BDBM50293495 3-(3-((N-(4-tert-butylbenzyl)thiazole-2-sulfonamido)methyl)phenyl)propanoic acid::CHEMBL541517

SMILES CC(C)(C)c1ccc(CN(Cc2cccc(CCC(O)=O)c2)S(=O)(=O)c2nccs2)cc1

InChI Key InChIKey=WVDZQCYXZZHZIL-UHFFFAOYSA-N

Data  2 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50293495   

LigandPNGBDBM50293495(3-(3-((N-(4-tert-butylbenzyl)thiazole-2-sulfonamid...)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity against rat EP2 receptor expressed in HEK293 cells assessed as stimulation of cAMP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293495(3-(3-((N-(4-tert-butylbenzyl)thiazole-2-sulfonamid...)
Affinity DataIC50: 63nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
LigandPNGBDBM50293495(3-(3-((N-(4-tert-butylbenzyl)thiazole-2-sulfonamid...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed