BDBM162317 US9051313, 8
SMILES C[C@H](n1cnnc1-c1nc(NC(=O)c2cc(c(cn2)N2CCCC2)-n2cnc(c2)C2CC2)cs1)C(F)(F)F
InChI Key InChIKey=ITXKFABJUPGBQB-AWEZNQCLSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 162317
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Gildead Sciences
US Patent
Gildead Sciences
US Patent
Affinity DataIC50: 2.20nMAssay Description:The assay measures the phosphorylation level of a biotinylated peptide substrate by the ASK1 kinase using HTRF detection (6.1). This is a competitive...More data for this Ligand-Target Pair