BDBM129369 US8802673, 11
SMILES FC(F)(F)c1ccc(Nc2ccc(cc2)C2CNCCO2)nc1
InChI Key InChIKey=ICJRJBTWDCPIOM-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 129369
Affinity DataKi: 1.5nM ΔG°: -12.5kcal/molepH: 7.4 T: 2°CAssay Description:HEK-293 cells stably expressing rat TAAR1 were maintained at 37 C. and 5% CO2 in DMEM high glucose medium, containing fetal calf serum (10%, heat ina...More data for this Ligand-Target Pair
Affinity DataKi: 23.3nM ΔG°: -10.8kcal/molepH: 7.4 T: 2°CAssay Description:HEK-293 cells stably expressing mouse TAAR1 were maintained at 37 C. and 5% CO2 in DMEM high glucose medium, containing fetal calf serum (10%, heat i...More data for this Ligand-Target Pair