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Found 59 for UniProtKB: P51050
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)
Affinity DataKi:  0.130nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50231291(CHEMBL421013)
Affinity DataKi:  0.230nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50231307(CHEMBL34622)
Affinity DataKi:  0.270nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.340nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072660(CHEMBL111866 | N-(7-Methoxy-1,2,3,4-tetrahydro-nap...)
Affinity DataKi:  0.450nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072651(CHEMBL113859 | N-(7-Methoxy-1,2,3,4-tetrahydro-nap...)
Affinity DataKi:  0.530nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072651(CHEMBL113859 | N-(7-Methoxy-1,2,3,4-tetrahydro-nap...)
Affinity DataKi:  0.530nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM85239(5-MeOT-N-propionyl)
Affinity DataKi:  0.540nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50037220(1-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-pyrrolidin...)
Affinity DataKi:  0.540nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM85239(5-MeOT-N-propionyl)
Affinity DataKi:  0.550nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.570nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50231304(CHEMBL288084)
Affinity DataKi:  0.730nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072656(CHEMBL111879 | N-(3-Methoxy-6,7,8,9-tetrahydro-5H-...)
Affinity DataKi:  1nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  1.21nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072652(CHEMBL113244 | N-(6-Methoxy-indan-1-ylmethyl)-prop...)
Affinity DataKi:  3nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072652(CHEMBL113244 | N-(6-Methoxy-indan-1-ylmethyl)-prop...)
Affinity DataKi:  3nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50231302(CHEMBL99376)
Affinity DataKi:  3.60nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50231292(CHEMBL95920)
Affinity DataKi:  3.80nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072654(CHEMBL113067 | N-(7-Methoxy-1,2,3,4-tetrahydro-nap...)
Affinity DataKi:  4nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50045843(8-M-PDOT | CHEMBL99377 | N-(8-Methoxy-1,2,3,4-tetr...)
Affinity DataKi:  7.40nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072653(CHEMBL113243 | N-(6-Methoxy-indan-1-ylmethyl)-buty...)
Affinity DataKi:  7.60nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072652(CHEMBL113244 | N-(6-Methoxy-indan-1-ylmethyl)-prop...)
Affinity DataKi:  16nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM85240(5-MeOT-N-pentanyl)
Affinity DataKi:  24.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM85240(5-MeOT-N-pentanyl)
Affinity DataKi:  24.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072661(CHEMBL111880 | N-(3-Methoxy-6,7,8,9-tetrahydro-5H-...)
Affinity DataKi:  29nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072657(CHEMBL320136 | N-(3-Methoxy-6,7,8,9-tetrahydro-5H-...)
Affinity DataKi:  34nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072658(CHEMBL114929 | N-(4-Methoxy-bicyclo[4.2.0]octa-1,3...)
Affinity DataKi:  40nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50231298(CHEMBL330385)
Affinity DataKi:  44nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50035176(8-M-ADOT | CHEMBL53015 | N-(8-Methoxy-1,2,3,4-tetr...)
Affinity DataKi:  46nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072655(CHEMBL112164 | N-(4-Methoxy-bicyclo[4.2.0]octa-1,3...)
Affinity DataKi:  49nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072659(CHEMBL111667 | N-(6-Methoxy-indan-1-ylmethyl)-acet...)
Affinity DataKi:  77nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50231294(CHEMBL95266)
Affinity DataKi:  95nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50231296(CHEMBL316854)
Affinity DataKi:  121nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50231303(CHEMBL95364)
Affinity DataKi:  141nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50231301(CHEMBL421569)
Affinity DataKi:  145nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282747(2-Bromo-N-[2-(1H-indol-3-yl)-ethyl]-acetamide | AA...)
Affinity DataKi:  153nMAssay Description:Binding affinity towards melatonin receptor using 2-[125I]iodomelatonin as radioligand in chick brain membranesMore data for this Ligand-Target Pair
In DepthDetails
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50035176(8-M-ADOT | CHEMBL53015 | N-(8-Methoxy-1,2,3,4-tetr...)
Affinity DataKi:  161nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072650(CHEMBL419939 | N-(4-Methoxy-bicyclo[4.2.0]octa-1,3...)
Affinity DataKi:  224nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50231299(CHEMBL95851)
Affinity DataKi:  312nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50231305(CHEMBL52801)
Affinity DataKi:  420nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50231306(CHEMBL53722)
Affinity DataKi:  581nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50231295(CHEMBL322193)
Affinity DataKi:  665nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50231308(CHEMBL299966)
Affinity DataKi:  748nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM85237(5-MeOT-N-hexanyl)
Affinity DataKi:  773nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM85383(Luzindole,5-MeOT-N-hexanyl)
Affinity DataKi:  776nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50231300(CHEMBL50943)
Affinity DataKi:  789nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM85384(Luzindole,N-pentanoyl)
Affinity DataKi:  933nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Chick)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072651(CHEMBL113859 | N-(7-Methoxy-1,2,3,4-tetrahydro-nap...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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