BDBM120221 US8691753, 70
SMILES OC(=O)CC[C@H](NC(=O)CCc1ccc(cc1)-c1ccc(cc1)-c1ccccc1)C(=O)N1CCCC(CC(O)=O)C1
InChI Key InChIKey=WLZQVNRDQZYTID-PEFOLFAWSA-N
Data 8 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 120221
TargetMacrophage metalloelastase(Homo sapiens (Human))
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Affinity DataKi: 4.70nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Affinity DataKi: 12nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
TargetCollagenase 3(Homo sapiens (Human))
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Affinity DataKi: 17nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
TargetNeutrophil collagenase(Homo sapiens (Human))
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Affinity DataKi: 105nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
TargetStromelysin-1(Homo sapiens (Human))
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Affinity DataKi: 231nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
TargetStromelysin-2(Homo sapiens (Human))
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Affinity DataKi: 421nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-14 [1-20,P8S](Homo sapiens (Human))
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Affinity DataKi: >1.00E+3nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Affinity DataKi: >5.00E+3nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair