BDBM50360140 CHEMBL1929362

SMILES CC(C)CN1CC[C@]23Cc4nc5ccccc5cc4C[C@H]2[C@H]1Cc1cccc(O)c31

InChI Key

Data  3 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50360140   

TargetDelta-type opioid receptor(Rat)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360140(CHEMBL1929362)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat cerebrum membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360140(CHEMBL1929362)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at human recombinant delta opioid receptor expressed in human HEK293 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360140(CHEMBL1929362)
Affinity DataKi:  323nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat cerebrum membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360140(CHEMBL1929362)
Affinity DataKi:  516nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in guinea pig cerebrum membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed