BDBM143710 US9682960, EM-9156::US9682960, EM-9288

SMILES CC1(C)N(CCCOc2ccc(cc2Cl)-c2cc[n+]([O-])cc2)C(=O)N(C1=O)c1ccc(C#N)c(Cl)c1

InChI Key InChIKey=UXZWTRYTKPERAO-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 143710   

TargetAndrogen receptor(Mus musculus)
Endorecherche

US Patent
LigandPNGBDBM143710(US9682960, EM-9156 | US9682960, EM-9288)
Affinity DataIC50:  14nMpH: 7.4 T: 2°CAssay Description:Androgen binding is measured using the hydroxylapatite (HAP) assay. In brief, the radioactive steroid [3H]R1881 solubilized in ethanol is diluted wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Mus musculus)
Endorecherche

US Patent
LigandPNGBDBM143710(US9682960, EM-9156 | US9682960, EM-9288)
Affinity DataIC50:  9.20nMpH: 7.4 T: 2°CAssay Description:Androgen binding is measured using the hydroxylapatite (HAP) assay. In brief, the radioactive steroid [3H]R1881 solubilized in ethanol is diluted wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Mus musculus)
Endorecherche

US Patent
LigandPNGBDBM143710(US9682960, EM-9156 | US9682960, EM-9288)
Affinity DataIC50:  15nMpH: 7.4 T: 2°CAssay Description:Androgen binding is measured using the hydroxylapatite (HAP) assay. In brief, the radioactive steroid [3H]R1881 solubilized in ethanol is diluted wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Mus musculus)
Endorecherche

US Patent
LigandPNGBDBM143710(US9682960, EM-9156 | US9682960, EM-9288)
Affinity DataIC50:  15nMpH: 7.4 T: 2°CAssay Description:Androgen binding is measured using the hydroxylapatite (HAP) assay. In brief, the radioactive steroid [3H]R1881 solubilized in ethanol is diluted wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent