anhydrase XIV |
53
|
0
|
0
|
0
|
0
|
0
|
0
|
7
|
2 |
| 122 |
Carbonic Anhydrase XV |
73
|
0
|
0
|
0
|
0
|
0
|
0
|
3
|
2 |
| 123 |
Carboxylesterase 1 |
271
|
0
|
0
|
0
|
0
|
0
|
0
|
4
|
5 |
| 124 |
Carboxylesterase 2 (intestine, liver) |
146
|
0
|
0
|
0
|
0
|
0
|
0
|
4
|
1 |
| 125 |
Carboxypeptidase A (CPA) |
7
|
8
|
0
|
0
|
0
|
0
|
0
|
2
|
1 |
| 126 |
Casein Kinase I |
0
|
13
|
0
|
0
|
0
|
0
|
0
|
4
|
20 |
| 127 |
Casein Kinase II |
38
|
7
|
0
|
0
|
0
|
0
|
0
|
6
|
10 |
| 128 |
Caspase-1 |
48
|
97
|
0
|
0
|
0
|
0
|
0
|
10
|
4 |
| 129 |
Caspase-2 |
17
|
7
|
0
|
0
|
0
|
0
|
0
|
3
|
5 |
| 130 |
Caspase-3 |
102
|
304
|
0
|
0
|
2
|
8
|
0
|
17
|
3 |
| 131 |
Caspase-3|IST-1 Complex |
7
|
0
|
0
|
0
|
0
|
9
|
0
|
1
|
3 |
| 132 |
Caspase-4 |
17
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
4 |
| 133 |
Caspase-5 |
9
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
4 |
| 134 |
Caspase-6 |
17
|
58
|
0
|
0
|
0
|
0
|
0
|
5
|
1 |
| 135 |
Caspase-7 |
18
|
114
|
0
|
0
|
0
|
0
|
0
|
8
|
5 |
| 136 |
Caspase-8 |
19
|
113
|
0
|
0
|
0
|
0
|
0
|
8
|
2 |
| 137 |
Caspase-9 |
8
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
5 |
| 138 |
Cathepsin B |
25
|
147
|
0
|
6
|
1
|
0
|
0
|
11
|
3 |
| 139 |
Cathepsin B |
0
|
56
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 140 |
Cathepsin B-Like Cysteine Protease (TbcatB) |
0
|
56
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 141 |
Cathepsin D |
104
|
155
|
0
|
0
|
35
|
0
|
0
|
17
|
1 |
| 142 |
Cathepsin K |
267
|
261
|
0
|
27
|
1
|
0
|
0
|
22
|
5 |
| 143 |
Cathepsin L |
269
|
177
|
0
|
6
|
0
|
0
|
0
|
21
|
6 |
| 144 |
Cathepsin L2 |
0
|
24
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 145 |
Cathepsin S |
257
|
213
|
0
|
13
|
0
|
0
|
0
|
21
|
6 |
| 146 |
Cathepsin V |
2
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 147 |
Cdc7 Kinase |
16
|
101
|
0
|
0
|
0
|
0
|
0
|
3
|
2 |
| 148 |
Cell Division Cycle 2-Like 1(CDC2L1) |
0
|
0
|
7
|
0
|
0
|
0
|
0
|
40
|
2 |
| 149 |
Cell Division Cycle 2-Like 2 (CDC2L2) |
0
|
0
|
7
|
0
|
0
|
0
|
0
|
40
|
1 |
| 150 |
Cell Division Cycle 2-Like 6 (CDK11) |
0
|
0
|
11
|
0
|
0
|
0
|
0
|
40
|
3 |
| 151 |
cGMP-Dependent Protein Kinase |
0
|
23
|
0
|
0
|
0
|
0
|
0
|
2
|
3 |
| 152 |
Checkpoint Kinase (Chk1) |
6
|
188
|
0
|
0
|
13
|
0
|
0
|
12
|
2 |
| 153 |
Checkpoint Kinase (Chk2) |
0
|
15
|
0
|
0
|
0
|
0
|
0
|
2
|
5 |
| 154 |
Chitinase |
3
|
10
|
25
|
0
|
0
|
0
|
0
|
2
|
6 |
| 155 |
Cholecystokinin-1 Receptor |
12
|
0
|
1
|
3
|
4
|
0
|
0
|
1
|
2 |
| 156 |
Cholecystokinin-2 Receptor |
16
|
0
|
1
|
13
|
0
|
0
|
0
|
1
|
1 |
| 157 |
Chymase |
2
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
4 |
| 158 |
Chymotrypsin |
2
|
24
|
0
|
0
|
3
|
0
|
0
|
2
|
2 |
| 159 |
cIAP-1 BIR3 |
10
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
5 |
| 160 |
cIAP-2 BIR3 |
10
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
1 |
| 161 |
cIAP1-BIR3 |
5
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
0
|
| 162 |
cIAP2-BIR3 |
3
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 163 |
CLK1 |
0
|
0
|
16
|
0
|
0
|
0
|
0
|
40
|
3 |
| 164 |
CLK4 |
0
|
0
|
13
|
0
|
0
|
0
|
0
|
40
|
5 |
| 165 |
Collagenase (ChC) |
187
|
0
|
0
|
0
|
0
|
0
|
0
|
3
|
1 |
| 166 |
Conantokin-G |
0
|
0
|
0
|
0
|
0
|
6
|
0
|
1
|
0
|
| 167 |
Conantokin-T |
0
|
0
|
0
|
0
|
0
|
4
|
0
|
1
|
0
|
| 168 |
Corticotropin-releasing Factor Receptor 1 |
0
|
135
|
0
|
0
|
0
|
0
|
0
|
5
|
2 |
| 169 |
cPLA2 C2 |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
1 |
| 170 |
Cyclin-Dependent Kinase 1 (CDK1) |
32
|
883
|
0
|
0
|
66
|
0
|
0
|
64
|
3 |
| 171 |
Cyclin-Dependent Kinase 2 (CDK2) |
103
|
1596
|
0
|
0
|
67
|
0
|
0
|
78
|
0
|
| 172 |
Cyclin-Dependent Kinase 4 (CDK4) |
74
|
967
|
0
|
0
|
2
|
0
|
0
|
49
|
0
|
| 173 |
Cyclin-Dependent Kinase 5 (CDK5) |
0
|
303
|
0
|
0
|
0
|
0
|
0
|
20
|
0
|
| 174 |
Cyclin-Dependent Kinase 6 (CDK6) |
0
|
8
|
0
|
0
|
0
|
0
|
0
|
2
|
0
|
| 175 |
Cyclin-Dependent Kinase 7 (CDK7) |
1
|
28
|
12
|
0
|
0
|
0
|
0
|
45
|
0
|
| 176 |
Cyclin-Dependent Kinase 8 (CDK8) |
0
|
0
|
8
|
0
|
0
|
0
|
0
|
40
|
1 |
| 177 |
Cyclin-Dependent Kinase 9 (CDK9) |
1
|
12
|
6
|
0
|
0
|
0
|
0
|
45
|
0
|
| 178 |
Cyclooxygenase-1 |
0
|
71
|
0
|
0
|
0
|
0
|
0
|
4
|
1 |
| 179 |
Cyclooxygenase-2 |
0
|
75
|
0
|
0
|
0
|
0
|
0
|
4
|
4 |
| 180 |
Cytochrome P450 1A2 |
0
|
1
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 181 |
Cytochrome P450 2A6 |
30
|
1
|
0
|
0
|
0
|
0
|
0
|
2
|
1 |
| 182 |
Cytochrome P450 2B4 |
0
|
0
|
0
|
0
|
0
|
4
|
0
|
1
|
0
|
| 183 |
Cytochrome P450 2C19 |
0
|
8
|
0
|
0
|
0
|
0
|
0
|
2
|
1 |
| 184 |
Cytochrome P450 2C9 |
0
|
28
|
0
|
0
|
1
|
0
|
0
|
3
|
3 |
| 185 |
Cytochrome P450 2D6 |
0
|
8
|
0
|
0
|
0
|
0
|
0
|
2
|
2 |
| 186 |
Cytochrome P450 2E1 |
0
|
9
|
0
|
0
|
0
|
0
|
0
|
1
|
3 |
| 187 |
Cytochrome P450 3A1 |
0
|
11
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 188 |
Cytochrome P450 3A4 |
30
|
61
|
0
|
0
|
0
|
0
|
0
|
6
|
4 |
| 189 |
Cytochrome P450 51(CYP51) |
0
|
0
|
28
|
0
|
0
|
0
|
0
|
2
|
9 |
| 190 |
Cytochrome P450 Reductase (CPR) |
0
|
0
|
0
|
0
|
0
|
5
|
0
|
1
|
2 |
| 191 |
D-Amino Acid Oxidase (DAAO) |
0
|
61
|
7
|
0
|
0
|
0
|
0
|
2
|
4 |
| 192 |
D-Aspartate Oxidase (DDO) |
0
|
23
|
0
|
0
|
0
|
0
|
0
|
1
|
3 |
| 193 |
D1.3 Fv |
0
|
0
|
0
|
0
|
0
|
6
|
0
|
2
|
0
|
| 194 |
D1.3 mAb |
0
|
0
|
0
|
0
|
0
|
2
|
0
|
2
|
0
|
| 195 |
D11.15 Fab |
0
|
0
|
0
|
0
|
0
|
2
|
0
|
1
|
0
|
| 196 |
D11.15 Fv |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 197 |
D11.15 mAb |
0
|
0
|
0
|
0
|
0
|
2
|
0
|
1
|
0
|
| 198 |
D44.1 Fab |
0
|
0
|
0
|
0
|
0
|
3
|
0
|
1
|
0
|
| 199 |
D44.1 mAb |
0
|
0
|
0
|
0
|
0
|
4
|
0
|
1
|
0
|
| 200 |
Delta Opioid Receptor |
140
|
0
|
3
|
43
|
0
|
0
|
0
|
8
|
2 |
| 201 |
Dengue Virus 1 (DENV1) NS2B-NS3 Protease |
0
|
10
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 202 |
Dengue Virus 2 (DENV2) NS2B-NS3 Protease |
5
|
10
|
7
|
0
|
0
|
0
|
0
|
2
|
0
|
| 203 |
Dengue Virus 3 (DENV3) NS2B-NS3 Protease |
0
|
10
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 204 |
Dengue Virus 4 (DENV4) NS2B-NS3 Protease |
0
|
10
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 205 |
Diacyl Glycerolacyltransferase 1 (DGAT-1) |
0
|
34
|
0
|
0
|
0
|
0
|
0
|
2
|
6 |
| 206 |
Diacyl Glycerolacyltransferase 2 (DGAT-2) |
0
|
0
|
0
|
0
|
2
|
0
|
0
|
1
|
1 |
| 207 |
Dihydrofolate Reductase (DHFR) |
26
|
597
|
0
|
6
|
1
|
0
|
0
|
20
|
119 |
| 208 |
Dihydrofolate Reductase-Thymidylate Synthase (DHFR-TS) |
21
|
22
|
0
|
0
|
0
|
0
|
0
|
2
|
6 |
| 209 |
Dihydrofolate Reductase-Thymidylate Synthase (DHFR-TS) KICB1 |
3
|
3
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 210 |
Dihydrofolate Reductase-Thymidylate Synthase (DHFR-TS) SP21 |
19
|
19
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 211 |
Dihydrofolate Reductase-Thymidylate Synthase (DHFR-TS) V1/S |
3
|
3
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 212 |
Dihydroorotate Dehydrogenase (DHODH) |
71
|
265
|
0
|
0
|
0
|
0
|
0
|
10
|
5 |
| 213 |
Dipeptidyl Peptidase IV (DPP-IV) |
254
|
492
|
0
|
0
|
1
|
0
|
0
|
30
|
5 |
| 214 |
Dipeptidyl Peptidase VII (DPP-VII) (QPP) |
0
|
381
|
0
|
0
|
0
|
0
|
0
|
14
|
2 |
| 215 |
DNA |
0
|
0
|
0
|
0
|
0
|
3
|
0
|
1
|
0
|
| 216 |
DNA (D12CA) |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 217 |
DNA (D12CC) |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 218 |
DNA (D12CG) |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 219 |
DNA (D12CT) |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 220 |
DNA (D9AA) |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 221 |
DNA (D9AC) |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 222 |
DNA (D9AG) |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 223 |
DNA (D9AT) |
0
|
0
|
0
|
0
|
0
|
5
|
0
|
1
|
0
|
| 224 |
DNA Gyrase |
44
|
5
|
0
|
0
|
0
|
4
|
0
|
3
|
7 |
| 225 |
DNA Ligase (MtuLigA) |
0
|
7
|
0
|
0
|
0
|
0
|
0
|
2
|
8 |
| 226 |
DNA Ligase I |
0
|
4
|
0
|
0
|
0
|
0
|
0
|
2
|
2 |
| 227 |
DNA Polymerase alpha |
2
|
10
|
0
|
0
|
0
|
0
|
0
|
2
|
1 |
| 228 |
DNA Polymerase beta |
0
|
10
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 229 |
DNA Polymerase gamma |
2
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
3 |
| 230 |
DNA polymerase IIIC |
2
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 231 |
DNA polymerase IIIE |
4
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
24 |
| 232 |
DNA Topoisomerase IV |
22
|
5
|
0
|
0
|
0
|
0
|
0
|
2
|
0
|
| 233 |
DNA(calf thymus) |
0
|
0
|
0
|
0
|
0
|
2
|
0
|
1
|
0
|
| 234 |
Dopamine Receptor D2 |
38
|
0
|
1
|
0
|
0
|
0
|
0
|
3
|
11 |
| 235 |
Dopamine Transporter (DAT) |
64
|
19
|
0
|
29
|
0
|
0
|
0
|
3
|
4 |
| 236 |
DPP8 |
38
|
362
|
0
|
0
|
0
|
0
|
0
|
20
|
1 |
| 237 |
DPP9 |
30
|
245
|
0
|
0
|
0
|
0
|
0
|
13
|
2 |
| 238 |
Dual Specificity Protein Phosphatase 1 |
0
|
165
|
0
|
0
|
0
|
0
|
0
|
2
|
0
|
| 239 |
DYRK1A |
0
|
3
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 240 |
EGF-R Tyrosine Kinase |
39
|
1137
|
34
|
0
|
2
|
0
|
0
|
87
|
2 |
| 241 |
Endothelin-Converting Enzyme 1 |
29
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
3 |
| 242 |
Enoyl-ACP Reductase (FabI) |
0
|
161
|
0
|
0
|
0
|
22
|
0
|
5
|
79 |
| 243 |
Enoyl-ACP Reductase (FabK) |
0
|
5
|
0
|
0
|
0
|
0
|
0
|
1
|
4 |
| 244 |
Enoyl-ACP Reductase (InhA) |
6
|
98
|
0
|
0
|
9
|
0
|
0
|
3
|
12 |
| 245 |
Enoyl-ACP Reductase (PfENR) |
0
|
28
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 246 |
Epoxide Hydrolase B (EHB) |
0
|
20
|
0
|
0
|
0
|
0
|
0
|
1
|
10 |
| 247 |
Equilibrative Nucleoside Transporter 1 (ENT1) |
33
|
33
|
0
|
0
|
47
|
0
|
0
|
1
|
3 |
| 248 |
ErbB-2 (HER2) Tyrosine Kinase |
0
|
144
|
0
|
0
|
0
|
0
|
0
|
8
|
2 |
| 249 |
ErbB-4 (HER4) Tyrosine Kinase |
0
|
9
|
0
|
0
|
0
|
0
|
0
|
1
|
4 |
| 250 |
ERK-2 |
57
|
15
|
0
|
0
|
0
|
0
|
0
|
7
|
4 |
| 251 |
ERK-8 |
0
|
0
|
9
|
0
|
0
|
0
|
0
|
40
|
1 |
| 252 |
Estrogen Receptor (ER-alpha) |
68
|
140
|
0
|
99
|
18
|
0
|
0
|
15
|
31 |
| 253 |
Estrogen Receptor (ER-beta) |
43
|
138
|
0
|
116
|
4
|
0
|
0
|
13
|
3 |
| 254 |
Estrogen-Related Receptor, alpha |
0
|
2
|
0
|
0
|
0
|
2
|
0
|
1
|
5 |
| 255 |
Estrogen-Related Receptor, gamma |
0
|
15
|
0
|
7
|
9
|
0
|
0
|
3
|
7 |
| 256 |
F9.13.7 Fab |
0
|
0
|
0
|
0
|
0
|
4
|
0
|
1
|
0
|
| 257 |
F9.13.7 mAb |
0
|
0
|
0
|
0
|
0
|
4
|
0
|
1
|
0
|
| 258 |
Factor IXa (fIXa) |
92
|
0
|
0
|
0
|
0
|
0
|
0
|
6
|
5 |
| 259 |
Factor VIIa (fVIIa) |
145
|
160
|
0
|
0
|
21
|
0
|
0
|
15
|
4 |
| 260 |
Factor Xa (fXa) |
1031
|
189
|
0
|
0
|
22
|
0
|
0
|
54
|
8 |
| 261 |
Factor XIa (fXIa) |
3
|
427
|
0
|
0
|
0
|
0
|
0
|
4
|
2 |
| 262 |
Factor XIIa (fXIIa) |
0
|
114
|
0
|
0
|
9
|
0
|
0
|
2
|
2 |
| 263 |
FAD-Binding Domain |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
2 |
| 264 |
Falcipain-2 |
0
|
30
|
0
|
0
|
0
|
0
|
0
|
2
|
2 |
| 265 |
Farnesoid X-Activated Receptor |
0
|
12
|
0
|
62
|
1
|
0
|
0
|
6
|
4 |
| 266 |
Farnesyl Diphosphate Synthase (FPPS) |
0
|
0
|
0
|
0
|
0
|
11
|
0
|
1
|
1 |
| 267 |
Fatty Acid Amide Hydrolase |
115
|
184
|
0
|
0
|
0
|
0
|
0
|
8
|
5 |
| 268 |
Fatty Acid Synthase |
5
|
38
|
0
|
0
|
3
|
0
|
0
|
3
|
1 |
| 269 |
ferricytochrome c peroxidase (CcP) |
0
|
0
|
0
|
0
|
0
|
13
|
0
|
1
|
2 |
| 270 |
FGFR-1 Tyrosine Kinase |
0
|
551
|
0
|
0
|
8
|
0
|
0
|
23
|
4 |
| 271 |
FGFR-2 Tyrosine Kinase |
0
|
10
|
0
|
0
|
0
|
0
|
0
|
3
|
8 |
| 272 |
Fibroblast Activation Protein (FAP) |
0
|
18
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 273 |
Formyl Peptide Receptor-Like 1 |
0
|
0
|
0
|
18
|
0
|
0
|
0
|
1
|
2 |
| 274 |
G-protein Coupled Receptor 40 |
0
|
0
|
0
|
52
|
0
|
0
|
0
|
2
|
1 |
| 275 |
G-protein Coupled Receptor 54 |
0
|
12
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 276 |
GABAA Receptor, alpha-1, beta-2, gamma-2 |
66
|
0
|
0
|
0
|
3
|
0
|
0
|
1
|
0
|
| 277 |
GABAA Receptor, alpha-1, beta-2, gamma-2 (Chimera) |
3
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 278 |
GABAA Receptor, alpha-1, beta-3, gamma-2 |
8
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 279 |
GABAA Receptor, alpha-2, beta-2, gamma-2 |
3
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 280 |
GABAA Receptor, alpha-2, beta-3, gamma-2 |
8
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 281 |
GABAA Receptor, alpha-3, beta-2, gamma-2 |
3
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 282 |
GABAA Receptor, alpha-3, beta-3, gamma-2 |
7
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 283 |
GABAA Receptor, alpha-4, beta-2, gamma-2 |
3
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 284 |
GABAA Receptor, alpha-4, beta-3, gamma-2 |
4
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 285 |
GABAA Receptor, alpha-5, beta-2, gamma-2 |
3
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 286 |
GABAA Receptor, alpha-5, beta-3, gamma-2 |
8
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 287 |
GABAA Receptor, alpha-6, beta-2, gamma-2 |
3
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 288 |
GABAA Receptor, alpha-6, beta-3, gamma-2 |
7
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 289 |
Galectin-1 |
0
|
0
|
14
|
0
|
0
|
0
|
0
|
1
|
2 |
| 290 |
Galectin-3 |
0
|
0
|
23
|
0
|
0
|
0
|
0
|
2
|
1 |
| 291 |
Galectin-7 |
0
|
0
|
12
|
0
|
0
|
0
|
0
|
1
|
2 |
| 292 |
Galectin-8 |
0
|
0
|
11
|
0
|
0
|
0
|
0
|
1
|
0
|
| 293 |
Galectin-9 |
0
|
0
|
12
|
0
|
0
|
0
|
0
|
1
|
5 |
| 294 |
gamma-Aminobutyric Acid Type B Receptor |
16
|
0
|
0
|
16
|
0
|
0
|
0
|
1
|
0
|
| 295 |
Gamma-Secretase |
0
|
0
|
0
|
98
|
0
|
0
|
0
|
4
|
0
|
| 296 |
GAR Tfase |
18
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
11 |
| 297 |
Gastric Inhibitory Polypeptide Receptor (GIPR) |
0
|
30
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 298 |
Geranylgeranyl Diphosphate Synthase (GGPPS) |
0
|
61
|
0
|
0
|
0
|
0
|
0
|
1
|
3 |
| 299 |
Geranylgeranyl Transferase (GGTase-I) |
0
|
101
|
0
|
0
|
1
|
0
|
0
|
7
|
1 |
| 300 |
Ghrelin Receptor (Growth Hormone Secretagogue Receptor Type 1) |
0
|
111
|
17
|
95
|
0
|
0
|
0
|
4
|
2 |
| 301 |
Glucagon Receptor |
0
|
30
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 302 |
Glucocerebrosidase (Acid beta-Glucosidase) |
30
|
76
|
0
|
0
|
0
|
0
|
0
|
4
|
2 |
| 303 |
Glucocorticoid Receptor (GR) |
13
|
127
|
0
|
66
|
0
|
0
|
0
|
7
|
9 |
| 304 |
Glucokinase |
0
|
0
|
0
|
6
|
28
|
0
|
0
|
1
|
1 |
| 305 |
Glutamate Carboxypeptidase II (GCPII) |
0
|
42
|
0
|
0
|
0
|
0
|
0
|
4
|
5 |
| 306 |
Glutaminyl Cyclase |
90
|
0
|
0
|
0
|
0
|
0
|
0
|
3
|
3 |
| 307 |
Glycogen Phosphorylase (PYGL) |
0
|
102
|
0
|
0
|
0
|
0
|
0
|
4
|
1 |
| 308 |
Glycogen Phosphorylase (PYGM) |
5
|
64
|
0
|
0
|
4
|
0
|
0
|
4
|
2 |
| 309 |
Glycogen Synthase Kinase-3, alpha |
6
|
169
|
0
|
0
|
0
|
0
|
0
|
6
|
3 |
| 310 |
Glycogen Synthase Kinase-3, beta |
37
|
588
|
0
|
0
|
0
|
0
|
0
|
29
|
4 |
| 311 |
Glyoxylate Regulatory Protein (C-AllR) |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
43 |
| 312 |
GRB2 |
0
|
15
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 313 |
Grb2-SH2 |
0
|
0
|
0
|
0
|
0
|
10
|
0
|
1
|
7 |
| 314 |
Guanylyl Cyclase C receptor mAb |
0
|
0
|
0
|
0
|
0
|
22
|
0
|
1
|
0
|
| 315 |
HCV NS3 Helicase |
0
|
6
|
0
|
0
|
6
|
0
|
0
|
1
|
0
|
| 316 |
HCV NS3-NS4A Serine Proteinase |
291
|
0
|
0
|
0
|
0
|
0
|
0
|
14
|
1 |
| 317 |
HCV NS5B Polymerase |
0
|
216
|
0
|
115
|
0
|
0
|
0
|
7
|
98 |
| 318 |
Heat Shock 70kDa Protein 1 |
0
|
50
|
8
|
0
|
0
|
0
|
0
|
2
|
5 |
| 319 |
Heat Shock Protein 90 (Hsp90) |
0
|
416
|
0
|
136
|
0
|
29
|
0
|
12
|
18 |
| 320 |
Heme Oxygenase 1 (HO-1) |
0
|
44
|
0
|
0
|
0
|
0
|
0
|
2
|
1 |
| 321 |
Heme Oxygenase 2 (HO-2) |
0
|
44
|
0
|
0
|
0
|
0
|
0
|
2
|
1 |
| 322 |
Hepsin |
6
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 323 |
hERG Potassium Channel 1 |
0
|
84
|
0
|
0
|
0
|
0
|
0
|
8
|
8 |
| 324 |
hIL-1beta |
0
|
0
|
0
|
0
|
0
|
9
|
0
|
1
|
3 |
| 325 |
Histamine H1 Receptor |
26
|
0
|
0
|
0
|
0
|
0
|
0
|
4
|
5 |
| 326 |
Histamine H2 Receptor |
6
|
0
|
0
|
0
|
0
|
0
|
0
|
3
|
7 |
| 327 |
Histamine H3 Receptor |
104
|
0
|
0
|
7
|
0
|
0
|
0
|
6
|
3 |
| 328 |
Histamine H4 Receptor |
118
|
0
|
0
|
0
|
1
|
0
|
0
|
8
|
5 |
| 329 |
Histone Deacetylase (pfHDAC-1) |
0
|
23
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 330 |
Histone Deacetylase 1 (HDAC1) |
8
|
175
|
0
|
0
|
20
|
0
|
0
|
15
|
6 |
| 331 |
Histone Deacetylase 10 (HDAC10) |
1
|
17
|
0
|
0
|
0
|
0
|
0
|
2
|
2 |
| 332 |
Histone Deacetylase 11 (HDAC11) |
0
|
1
|
0
|
0
|
0
|
0
|
0
|
1
|
9 |
| 333 |
Histone Deacetylase 2 (HDAC2) |
1
|
42
|
0
|
0
|
0
|
0
|
0
|
5
|
3 |
| 334 |
Histone Deacetylase 3 (HDAC3) |
1
|
66
|
0
|
0
|
21
|
0
|
0
|
8
|
3 |
| 335 |
Histone Deacetylase 4 (HDAC4) |
0
|
91
|
0
|
0
|
33
|
0
|
0
|
6
|
5 |
| 336 |
Histone Deacetylase 5 (HDAC5) |
0
|
5
|
0
|
0
|
1
|
0
|
0
|
2
|
3 |
| 337 |
Histone Deacetylase 6 (HDAC6) |
4
|
88
|
0
|
0
|
11
|
0
|
0
|
10
|
8 |
| 338 |
Histone Deacetylase 7 (HDAC7) |
0
|
6
|
0
|
0
|
0
|
0
|
0
|
2
|
9 |
| 339 |
Histone Deacetylase 8 (HDAC8) |
4
|
47
|
0
|
0
|
1
|
0
|
0
|
7
|
6 |
| 340 |
Histone Lysine Demethylase |
0
|
19
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 341 |
Histone-Arginine Methyltransferase CARM1 |
0
|
19
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 342 |
HIV-1 Integrase |
0
|
245
|
0
|
0
|
0
|
0
|
0
|
8
|
0
|
| 343 |
HIV-1 Nef |
0
|
0
|
0
|
0
|
0
|
5
|
0
|
1
|
13 |
| 344 |
HIV-1 Protease |
1509
|
1158
|
0
|
38
|
22
|
48
|
0
|
126
|
0
|
| 345 |
HIV-1 Protease A Subtype |
0
|
0
|
0
|
0
|
0
|
10
|
0
|
1
|
0
|
| 346 |
HIV-1 Protease AE |
14
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 347 |
HIV-1 Protease AE-P |
14
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 348 |
HIV-1 Protease B Subtype |
14
|
0
|
0
|
0
|
0
|
10
|
0
|
2
|
0
|
| 349 |
HIV-1 Protease C Subtype |
0
|
0
|
0
|
0
|
0
|
10
|
0
|
1
|
0
|
| 350 |
HIV-1 Protease (L10I,L19Q,K20R,E35D,M36I, ..) |
6
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
0
|
| 351 |
HIV-1 Protease (M46I,L63P,A71V,V82F,I84V) |
6
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
0
|
| 352 |
HIV-1 Protease K-60C |
0
|
15
|
0
|
0
|
0
|
0
|
0
|
4
|
0
|
| 353 |
HIV-1 Protease M1 |
19
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
0
|
| 354 |
HIV-1 Protease M2 |
19
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
0
|
| 355 |
HIV-1 Protease M3 |
19
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
0
|
| 356 |
HIV-1 Protease Q-60C |
0
|
11
|
0
|
0
|
0
|
0
|
0
|
4
|
0
|
| 357 |
HIV-1 Protease V-18C |
0
|
27
|
0
|
0
|
0
|
0
|
0
|
5
|
0
|
| 358 |
HIV-1 Protease V6 |
4
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 359 |
HIV-1 Protease V6(46) |
4
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 360 |
HIV-1 Protease V6(46/54/84) |
4
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 361 |
HIV-1 Protease V6(46/84) |
4
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 362 |
HIV-1 Protease V6(54) |
4
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 363 |
HIV-1 Protease V6(54/84) |
4
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 364 |
HIV-1 Protease V6(84) |
4
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 365 |
HIV-1 Protease, A-1 |
4
|
0
|
0
|
0
|
0
|
4
|
0
|
1
|
0
|
| 366 |
HIV-1 Protease, ANAM-11 |
4
|
0
|
0
|
0
|
0
|
4
|
0
|
1
|
0
|
| 367 |
HIV-1 Protease, MDR-HM |
0
|
0
|
0
|
0
|
0
|
9
|
0
|
2
|
0
|
| 368 |
HIV-1 Protease, MDR-QM |
0
|
0
|
0
|
0
|
0
|
9
|
0
|
2
|
0
|
| 369 |
HIV-1 Protease, NAM-10 |
4
|
0
|
0
|
0
|
0
|
4
|
0
|
1
|
0
|
| 370 |
HIV-1 Reverse Transcriptase |
30
|
2198
|
0
|
25
|
23
|
0
|
0
|
62
|
0
|
| 371 |
HIV-1 Reverse Transcriptase RNase H |
0
|
379
|
0
|
0
|
5
|
0
|
0
|
4
|
0
|
| 372 |
HIV-2 Protease |
16
|
7
|
0
|
0
|
0
|
0
|
0
|
7
|
0
|
| 373 |
HIV-2 Reverse Transcriptase |
0
|
3
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 374 |
HIV-2 Reverse Transcriptase RNase H |
0
|
2
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 375 |
HMG-CoA Reductase |
0
|
107
|
0
|
51
|
0
|
27
|
0
|
5
|
3 |
| 376 |
Homoisocitrate Dehydrogenase (HICDH) |
12
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
4 |
| 377 |
HyHEL-10 |
0
|
0
|
0
|
0
|
0
|
3
|
0
|
2
|
0
|
| 378 |
HyHEL-10 Fv (HD32A) |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 379 |
HyHEL-10 Fv (HD32E) |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 380 |
HyHEL-10 Fv (HD32N) |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 381 |
HyHEL-10 (AEAF) |
0
|
0
|
0
|
0
|
0
|
2
|
0
|
1
|
0
|
| 382 |
HyHEL-10 (ETKF) |
0
|
0
|
0
|
0
|
0
|
2
|
0
|
1
|
0
|
| 383 |
HyHEL-10 (HY58A) |
0
|
0
|
0
|
0
|
0
|
2
|
0
|
1
|
0
|
| 384 |
HyHEL-10 (HY58F) |
0
|
0
|
0
|
0
|
0
|
2
|
0
|
1
|
0
|
| 385 |
HyHEL-10 (SFSF) |
0
|
0
|
0
|
0
|
0
|
2
|
0
|
1
|
0
|
| 386 |
HyHEL-5 Fab |
0
|
0
|
0
|
0
|
0
|
2
|
0
|
1
|
0
|
| 387 |
HyHEL-5 |
0
|
0
|
0
|
0
|
0
|
4
|
0
|
1
|
0
|
| 388 |
I-kappa-B Kinase 1 (IKK-alpha) |
0
|
142
|
0
|
0
|
0
|
0
|
0
|
6
|
2 |
| 389 |
I-kappa-B Kinase 2 (IKK-beta) |
0
|
173
|
0
|
0
|
0
|
0
|
0
|
7
|
5 |
| 390 |
I-kappa-B Kinase 3 (IKK-epsilon) |
0
|
40
|
0
|
0
|
0
|
0
|
0
|
2
|
2 |
| 391 |
Immunophilin FKBP12 |
79
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
5 |
| 392 |
IMP Cyclohydrolase (IMPCH) |
3
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 393 |
Indoleamine 2,3-Dioxygenase |
34
|
58
|
0
|
0
|
19
|
0
|
0
|
4
|
2 |
| 394 |
Inosine Monophosphate Dehydrogenase Type 1 (IMPDH1) |
14
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
4 |
| 395 |
Inosine Monophosphate Dehydrogenase Type 2 (IMPDH2) |
14
|
26
|
0
|
23
|
0
|
0
|
0
|
2
|
3 |
| 396 |
Insulin Receptor Tyrosine Kinase (IRK) |
0
|
95
|
0
|
0
|
0
|
0
|
0
|
7
|
6 |
| 397 |
Insulin Receptor-Related Protein (INSRR) |
0
|
0
|
6
|
0
|
0
|
0
|
0
|
40
|
1 |
| 398 |
Insulin-like Growth Factor 1 Receptor (IGF-1R) |
0
|
180
|
0
|
0
|
0
|
0
|
0
|
9
|
3 |
| 399 |
Integrin alpha1beta1 |
0
|
0
|
0
|
0
|
5
|
0
|
0
|
1
|
0
|
| 400 |
Integrin alpha2beta1 |
0
|
33
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 401 |
Integrin alpha4beta1 (VLA-4) |
44
|
201
|
0
|
0
|
3
|
0
|
0
|
11
|
0
|
| 402 |
Integrin alpha4beta7 |
0
|
71
|
0
|
0
|
0
|
0
|
0
|
3
|
0
|
| 403 |
Integrin alpha5beta1 |
0
|
5
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 404 |
iso-1-cytochrome c (Cc) |
0
|
0
|
0
|
0
|
0
|
13
|
0
|
1
|
5 |
| 405 |
Kallikrein |
0
|
15
|
0
|
0
|
39
|
0
|
0
|
2
|
0
|
| 406 |
Kappa Opioid Receptor |
95
|
0
|
0
|
0
|
0
|
0
|
0
|
4
|
3 |
| 407 |
KIAA1363 |
0
|
1
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 408 |
Kinesin Spindle Protein Eg5 |
35
|
133
|
0
|
0
|
30
|
0
|
0
|
6
|
1 |
| 409 |
Kynurenine Aminotransferase 1/Glutamine Transaminase K |
0
|
2
|
0
|
0
|
0
|
0
|
0
|
1
|
5 |
| 410 |
Lactate Dehydrogenase |
3
|
68
|
0
|
0
|
0
|
0
|
0
|
2
|
11 |
| 411 |
Lck |
5
|
238
|
0
|
0
|
6
|
0
|
0
|
13
|
5 |
| 412 |
Leucine Aminopeptidase |
1
|
18
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 413 |
Leukotriene A4 Hydrolase |
3
|
114
|
0
|
0
|
0
|
0
|
0
|
3
|
3 |
| 414 |
Lipoxygenase-1 |
0
|
8
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 415 |
Liver Receptor Homolog 1 |
0
|
0
|
0
|
23
|
0
|
0
|
0
|
1
|
9 |
| 416 |
Liver X Receptor alpha (LXR-alpha) |
0
|
136
|
0
|
129
|
8
|
0
|
0
|
14
|
8 |
| 417 |
Liver X Receptor beta (LXR-beta) |
0
|
134
|
0
|
237
|
2
|
0
|
0
|
12
|
1 |
| 418 |
LNoxaB |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 419 |
Lysozyme (bobwhite quail) |
0
|
0
|
0
|
0
|
0
|
3
|
0
|
1
|
1 |
| 420 |
Lysozyme (hen egg) |
0
|
0
|
0
|
0
|
0
|
48
|
0
|
6
|
4 |
| 421 |
Lysozyme (turkey egg) |
0
|
0
|
0
|
0
|
0
|
6
|
0
|
1
|
1 |
| 422 |
Major Urinary Protein (MUP-1) |
0
|
0
|
0
|
0
|
0
|
8
|
0
|
3
|
5 |
| 423 |
Malate Dehydrogenase (pfMDH) |
0
|
8
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 424 |
Malate Dehydrogenase, cytoplasmic |
0
|
7
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 425 |
Malate Dehydrogenase, mitochondrial |
0
|
9
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 426 |
Mammalian Target of Rapamycin (mTOR) |
1
|
91
|
0
|
0
|
0
|
0
|
0
|
4
|
4 |
| 427 |
MAP Kinase Kinase 1 (MEK1) |
0
|
1
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 428 |
MAP Kinase p38 alpha |
50
|
451
|
39
|
31
|
4
|
5
|
0
|
25
|
10 |
| 429 |
MAP Kinase p38 beta |
0
|
15
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 430 |
MAP Kinase-Interacting Protein Kinase (MNK1) |
0
|
4
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 431 |
MAP-Microtubule Affinity-Regulating Kinase 3 (MARK3) |
0
|
1
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 432 |
MAP4K4 (HGK) |
0
|
1
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 433 |
MAPK-Activated Protein Kinase 2 (MK2) |
0
|
150
|
0
|
0
|
0
|
0
|
0
|
4
|
3 |
| 434 |
MAPK-Activated Protein Kinase 3 (MK3) |
0
|
4
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 435 |
MAPK-Activated Protein Kinase 5 (MK5) |
0
|
4
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 436 |
Matriptase |
68
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
1 |
| 437 |
Matrix Metalloproteinase-1 (MMP-1) |
132
|
58
|
0
|
0
|
0
|
0
|
0
|
11
|
3 |
| 438 |
Matrix Metalloproteinase-10 (MMP-10) |
0
|
4
|
0
|
0
|
0
|
0
|
0
|
2
|
0
|
| 439 |
Matrix Metalloproteinase-12 (MMP-12) |
16
|
48
|
9
|
0
|
1
|
0
|
0
|
6
|
0
|
| 440 |
Matrix Metalloproteinase-13 (MMP-13) |
51
|
170
|
0
|
0
|
0
|
0
|
0
|
16
|
4 |
| 441 |
Matrix Metalloproteinase-14 (MMP-14) |
0
|
11
|
0
|
0
|
0
|
0
|
0
|
4
|
2 |
| 442 |
Matrix Metalloproteinase-2 (MMP-2) |
157
|
66
|
0
|
0
|
0
|
0
|
0
|
16
|
3 |
| 443 |
Matrix Metalloproteinase-3 (MMP-3) |
101
|
9
|
0
|
0
|
1
|
0
|
0
|
7
|
2 |
| 444 |
Matrix Metalloproteinase-7 (MMP-7) |
25
|
4
|
0
|
0
|
0
|
0
|
0
|
7
|
2 |
| 445 |
Matrix Metalloproteinase-8 (MMP-8) |
119
|
3
|
0
|
0
|
0
|
0
|
0
|
9
|
1 |
| 446 |
Matrix Metalloproteinase-9 (MMP-9) |
131
|
34
|
0
|
0
|
0
|
0
|
0
|
12
|
2 |
| 447 |
Mcl-1 |
0
|
10
|
0
|
0
|
0
|
10
|
0
|
2
|
4 |
| 448 |
MEK Kinase 1 (MEKK1) |
0
|
1
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 449 |
Melanin-Concentrating Hormone Receptor 1 (MCH1R) |
0
|
21
|
0
|
3
|
0
|
0
|
0
|
1
|
5 |
| 450 |
Methionine Aminopeptidase (MAP) |
0
|
20
|
0
|
0
|
0
|
0
|
0
|
3
|
74 |
| 451 |
Methionine Aminopeptidase Type 1 (MetAP1) |
0
|
14
|
0
|
0
|
0
|
0
|
0
|
2
|
2 |
| 452 |
Methionine Aminopeptidase Type 2 (MetAP2) |
123
|
164
|
0
|
0
|
1
|
0
|
0
|
7
|
4 |
| 453 |
Methylthioadenosine Nucleosidase(MTAN) |
6
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
51 |
| 454 |
Methylthioadenosine Phosphorylase (MTAP) |
3
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 455 |
Mineralocorticoid Receptor (MR) |
8
|
14
|
0
|
0
|
0
|
0
|
0
|
4
|
9 |
| 456 |
Mitogen- and Stress-Activated Protein Kinase 1 (MSK1) |
0
|
15
|
0
|
0
|
0
|
0
|
0
|
2
|
3 |
| 457 |
Mitogen- and Stress-Activated Protein Kinase 2 (MSK2) |
0
|
4
|
0
|
0
|
0
|
0
|
0
|
1
|
3 |
| 458 |
Mitogen-Activated Protein Kinase 1 |
0
|
4
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 459 |
Mitogen-Activated Protein Kinase 10 (JNK3) |
39
|
59
|
0
|
0
|
0
|
0
|
0
|
7
|
9 |
| 460 |
Mitogen-Activated Protein Kinase 8 (JNK1) |
6
|
301
|
0
|
0
|
15
|
0
|
0
|
9
|
7 |
| 461 |
Mitogen-Activated Protein Kinase 9 (JNK2) |
6
|
69
|
5
|
0
|
0
|
3
|
0
|
44
|
3 |
| 462 |
Mixed Lineage Kinase 1 (MLK1) |
0
|
26
|
0
|
0
|
11
|
0
|
0
|
2
|
2 |
| 463 |
Mixed Lineage Kinase 2 (MLK2) |
0
|
8
|
0
|
0
|
0
|
0
|
0
|
2
|
1 |
| 464 |
Mixed Lineage Kinase 3 (MLK3) |
0
|
26
|
0
|
0
|
11
|
0
|
0
|
2
|
3 |
| 465 |
MKP-3 |
0
|
45
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 466 |
ML-IAP-BIR |
32
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
0
|
| 467 |
Monoamine Oxidase Type A (MAO-A) |
69
|
133
|
0
|
0
|
49
|
0
|
0
|
10
|
7 |
| 468 |
Monoamine Oxidase Type B (MAO-B) |
85
|
160
|
0
|
0
|
21
|
0
|
0
|
10
|
4 |
| 469 |
Monocarboxylate Transporter 1 |
43
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
4 |
| 470 |
Monoglyceride Lipase (MGL) |
0
|
9
|
0
|
0
|
13
|
0
|
0
|
2
|
5 |
| 471 |
MPI protein |
0
|
462
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 472 |
MRCK alpha |
0
|
5
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 473 |
Mu Opioid Receptor |
158
|
3
|
3
|
45
|
1
|
0
|
0
|
9
|
15 |
| 474 |
MurD |
0
|
28
|
0
|
0
|
9
|
0
|
0
|
1
|
19 |
| 475 |
Myosin Light-Chain Kinase |
0
|
18
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 476 |
NAD-Dependent Deacetylase Sirtuin-1 |
0
|
8
|
0
|
0
|
13
|
0
|
0
|
1
|
2 |
| 477 |
NAD-Dependent Deacetylase Sirtuin-2 |
0
|
7
|
0
|
0
|
13
|
0
|
0
|
1
|
8 |
| 478 |
Neuraminidase A |
16
|
254
|
0
|
0
|
0
|
0
|
0
|
17
|
9 |
| 479 |
Neuraminidase B |
19
|
162
|
0
|
0
|
0
|
0
|
0
|
13
|
7 |
| 480 |
Neutral Endopeptidase |
29
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 481 |
Neutrophil Elastase (NE) |
33
|
23
|
0
|
0
|
0
|
0
|
0
|
2
|
2 |
| 482 |
Niacin Receptor GPR109A |
0
|
18
|
0
|
18
|
0
|
0
|
0
|
1
|
1 |
| 483 |
Nitric Oxide Synthase, brain |
27
|
8
|
0
|
30
|
0
|
0
|
0
|
5
|
5 |
| 484 |
Nitric Oxide Synthase, endothelial |
19
|
8
|
0
|
32
|
0
|
0
|
0
|
5
|
7 |
| 485 |
Nitric Oxide Synthase, inducible |
6
|
8
|
0
|
41
|
0
|
0
|
0
|
3
|
5 |
| 486 |
NK1 Receptor |
21
|
0
|
0
|
0
|
2
|
0
|
0
|
2
|
5 |
| 487 |
Nociceptin Receptor (ORL1 Receptor) |
110
|
58
|
0
|
34
|
0
|
0
|
0
|
6
|
4 |
| 488 |
Norepinephrine Transporter (NET) |
69
|
16
|
0
|
29
|
6
|
0
|
0
|
3
|
3 |
| 489 |
NoxaA |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 490 |
NoxaB |
0
|
0
|
0
|
0
|
0
|
2
|
0
|
1
|
0
|
| 491 |
Orotidine Monophosphate Decarboxylase (ODCase) |
23
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
11 |
| 492 |
Outer Membrane Phospholipase A |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
1 |
| 493 |
Outer Membrane Phospholipase A |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 494 |
p53-Binding Protein HDMX |
0
|
24
|
0
|
0
|
1
|
0
|
0
|
1
|
4 |
| 495 |
p53-Binding Protein MDM2 |
32
|
139
|
8
|
0
|
1
|
0
|
0
|
12
|
11 |
| 496 |
Papain |
48
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 497 |
PDGFR-beta |
0
|
637
|
0
|
0
|
8
|
0
|
0
|
27
|
5 |
| 498 |
Pepsin |
6
|
20
|
0
|
0
|
0
|
0
|
0
|
3
|
3 |
| 499 |
Peptide Deformylase |
0
|
12
|
0
|
0
|
0
|
0
|
0
|
1
|
75 |
| 500 |
peptide ENIFPLE |
0
|
0
|
0
|
0
|
0
|
6
|
0
|
1
|
0
|
| 501 |
peptide HIPPEN |
0
|
0
|
0
|
0
|
0
|
7
|
0
|
1
|
0
|
| 502 |
peptide HIPPENIFPLE |
0
|
0
|
0
|
0
|
0
|
9
|
0
|
1
|
0
|
| 503 |
Peripheral-Type Benzodiazepine Receptor |
10
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 504 |
Peroxisome Proliferator-Activated Receptor alpha |
29
|
54
|
0
|
244
|
2
|
0
|
0
|
11
|
5 |
| 505 |
Peroxisome Proliferator-Activated Receptor delta |
29
|
35
|
0
|
226
|
0
|
0
|
0
|
8
|
4 |
| 506 |
Peroxisome Proliferator-Activated Receptor gamma |
32
|
75
|
3
|
229
|
0
|
0
|
0
|
12
|
5 |
| 507 |
Phenylethanolamine N-Methyltransferase (PNMT) |
31
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
3 |
| 508 |
Phosphodiesterase Type 1 (PDE1B) |
0
|
10
|
0
|
0
|
0
|
0
|
0
|
1
|
4 |
| 509 |
Phosphodiesterase Type 10 (PDE10A) |
30
|
29
|
0
|
0
|
0
|
0
|
0
|
3
|
1 |
| 510 |
Phosphodiesterase Type 11 (PDE11A) |
0
|
10
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 511 |
Phosphodiesterase Type 2 (PDE2A) |
0
|
10
|
0
|
0
|
0
|
0
|
0
|
1
|
5 |
| 512 |
Phosphodiesterase Type 3 (PDE3A) |
29
|
40
|
0
|
0
|
0
|
0
|
0
|
2
|
1 |
| 513 |
Phosphodiesterase Type 3 (PDE3B) |
29
|
52
|
0
|
0
|
0
|
0
|
0
|
4
|
2 |
| 514 |
Phosphodiesterase Type 4 (PDE4A) |
32
|
112
|
0
|
0
|
0
|
0
|
0
|
6
|
5 |
| 515 |
Phosphodiesterase Type 4 (PDE4B) |
32
|
49
|
0
|
0
|
0
|
0
|
0
|
6
|
7 |
| 516 |
Phosphodiesterase Type 4 (PDE4C) |
0
|
2
|
0
|
0
|
0
|
0
|
0
|
1
|
8 |
| 517 |
Phosphodiesterase Type 4 (PDE4D) |
92
|
47
|
0
|
0
|
0
|
0
|
0
|
6
|
5 |
| 518 |
Phosphodiesterase Type 5 (PDE5) |
0
|
26
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 519 |
Phosphodiesterase Type 5 (PDE5A) |
0
|
13
|
0
|
0
|
0
|
0
|
0
|
2
|
2 |
| 520 |
Phosphodiesterase Type 5 (PDE5A) (661-681 deletion) |
0
|
3
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 521 |
Phosphodiesterase Type 5 (PDE5A) (663-678 deletion) |
0
|
3
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 522 |
Phosphodiesterase Type 6 (PDE6) |
0
|
7
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 523 |
Phosphodiesterase Type 7 (PDE7B) |
0
|
10
|
0
|
0
|
0
|
0
|
0
|
1
|
6 |
| 524 |
Phosphodiesterase Type 8 (PDE8A) |
0
|
10
|
0
|
0
|
0
|
0
|
0
|
1
|
4 |
| 525 |
Phosphodiesterase Type 9 (PDE9A) |
0
|
10
|
0
|
0
|
0
|
0
|
0
|
1
|
4 |
| 526 |
Phosphoinositide 3-Kinase (PI3K), alpha |
0
|
142
|
0
|
0
|
0
|
0
|
0
|
9
|
3 |
| 527 |
Phosphoinositide 3-Kinase (PI3K), beta |
0
|
14
|
0
|
0
|
0
|
0
|
0
|
6
|
0
|
| 528 |
Phosphoinositide 3-Kinase (PI3K), C2beta |
0
|
7
|
0
|
0
|
0
|
0
|
0
|
3
|
5 |
| 529 |
Phosphoinositide 3-Kinase (PI3K), delta |
0
|
8
|
0
|
0
|
0
|
0
|
0
|
4
|
0
|
| 530 |
Phosphoinositide 3-Kinase (PI3K), gamma |
0
|
65
|
4
|
0
|
8
|
0
|
0
|
8
|
0
|
| 531 |
Phosphoinositide 3-Kinase (PI3K), Vps34 |
0
|
1
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 532 |
Phospholipase A2, major isoenzyme |
0
|
21
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 533 |
Phospholipase A2, membrane associated |
0
|
32
|
0
|
0
|
0
|
0
|
0
|
2
|
2 |
| 534 |
Phosphorylase Kinase |
0
|
13
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 535 |
PIM-1 Kinase |
85
|
90
|
0
|
0
|
0
|
9
|
0
|
10
|
2 |
| 536 |
PIM-2 Kinase |
80
|
62
|
0
|
0
|
0
|
0
|
0
|
5
|
2 |
| 537 |
PIM-3 Kinase |
2
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 538 |
Plasma Kallikrein |
4
|
0
|
0
|
0
|
0
|
0
|
0
|
2
|
1 |
| 539 |
Plasmepsin I |
93
|
0
|
0
|
0
|
0
|
0
|
0
|
4
|
3 |
| 540 |
Plasmepsin II |
107
|
0
|
0
|
0
|
0
|
0
|
0
|
5
|
3 |
| 541 |
Plasmepsin IV |
11
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 542 |
Plasmin |
129
|
25
|
0
|
0
|
0
|
0
|
0
|
7
|
5 |
| 543 |
PLD alpha C2 |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 544 |
PLD beta C2 |
0
|
0
|
0
|
0
|
0
|
2
|
0
|
1
|
0
|
| 545 |
PNA |
0
|
0
|
0
|
0
|
0
|
4
|
0
|
1
|
0
|
| 546 |
PNA (P9CT) |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 547 |
PNA (P9GT) |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 548 |
PNA (P9TT) |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 549 |
PNA(P9) |
0
|
0
|
0
|
0
|
0
|
5
|
0
|
1
|
0
|
| 550 |
Polo-Like Kinase 1 |
21
|
122
|
0
|
0
|
0
|
0
|
0
|
9
|
3 |
| 551 |
Polo-Like Kinase 2 |
21
|
9
|
0
|
0
|
0
|
0
|
0
|
4
|
1 |
| 552 |
Polo-Like Kinase 3 |
22
|
26
|
0
|
0
|
0
|
0
|
0
|
7
|
3 |
| 553 |
Polo-Like Kinase 4 |
21
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
3 |
| 554 |
Poly (ADP-ribose) Polymerase-1 (PARP-1) |
81
|
145
|
0
|
0
|
0
|
0
|
0
|
8
|
4 |
| 555 |
Poly (ADP-ribose) Polymerase-2 (PARP-2) |
0
|
36
|
0
|
0
|
0
|
0
|
0
|
3
|
1 |
| 556 |
PPIase Pin1 |
15
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 557 |
Pregnane X Receptor |
0
|
12
|
0
|
12
|
0
|
0
|
0
|
1
|
0
|
| 558 |
Progesterone Receptor (PR) |
16
|
62
|
0
|
0
|
0
|
0
|
0
|
7
|
14 |
| 559 |
Prokineticin Receptor 1 (PKR1) |
3
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 560 |
Prokineticin Receptor 2 (PKR2) |
3
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 561 |
Prostacyclin (IP) Receptor |
0
|
17
|
0
|
16
|
0
|
0
|
0
|
1
|
1 |
| 562 |
Prostaglandin D Synthase |
0
|
16
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 563 |
Prostaglandin D2 Receptor CRTH2 |
75
|
0
|
0
|
17
|
0
|
0
|
0
|
1
|
3 |
| 564 |
Prostanoid EP1 Receptor |
19
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 565 |
Prostanoid EP2 Receptor |
19
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 566 |
Prostanoid EP3 Receptor |
19
|
0
|
0
|
19
|
0
|
0
|
0
|
1
|
1 |
| 567 |
Prostanoid EP4 Receptor |
19
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 568 |
Protein Farnesyltransferase (PFT) |
0
|
244
|
0
|
0
|
0
|
0
|
0
|
12
|
8 |
| 569 |
Protein kinase B (Akt 1) |
30
|
429
|
0
|
0
|
17
|
0
|
0
|
20
|
4 |
| 570 |
Protein kinase B (Akt 2) |
0
|
161
|
0
|
0
|
0
|
0
|
0
|
12
|
7 |
| 571 |
Protein kinase B (Akt 3) |
0
|
69
|
0
|
0
|
0
|
0
|
0
|
8
|
1 |
| 572 |
Protein Kinase C |
0
|
162
|
0
|
0
|
0
|
0
|
0
|
6
|
0
|
| 573 |
Protein Kinase C, alpha |
1
|
138
|
0
|
0
|
0
|
0
|
0
|
10
|
5 |
| 574 |
Protein Kinase C, beta I |
0
|
49
|
0
|
0
|
0
|
0
|
0
|
4
|
2 |
| 575 |
Protein Kinase C, beta II |
0
|
94
|
0
|
0
|
0
|
0
|
0
|
5
|
3 |
| 576 |
Protein Kinase C, delta |
0
|
113
|
0
|
0
|
0
|
0
|
0
|
6
|
3 |
| 577 |
Protein Kinase C, epsilon |
0
|
100
|
0
|
0
|
0
|
0
|
0
|
6
|
5 |
| 578 |
Protein Kinase C, eta |
0
|
65
|
0
|
0
|
0
|
0
|
0
|
5
|
3 |
| 579 |
Protein Kinase C, gamma |
0
|
45
|
0
|
0
|
0
|
0
|
0
|
5
|
3 |
| 580 |
Protein Kinase C, theta |
2
|
93
|
0
|
0
|
0
|
0
|
0
|
5
|
3 |
| 581 |
Protein Kinase C, zeta |
0
|
44
|
0
|
0
|
0
|
0
|
0
|
5
|
3 |
| 582 |
Protein Kinase D1 |
0
|
30
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 583 |
Protein Kinase YpkA |
0
|
4
|
0
|
0
|
0
|
0
|
0
|
1
|
13 |
| 584 |
Protein Tyrosine Phosphatase CD45 |
1
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
5 |
| 585 |
Protein Tyrosine Phosphatase LAR |
1
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
3 |
| 586 |
Protein Tyrosine Phosphatase PTPA |
1
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
8 |
| 587 |
Protein Tyrosine Phosphatase PTPB |
5
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
7 |
| 588 |
Protein Tyrosine Phosphatase TC-PTP |
1
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
0
|
| 589 |
Protein Tyrosine Phosphatase VHR |
1
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
4 |
| 590 |
Protein-Tyrosine Phosphatase 1B (PTP1B) |
134
|
160
|
10
|
0
|
0
|
0
|
0
|
15
|
4 |
| 591 |
Protein-Tyrosine Phosphatase SHP-1 |
0
|
22
|
0
|
0
|
0
|
0
|
0
|
1
|
4 |
| 592 |
Protein-Tyrosine Phosphatase SHP-2 |
17
|
34
|
0
|
0
|
0
|
0
|
0
|
3
|
5 |
| 593 |
Pteridine Reductase 1 (PTR1) |
11
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 594 |
Puma |
0
|
0
|
0
|
0
|
0
|
2
|
0
|
1
|
0
|
| 595 |
Purine Nucleoside Phosphorylase (PNP) |
18
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
5 |
| 596 |
pY317 (phosphotyrosine polypeptide) |
0
|
0
|
0
|
0
|
0
|
5
|
0
|
1
|
0
|
| 597 |
pY317 N(+2)A |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 598 |
pY317 Q(+4)A |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 599 |
pY317 S(-1)A |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 600 |
pY317 V(+1)A |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 601 |
pY317 V(+3)A |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 602 |
Quinone Reductase 1 |
0
|
58
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 603 |
Quinone Reductase 2 (QR2) |
0
|
27
|
0
|
0
|
0
|
3
|
0
|
2
|
2 |
| 604 |
RAF-1 |
0
|
1
|
0
|
0
|
0
|
0
|
0
|
1
|
4 |
| 605 |
Receptor Tyrosine Kinase TrkA |
0
|
44
|
0
|
0
|
0
|
0
|
0
|
3
|
4 |
| 606 |
Receptor Tyrosine Kinase TrkB |
0
|
2
|
0
|
0
|
0
|
0
|
0
|
1
|
5 |
| 607 |
Renin |
2
|
230
|
0
|
0
|
0
|
11
|
0
|
12
|
3 |
| 608 |
Retinoic Acid Receptor, alpha |
0
|
0
|
8
|
0
|
2
|
0
|
0
|
1
|
5 |
| 609 |
Retinoic Acid Receptor, beta |
0
|
0
|
8
|
0
|
2
|
0
|
0
|
1
|
3 |
| 610 |
Retinoic Acid Receptor, gamma |
0
|
0
|
9
|
0
|
1
|
0
|
0
|
1
|
7 |
| 611 |
Rho Transcription Termination Factor |
0
|
0
|
0
|
0
|
0
|
3
|
0
|
1
|
50 |
| 612 |
Rho-kinase (ROCK I) |
4
|
67
|
0
|
0
|
0
|
0
|
0
|
5
|
6 |
| 613 |
Rho-kinase (ROCK II) |
0
|
12
|
8
|
0
|
0
|
0
|
0
|
3
|
0
|
| 614 |
Ribonuclease H |
0
|
2
|
0
|
0
|
0
|
0
|
0
|
1
|
35 |
| 615 |
Ribonuclease H1 |
0
|
8
|
0
|
0
|
0
|
0
|
0
|
2
|
2 |
| 616 |
Ribosomal S6 Kinase 1 (RSK-1) |
0
|
9
|
0
|
0
|
0
|
0
|
0
|
2
|
5 |
| 617 |
Ribosomal S6 Kinase 2 (RSK-2) |
0
|
1
|
0
|
0
|
0
|
0
|
0
|
1
|
7 |
| 618 |
Ribosomal S6 Kinase 3 (RSK-3) |
0
|
1
|
0
|
0
|
0
|
0
|
0
|
1
|
5 |
| 619 |
Ribosomal S6 Kinase 4 (RSK-4) |
0
|
1
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 620 |
RNA(23-mer) |
0
|
0
|
0
|
0
|
0
|
9
|
0
|
1
|
0
|
| 621 |
Runt-Related Transcription Factor 1 Isoform AML1C |
0
|
214
|
0
|
0
|
6
|
0
|
0
|
4
|
5 |
| 622 |
Runt-Related Transcription Factor 1 Isoform AML1C |
0
|
189
|
0
|
0
|
0
|
0
|
0
|
3
|
5 |
| 623 |
S-Adenosylmethionine Decarboxylase (AdoMetDC) |
0
|
24
|
0
|
0
|
10
|
0
|
0
|
1
|
3 |
| 624 |
Sarco/endoplasmic Reticulum Ca2+ ATPase 1 |
0
|
31
|
0
|
0
|
0
|
0
|
0
|
2
|
2 |
| 625 |
SARS Coronavirus 3C-like Protease |
17
|
81
|
0
|
0
|
0
|
0
|
0
|
6
|
64 |
| 626 |
SARS Coronavirus Coronavirus Papain-Like Protease |
0
|
20
|
0
|
0
|
4
|
0
|
0
|
1
|
9 |
| 627 |
sc1E3 |
0
|
0
|
0
|
0
|
0
|
9
|
0
|
1
|
0
|
| 628 |
SecB |
0
|
0
|
0
|
0
|
0
|
15
|
0
|
1
|
39 |
| 629 |
Serine Hydroxymethyltransferase |
0
|
0
|
0
|
0
|
0
|
5
|
0
|
4
|
1 |
| 630 |
Serotonin Receptor 1A |
62
|
44
|
0
|
51
|
0
|
0
|
0
|
6
|
6 |
| 631 |
Serotonin Receptor 1A |
0
|
0
|
0
|
346
|
0
|
0
|
0
|
1
|
0
|
| 632 |
Serotonin Receptor 1B |
3
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 633 |
Serotonin Receptor 1D |
3
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
2 |
| 634 |
Serotonin Receptor 1E |
0
|
75
|
0
|
51
|
0
|
0
|
0
|
3
|
3 |
| 635 |
Serotonin Receptor 2A |
57
|
15
|
0
|
0
|
1
|
0
|
0
|
3
|
10 |
| 636 |
Serotonin Receptor 2B |
4
|
0
|
0
|
0
|
1
|
0
|
0
|
3
|
14 |
| 637 |
Serotonin Receptor 2C |
5
|
0
|
0
|
0
|
0
|
0
|
0
|
3
|
10 |
| 638 |
Serotonin Receptor 4 |
7
|
0
|
0
|
8
|
1
|
0
|
0
|
1
|
4 |
| 639 |
Serotonin Receptor 6 |
105
|
3
|
0
|
20
|
3
|
0
|
0
|
5
|
2 |
| 640 |
Serotonin Receptor 7 |
64
|
0
|
0
|
0
|
0
|
0
|
0
|
5
|
4 |
| 641 |
Serotonin Transporter (SERT) |
83
|
8
|
0
|
29
|
0
|
0
|
0
|
4
|
10 |
| 642 |
single stranded DNA |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 643 |
single stranded DNA binding protein |
0
|
0
|
0
|
0
|
0
|
1
|
0
|
1
|
0
|
| 644 |
Sodium-Dependent Glucose Cotransporter 1 (SGLT1) |
0
|
0
|
0
|
5
|
0
|
0
|
0
|
1
|
4 |
| 645 |
Sodium-Dependent Glucose Cotransporter 2 (SGLT2) |
0
|
0
|
0
|
5
|
0
|
0
|
0
|
1
|
2 |
| 646 |
Sortase A (SrtA) |
0
|
113
|
0
|
0
|
0
|
0
|
0
|
1
|
21 |
| 647 |
Sphingosine 1-Phosphate Receptor 1 |
4
|
20
|
0
|
8
|
0
|
0
|
0
|
3
|
0
|
| 648 |
Sphingosine 1-Phosphate Receptor 2 |
4
|
0
|
0
|
0
|
0
|
0
|
0
|
1
|
1 |
| 649 |
Sphingosine 1-Phosphate Receptor 3 |
4
|
20
|
0
|
8
|
0
|
0
|
0
|
3
|
1 |
| 650 |
Sphingosine 1-Phosphate Receptor 4 |
4
|
19
|
0
|
0
|
0
|
0
|
0
|
2
|
1 |
| 651 |
Sphingosine 1-Phosphate Receptor 5 |
4
|
19
|
0
|
8
|
0
|
0
|
0
|
3
|
3 |
| 652 |
Src |
1
|
995
|
6
|
0
|
15
|
0
|
0
|
44
|
6 |
| 653 |
STE20-Like Kinase MST2 |
0
|
1
|
0
|
0
|
0
|
0
|
0
|
1
|
3 |
| 654 |
Steroid 11-beta-Hydroxylase (CYP11B1) |
0
|
101
|
0
|
0
|
0
|
0
|
0
|
7
|
1 |
| 655 |
Steroid 17-alpha-Monooxygenase (CYP17) |
0
|
32
|
0
|
0
|
77
|
0
|
0
|
7
|
3 |
| 656 |
Steroid Sulfatase (STS) |
0
|
41
|
0
|
0
|
4
|
0
|
0
|
4
|
0
|
| 657 |
Steroidogenic Factor 1 |
0
|
0
|
0
|
44
|
3
|
0
|
0
|
2
|
6 |
| 658 |
Streptavadin |
0
|
0
|
0
|
0
|
0
|
11
|
0
|
2
|
0
|
| 659 |
Streptavidin |
0
|
0
|
0
|
0
|
0
|
5
|
0
|
2
|
0
|
| 660 |
T-Cell Protein-Tyrosine Phosphatase (TCPTP) |
43
|
14
|
0
|
0
|
0
|
0
|
0
|
9
|
2 |
| 661 |
t-Plasminogen Activator (tPA) |
81
|
0
|
0
|
0
|
0
|
0
|
0
|
7
|
4 |
| 662 |
Tankyrase-1 |
0
|
1
|
0
|
0
|
0
|
0
|
0
|
1
|
|