BDBM9153 US8829010, 58::US8829010, 59

SMILES CNc1ncnc2n(C)nc(-c3cnn(C)c3-c3ccc(cc3)C(F)(F)F)c12

InChI Key InChIKey=RCPKOFJPUJIKJL-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 9153   

LigandPNGBDBM9153(US8829010, 59 | US8829010, 58)
Affinity DataIC50: 13.7nMAssay Description:In the present assay, the activity of the test substances on human full-length PDE2A3 enzyme was determined using the [3H]-cGMP scintillation proximi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2015
Entry Details
US Patent

LigandPNGBDBM9153(US8829010, 59 | US8829010, 58)
Affinity DataIC50: 27nMAssay Description:In the present assay, the activity of the test substances on human full-length PDE2A3 enzyme was determined using the [3H]-cGMP scintillation proximi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2015
Entry Details
US Patent