BDBM50182739 CHEMBL3819427

SMILES NC(=O)c1ccc(cc1)C(=O)CCCN1CCc2ccccc2C1

InChI Key InChIKey=HNPAUMYBQXZAJH-UHFFFAOYSA-N

Data  16 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 16 hits for monomerid = 50182739   

Target5-hydroxytryptamine receptor 7(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50182739(CHEMBL3819427)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]LSD from human 5-HT7 receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50182739(CHEMBL3819427)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]N-methylspiperone from human D3 receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50182739(CHEMBL3819427)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]N-methylspiperone from human D3 receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50182739(CHEMBL3819427)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2017
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50182739(CHEMBL3819427)
Affinity DataKi:  204nMAssay Description:Displacement of [3H]N-methylspiperone from rat D4 receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2017
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50182739(CHEMBL3819427)
Affinity DataKi:  205nMAssay Description:Displacement of [3H]N-methylspiperone from rat D4 receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2017
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50182739(CHEMBL3819427)
Affinity DataKi:  218nMAssay Description:Displacement of [3H]N-methylspiperone from human D2 receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2017
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50182739(CHEMBL3819427)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]N-methylspiperone from human D2 receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50182739(CHEMBL3819427)
Affinity DataKi:  404nMAssay Description:Displacement of [3H]Ketanserin from human 5-HT2A receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50182739(CHEMBL3819427)
Affinity DataKi:  407nMAssay Description:Displacement of [3H]Ketanserin from human 5-HT2A receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50182739(CHEMBL3819427)
Affinity DataKi:  587nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50182739(CHEMBL3819427)
Affinity DataKi:  589nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2017
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50182739(CHEMBL3819427)
Affinity DataKi:  1.42E+3nMAssay Description:Displacement of [3H]Pyrilamine from human H1 receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2017
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50182739(CHEMBL3819427)
Affinity DataKi:  1.43E+3nMAssay Description:Displacement of [3H]Pyrilamine from human H1 receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50182739(CHEMBL3819427)
Affinity DataKi:  1.89E+3nMAssay Description:Displacement of [3H]Mesulergine from rat 5-HT2C receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50182739(CHEMBL3819427)
Affinity DataKi:  1.91E+3nMAssay Description:Displacement of [3H]Mesulergine from rat 5-HT2C receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2017
Entry Details Article
PubMed