BDBM11454 5-N-(4-aminocyclohexyl)-7-N-(4-methanesulfonylphenyl)-[1,2,4]triazolo[1,5-a]pyrimidine-5,7-diamine::triazolo[1,5-a]pyrimidine 16
SMILES CS(=O)(=O)c1ccc(Nc2cc(N[C@H]3CC[C@H](N)CC3)nc3ncnn23)cc1
InChI Key InChIKey=UDVYMPJUORTTMR-JOCQHMNTSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 11454
Affinity DataIC50: 250nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified CDK enzyme was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [...More data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+4nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified GSK-3 beta was incubated at room temperature with substrate, and test compounds in the presence of 10 uM ATP/ [g...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+4nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified CDK enzyme was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [...More data for this Ligand-Target Pair