BindingDB logo
myBDB logout

BDBM153951 US8999981, F7

SMILES: COCCCN1C[C@H](C)N(C[C@H]1C)C(=O)N1Cc2c(NC(=O)Cc3c(C)noc3C)n[nH]c2C1(C)C

InChI Key:

Data: 1 KI

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 153951   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
PKC alpha and beta-2


(Homo sapiens (Human))
BDBM153951
PNG
(US8999981, F7)
Show SMILES COCCCN1C[C@H](C)N(C[C@H]1C)C(=O)N1Cc2c(NC(=O)Cc3c(C)noc3C)n[nH]c2C1(C)C
PDB
MMDB

NCI pathway
Reactome pathway
KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
antibodypedia
GoogleScholar
PC cid
PC sid
UniChem

Similars

US Patent
67.1 -9.94n/an/an/an/an/a7.430



Pfizer Inc

US Patent


Assay Description
Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...


US Patent US8999981 (2015)


BindingDB Entry DOI: 10.7270/Q2RR1X0K
More data for this
Ligand-Target Pair