BDBM50158619 CHEMBL3785262

SMILES CN1C(=O)Nc2ccc(cc2C1(C)c1ccccc1)-c1c(C)noc1C

InChI Key InChIKey=HPNKVGAQIXCTBD-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50158619   

TargetBromodomain-containing protein 4(Human)
Genentech

Curated by ChEMBL
LigandPNGBDBM50158619(CHEMBL3785262)
Affinity DataIC50: 34nMAssay Description:Displacement of biotinylated tetra-acetylated histone H4 from His-tagged BRD4 bromodomain1 (42 to 168 residues) (unknown origin) incubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed