BDBM141889 US8921410, Table 2 Compound 27

SMILES O=C(N1CC2CNCC(C2)C1)c1cnco1

InChI Key InChIKey=HVYPEWIFRMKLAK-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 141889   

TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Targacept

US Patent
LigandPNGBDBM141889(US8921410, Table 2 Compound 27)
Affinity DataKi:  26nM ΔG°:  -10.2kcal/moleT: 2°CAssay Description:The binding of [3H]MLA was measured using a modification of the methods of Davies et al., Neuropharmacol. 38: 679 (1999). [3H]MLA (Specific Activity=...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Targacept

US Patent
LigandPNGBDBM141889(US8921410, Table 2 Compound 27)
Affinity DataKi:  28nM ΔG°:  -10.2kcal/moleT: 2°CAssay Description:The binding of [3H]MLA was measured using a modification of the methods of Davies et al., Neuropharmacol. 38: 679 (1999). [3H]MLA (Specific Activity=...More data for this Ligand-Target Pair
In DepthDetails US Patent