BDBM100954 US10189794, Compound I-241::US10618902, Compound I-241::US10774052, Compound I-241::US9695132, I-241

SMILES: CN1c2c(cnc(n2)N[C@@H]3COC[C@@H]3NC(=O)C=C)C=C(C1=O)c4c(c(cc(c4Cl)OC)OC)Cl

InChI Key: InChIKey=ZIJVLVUPDVUSMA-UHFFFAOYSA-N

Data: 8 IC50

PDB links: 1 PDB ID matches this monomer.

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 100954   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Fibroblast growth factor receptor 4 (Human)	BDBM100954 (US9695132, I-241 | US10189794, Compound I-241 | US...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	<100	n/a	n/a	n/a	n/a	7.5	n/a
TBA									Citation and Details
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Fibroblast growth factor receptor 4 (Human)	BDBM100954 (US9695132, I-241 | US10189794, Compound I-241 | US...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	<100	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 4 (Human)	BDBM100954 (US9695132, I-241 | US10189794, Compound I-241 | US...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	<500	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 4 (Human)	BDBM100954 (US9695132, I-241 | US10189794, Compound I-241 | US...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	<100	n/a	n/a	n/a	n/a	n/a	n/a
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Fibroblast growth factor receptor 2 (Human)	BDBM100954 (US9695132, I-241 | US10189794, Compound I-241 | US...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	505	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 4 (Human)	BDBM100954 (US9695132, I-241 | US10189794, Compound I-241 | US...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	6.5	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 4 (Human)	BDBM100954 (US9695132, I-241 | US10189794, Compound I-241 | US...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	8.80	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 2 (Human)	BDBM100954 (US9695132, I-241 | US10189794, Compound I-241 | US...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	842	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair