BDBM154188 US9012443, 197

SMILES COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncc(s1)C#N)C(F)(F)F

InChI Key InChIKey=PZJXPTLCGPWBHN-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 154188   

LigandPNGBDBM154188(US9012443, 197)
Affinity DataIC50: 2.93E+3nMAssay Description:293 Cells stably transfected with either Nav 1.7 or Nav 1.5 were recorded in population patch-clamp mode with the IonWorks Quattro automated electrop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2015
Entry Details
US Patent

LigandPNGBDBM154188(US9012443, 197)
Affinity DataIC50: 3.06E+3nMAssay Description:293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology system...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2015
Entry Details
US Patent