BDBM50439463 CHEMBL2420911

SMILES C1CNCC2(C1)CCN(CC2)c1ncnc2nc[nH]c12

InChI Key InChIKey=ZXMGQAIKNOIWHC-UHFFFAOYSA-N

Data  12 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 12 hits for monomerid = 50439463   

TargetRibosomal protein S6 kinase alpha-5(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50439463(CHEMBL2420911)
Affinity DataIC50: 700nMAssay Description:Inhibition of MSK1 (unknown origin) by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50439463(CHEMBL2420911)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of PKD2 (unknown origin) by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50439463(CHEMBL2420911)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of AKT1 (unknown origin) by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50439463(CHEMBL2420911)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of CHK1 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50439463(CHEMBL2420911)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of ABL (unknown origin) by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAurora kinase A(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50439463(CHEMBL2420911)
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of AURA (unknown origin) by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk2(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50439463(CHEMBL2420911)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of CHK2 (unknown origin) by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetRibosomal protein S6 kinase alpha-1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50439463(CHEMBL2420911)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of RSK1 (unknown origin) by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50439463(CHEMBL2420911)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of ERK2 (unknown origin) by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 5(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50439463(CHEMBL2420911)
Affinity DataIC50: 4.10E+4nMAssay Description:Inhibition of PRAK (unknown origin) by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50439463(CHEMBL2420911)
Affinity DataIC50: 9.70E+4nMAssay Description:Inhibition of CK1delta (unknown origin) by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50439463(CHEMBL2420911)
Affinity DataIC50: 1.83E+5nMAssay Description:Inhibition of MET (unknown origin) by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed