BDBM50254922 CHEMBL481984::N-(4,5-dichlorothiophen-2-ylsulfonyl)-2-(3-(1-methyl-1H-tetrazol-5-ylthio)-1H-indol-4-yloxy)acetamide

SMILES Cn1nnnc1Sc1c[nH]c2cccc(OCC(=O)NS(=O)(=O)c3cc(Cl)c(Cl)s3)c12

InChI Key InChIKey=BUSNTZZXCDQEGI-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50254922   

TargetProstaglandin E2 receptor EP3 subtype(Human)
Decode Chemistry

Curated by ChEMBL
LigandPNGBDBM50254922(N-(4,5-dichlorothiophen-2-ylsulfonyl)-2-(3-(1-meth...)
Affinity DataIC50: 8.20nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Decode Chemistry

Curated by ChEMBL
LigandPNGBDBM50254922(N-(4,5-dichlorothiophen-2-ylsulfonyl)-2-(3-(1-meth...)
Affinity DataIC50: 58.3nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor in presence of 10% human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed