BDBM50149701 CHEMBL3769806

SMILES CC(C)n1ncc2cc(ccc12)C(=O)NCc1c(C)cc(C)[nH]c1=O

InChI Key InChIKey=PGMGXFREQYSDRS-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50149701   

TargetHistone-lysine N-methyltransferase EZH2(Human)
Epizyme

Curated by ChEMBL
LigandPNGBDBM50149701(CHEMBL3769806)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of methyltransferase activity of human EZH2 using chicken oligonucleotide as substrate by pull down assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed