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BDBM100652 US8507676, 1

SMILES: CCO\N=C(/C)c1ccc2ncc(Cc3cc4cccnc4cc3F)n2n1

InChI Key: InChIKey=SQUIMUNWIZKHQI-DHRITJCHSA-N

Data: 1 IC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 100652   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM100652
PNG
(US8507676, 1)
Show SMILES CCO\N=C(/C)c1ccc2ncc(Cc3cc4cccnc4cc3F)n2n1
Show InChI InChI=1S/C20H18FN5O/c1-3-27-25-13(2)18-6-7-20-23-12-16(26(20)24-18)10-15-9-14-5-4-8-22-19(14)11-17(15)21/h4-9,11-12H,3,10H2,1-2H3/b25-13+
PDB
MMDB

KEGG

UniProtKB/SwissProt
UniProtKB/TrEMBL

B.MOAD
DrugBank
GoogleScholar
PC cid
PC sid
UniChem

Similars

US Patent
n/an/a 36n/an/an/an/an/an/a



Novartis AG

US Patent


Assay Description
The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...


US Patent US8507676 (2013)


BindingDB Entry DOI: 10.7270/Q2MS3RC9
More data for this
Ligand-Target Pair