BDBM158290 US9029370, 84
SMILES CCOc1cc(ccn1)C(=O)Nc1ccc([C@@H]2CNCCO2)c(F)c1
InChI Key InChIKey=AOTQIDPOBHBGSP-INIZCTEOSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 158290
Affinity DataKi: 3.60nM ΔG°: -12.0kcal/molepH: 7.4 T: 2°CAssay Description:Membrane Preparation and Radioligand Binding. HEK-293 cells stably expressing mouse TAA 1 were maintained at 37 C and 5% C02 in DMEM high glucose med...More data for this Ligand-Target Pair
Affinity DataKi: 4.70nM ΔG°: -11.8kcal/molepH: 7.4 T: 2°CAssay Description:HEK-293 cells stably expressing rat TAAR1 were maintained at 37 C and 5% CO2 in DMEM high glucose medium, containing fetal calf serum (10%, heat inac...More data for this Ligand-Target Pair