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BDBM127657 US10251889, Example 30::US8791123, 30::US9782415, Example 30::US9796724, Example 30

SMILES: NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F

InChI Key: InChIKey=JBTQGTQNCVBRNY-YQTOOIBONA-N

Data: 25 IC50

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 25 hits for monomerid = 127657   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
High affinity nerve growth factor receptor


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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US Patent
n/an/a 1.95n/an/an/an/a7.5n/a



Array Biopharma, Inc.

US Patent


Assay Description
An enzyme-linked immunosorbant assay (ELISA) was used to assess TrkA kinase activity in the presence of inhibitors. Immulon 4HBX 384-well microtiter ...


US Patent US8791123 (2014)


BindingDB Entry DOI: 10.7270/Q2Q23XX7
More data for this
Ligand-Target Pair
Non-receptor tyrosine-protein kinase TYK2


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array BioPharma, Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Tyk2 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US9796724 (2017)


Article DOI: 10.1021/jm0701019
BindingDB Entry DOI: 10.7270/Q27M0B21
More data for this
Ligand-Target Pair
Tyrosine-protein kinase JAK1


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array Biopharma, Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Jak1 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US8791123 (2014)


BindingDB Entry DOI: 10.7270/Q2Q23XX7
More data for this
Ligand-Target Pair
Tyrosine-protein kinase JAK3


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array Biopharma, Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Jak3 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US8791123 (2014)


BindingDB Entry DOI: 10.7270/Q2Q23XX7
More data for this
Ligand-Target Pair
Non-receptor tyrosine-protein kinase TYK2


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array Biopharma, Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Tyk2 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US8791123 (2014)


BindingDB Entry DOI: 10.7270/Q2Q23XX7
More data for this
Ligand-Target Pair
High affinity nerve growth factor receptor


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a 1.95n/an/an/an/an/an/a



Array BioPharma, Inc.

US Patent


Assay Description
An enzyme-linked immunosorbant assay (ELISA) was used to assess TrkA kinase activity in the presence of inhibitors. Immulon 4HBX 384-well microtiter ...


US Patent US9782415 (2017)


Article DOI: 10.1021/jm030131l
BindingDB Entry DOI: 10.7270/Q2P84F0G
More data for this
Ligand-Target Pair
Tyrosine-protein kinase JAK2


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array BioPharma, Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Jak2 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US9782415 (2017)


Article DOI: 10.1021/jm030131l
BindingDB Entry DOI: 10.7270/Q2P84F0G
More data for this
Ligand-Target Pair
High affinity nerve growth factor receptor


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a 1.90n/an/an/an/an/an/a



Array BioPharma, Inc.

US Patent


Assay Description
An enzyme-linked immunosorbant assay (ELISA) was used to assess TrkA kinase activity in the presence of inhibitors. Immulon 4HBX 384-well microtiter ...


US Patent US9782415 (2017)


Article DOI: 10.1021/jm030131l
BindingDB Entry DOI: 10.7270/Q2P84F0G
More data for this
Ligand-Target Pair
Tyrosine-protein kinase JAK1


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array BioPharma, Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Jak1 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US9782415 (2017)


Article DOI: 10.1021/jm030131l
BindingDB Entry DOI: 10.7270/Q2P84F0G
More data for this
Ligand-Target Pair
Tyrosine-protein kinase JAK2


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array BioPharma, Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Jak2 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US9782415 (2017)


Article DOI: 10.1021/jm030131l
BindingDB Entry DOI: 10.7270/Q2P84F0G
More data for this
Ligand-Target Pair
Tyrosine-protein kinase JAK3


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array BioPharma, Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Jak3 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US9782415 (2017)


Article DOI: 10.1021/jm030131l
BindingDB Entry DOI: 10.7270/Q2P84F0G
More data for this
Ligand-Target Pair
Tyk2


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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US Patent
n/an/a>1.00E+3n/an/an/an/an/an/a



Array BioPharma, Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Tyk2 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US9782415 (2017)


Article DOI: 10.1021/jm030131l
BindingDB Entry DOI: 10.7270/Q2P84F0G
More data for this
Ligand-Target Pair
Tyrosine-protein kinase JAK2


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a 1.95n/an/an/an/an/an/a



Array BioPharm Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Jak2 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US10251889 (2019)

More data for this
Ligand-Target Pair
High affinity nerve growth factor receptor


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array BioPharm Inc.

US Patent


Assay Description
An enzyme-linked immunosorbant assay (ELISA) was used to assess TrkA kinase activity in the presence of inhibitors. Immulon 4HBX 384-well microtiter ...


US Patent US10251889 (2019)

More data for this
Ligand-Target Pair
High affinity nerve growth factor receptor


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a 1.90n/an/an/an/an/an/a



Array BioPharm Inc.

US Patent


Assay Description
Trk enzymatic selectivity was assessed using Omnia™ Kinase Assay reagents from Invitrogen Corp. Enzyme (either TrkA or TrkB from Invitrogen Corp.) an...


US Patent US10251889 (2019)

More data for this
Ligand-Target Pair
Tyrosine-protein kinase JAK1


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array BioPharm Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Jak1 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US10251889 (2019)

More data for this
Ligand-Target Pair
Tyrosine-protein kinase JAK2


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array BioPharm Inc.

US Patent




US Patent US10251889 (2019)

More data for this
Ligand-Target Pair
Tyrosine-protein kinase JAK3


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array BioPharm Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Jak3 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US10251889 (2019)

More data for this
Ligand-Target Pair
Non-receptor tyrosine-protein kinase TYK2


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array BioPharm Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Tyk2 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US10251889 (2019)

More data for this
Ligand-Target Pair
High affinity nerve growth factor receptor


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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Article
US Patent
n/an/a 1.95n/an/an/an/an/an/a



Array BioPharma, Inc.

US Patent


Assay Description
Trk enzymatic selectivity was assessed using Omnia™ Kinase Assay reagents from Invitrogen Corp. Enzyme (either TrkA or TrkB from Invitrogen Corp.) an...


US Patent US9796724 (2017)


Article DOI: 10.1021/jm0701019
BindingDB Entry DOI: 10.7270/Q27M0B21
More data for this
Ligand-Target Pair
JAK2 (aa 808-1132)


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array BioPharma, Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Jak2 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US9796724 (2017)


Article DOI: 10.1021/jm0701019
BindingDB Entry DOI: 10.7270/Q27M0B21
More data for this
Ligand-Target Pair
JAK1 (aa 866-1154)


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array BioPharma, Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Jak1 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US9796724 (2017)


Article DOI: 10.1021/jm0701019
BindingDB Entry DOI: 10.7270/Q27M0B21
More data for this
Ligand-Target Pair
JAK2 (aa 808-1132)


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array BioPharma, Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Jak2 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US9796724 (2017)


Article DOI: 10.1021/jm0701019
BindingDB Entry DOI: 10.7270/Q27M0B21
More data for this
Ligand-Target Pair
JAK3 (aa 781-1124)


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array BioPharma, Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Jak3 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US9796724 (2017)


Article DOI: 10.1021/jm0701019
BindingDB Entry DOI: 10.7270/Q27M0B21
More data for this
Ligand-Target Pair
Tyrosine-protein kinase JAK2


(Homo sapiens (Human))
BDBM127657
PNG
(US10251889, Example 30 | US8791123, 30 | US9782415...)
Show SMILES NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Show InChI InChI=1/C17H15F2N5O/c18-10-3-4-13(19)11(8-10)14-2-1-6-23(14)15-5-7-24-17(22-15)12(9-21-24)16(20)25/h3-5,7-9,14H,1-2,6H2,(H2,20,25)/t14-/s2
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n/an/a>1.00E+3n/an/an/an/an/an/a



Array Biopharma, Inc.

US Patent


Assay Description
Compounds of Formula I were screened for their ability to inhibit Jak2 using the general enzyme inhibition assay method, in which the assay mixture c...


US Patent US8791123 (2014)


BindingDB Entry DOI: 10.7270/Q2Q23XX7
More data for this
Ligand-Target Pair