BDBM50200264 (4-bromo-2-{[(5-phenyl-1,2,4-triazin-3-yl)hydrazono]methyl}phenoxy)acetic acid::CHEMBL216189

SMILES OC(=O)COc1ccc(Br)cc1CN=Nc1nncc(n1)-c1ccccc1

InChI Key InChIKey=JFJFFXZVMBZBDI-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50200264   

TargetProstaglandin D2 receptor 2(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50200264((4-bromo-2-{[(5-phenyl-1,2,4-triazin-3-yl)hydrazon...)
Affinity DataIC50: 89nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50200264((4-bromo-2-{[(5-phenyl-1,2,4-triazin-3-yl)hydrazon...)
Affinity DataIC50: 3.21E+3nMAssay Description:Antagonist activity against CRTH2 receptor measured as inhibition of PGD2-induced beta-arrestin translocation in HEK293 cells by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed