BDBM50231102 CHEMBL254671::N-(2-(1H-indol-3-yl)ethyl)-4-(trifluoromethoxy)benzamide

SMILES FC(F)(F)Oc1ccc(cc1)C(=O)NCCc1c[nH]c2ccccc12

InChI Key InChIKey=AYBQHQMSAIQAFG-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50231102   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50231102(N-(2-(1H-indol-3-yl)ethyl)-4-(trifluoromethoxy)ben...)Copy SMILESCopy InChI

Affinity DataIC50: 7.35E+3nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced calcium influx in HEK293 cellsMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL