BDBM50006416 CHEMBL3234708

SMILES Cc1c2CCCCn2c(=O)c2cc(OC(=O)C(C)(C)C)cc(OC(=O)C(C)(C)C)c12

InChI Key InChIKey=PIRXZRZNBGBOKB-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50006416   

TargetCannabinoid receptor 2(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50006416(CHEMBL3234708)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]-CP55940 from rat CB2 receptor expressed in CHO-K1 cells by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50006416(CHEMBL3234708)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]-CP55940 from mouse CB2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50006416(CHEMBL3234708)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50006416(CHEMBL3234708)
Affinity DataKi:  2.63E+3nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed