BDBM50172419 (E)-N-{2-[(2-Dimethylamino-ethyl)-methyl-amino]-quinolin-6-yl}-3-p-tolyl-acrylamide::CHEMBL194477

SMILES CN(C)CCN(C)c1ccc2cc(NC(=O)\C=C\c3ccc(C)cc3)ccc2n1

InChI Key InChIKey=GEGLJDPEPGLWCZ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50172419   

TargetMelanin-concentrating hormone receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50172419((E)-N-{2-[(2-Dimethylamino-ethyl)-methyl-amino]-qu...)
Affinity DataIC50: 20nMAssay Description:Displacement of 15 pM [125I]MCH from human MCH1R expressed in CHO-K1 in whole-cell binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50172419((E)-N-{2-[(2-Dimethylamino-ethyl)-methyl-amino]-qu...)
Affinity DataIC50: 804nMAssay Description:Displacement of 150p M [125I]MCH from human MCH1R expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed