BDBM162310 US10307427, Compound 1::US9051313, 1
SMILES O=C(Nc1csc(n1)-c1nncn1C1CC1)c1cc(c(cn1)N1CCOCC1)-n1cnc(c1)C1CC1
InChI Key InChIKey=HIQBMNWLSRWMLZ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 162310
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Gildead Sciences
US Patent
Gildead Sciences
US Patent
Affinity DataIC50: 1.44nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection (6.1). This is a competitive...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Gildead Sciences
US Patent
Gildead Sciences
US Patent
Affinity DataEC50: 13.2nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection (6.1). This is a competitive...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Gildead Sciences
US Patent
Gildead Sciences
US Patent
Affinity DataIC50: 1.44nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection (6.1). This is a competitive...More data for this Ligand-Target Pair