BDBM162314 US9051313, 5

SMILES C[C@H](n1cnnc1-c1nc(NC(=O)c2cc(c(cn2)N(C)C)-n2cnc(c2)C2CC2)cs1)C(F)(F)F

InChI Key InChIKey=RLSCTEQIUJARIV-LBPRGKRZSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 162314   

TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Gildead Sciences

US Patent
LigandPNGBDBM162314(US9051313, 5)
Affinity DataIC50:  1.88nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection (6.1). This is a competitive...More data for this Ligand-Target Pair
In DepthDetails US Patent