BDBM50189844 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-5-(pyrazol-1-yl)imidazo[1,2-a]pyridine::CHEMBL212160

SMILES COc1ccccc1N1CCN(Cc2cn3c(cccc3n2)-n2cccn2)CC1

InChI Key InChIKey=BZHJMSJFFNOURP-UHFFFAOYSA-N

Data  5 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50189844   

TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189844(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-5-(pyr...)
Affinity DataKi:  0.940nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189844(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-5-(pyr...)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(short) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189844(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-5-(pyr...)
Affinity DataKi:  590nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(long) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189844(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-5-(pyr...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D3 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Pig)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189844(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-5-(pyr...)
Affinity DataKi:  2.70E+4nMAssay Description:Displacement of [3H]SCH 23990 from dopamine receptor D1 in porcine striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed