BDBM158304 US9029370, 98
SMILES Clc1cc(ccc1NC(=O)c1cccc(n1)C#N)[C@H]1CNCCO1
InChI Key InChIKey=BMWYGXDSJAMYPG-MRXNPFEDSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 158304
Affinity DataKi: 27.6nM ΔG°: -10.7kcal/molepH: 7.4 T: 2°CAssay Description:Membrane Preparation and Radioligand Binding. HEK-293 cells stably expressing mouse TAA 1 were maintained at 37 C and 5% C02 in DMEM high glucose med...More data for this Ligand-Target Pair
Affinity DataKi: 565nM ΔG°: -8.86kcal/molepH: 7.4 T: 2°CAssay Description:HEK-293 cells stably expressing rat TAAR1 were maintained at 37 C and 5% CO2 in DMEM high glucose medium, containing fetal calf serum (10%, heat inac...More data for this Ligand-Target Pair