BDBM50007396 4-Phenyl-1-(5-phenyl-pentyl)-piperidine::CHEMBL112474

SMILES C(CCN1CCC(CC1)c1ccccc1)CCc1ccccc1

InChI Key InChIKey=IOOPAUYHVADGIS-UHFFFAOYSA-N

Data  1 KI  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50007396   

TargetSigma non-opioid intracellular receptor 1(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50007396(CHEMBL112474 | 4-Phenyl-1-(5-phenyl-pentyl)-piperi...)
Affinity DataKi:  0.900nMAssay Description:The compound was tested for its binding affinity towards sigma receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50007396(CHEMBL112474 | 4-Phenyl-1-(5-phenyl-pentyl)-piperi...)
Affinity DataIC50: 210nMAssay Description:Compound was tested for its binding affinity towards dopamine receptor D2 by using [3H]domperidone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50007396(CHEMBL112474 | 4-Phenyl-1-(5-phenyl-pentyl)-piperi...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity determined in radioreceptor binding assay by using [3H]SCH-23390 radioligand against dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50007396(CHEMBL112474 | 4-Phenyl-1-(5-phenyl-pentyl)-piperi...)
Affinity DataIC50: 1.00E+4nMAssay Description:Compound was tested for its affinity towards PCP receptor in rat brain membrane [3H]MK-801 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed