BDBM154478 US9012443, 231

SMILES COc1cnc(-c2ccc(cc2O)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1nccs1

InChI Key InChIKey=VPKDTLALYQWDMG-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 154478   

LigandPNGBDBM154478(US9012443, 231)
Affinity DataIC50: 40nMAssay Description:293 Cells stably transfected with either Nav 1.7 or Nav 1.5 were recorded in population patch-clamp mode with the IonWorks Quattro automated electrop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2015
Entry Details
US Patent

LigandPNGBDBM154478(US9012443, 231)
Affinity DataIC50: 270nMAssay Description:293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology system...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2015
Entry Details
US Patent