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BDBM17716 2,3-Diarylfuro[2,3-b]pyridine-4-amine, 8::2,3-diphenyl-N-[2-(piperazin-1-yl)ethyl]furo[2,3-b]pyridin-4-amine

SMILES: C(CN1CCNCC1)Nc1ccnc2oc(c(-c3ccccc3)c12)-c1ccccc1

InChI Key: InChIKey=QUIQCYFSBGOBKE-UHFFFAOYSA-N

Data: 4 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 17716
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Vascular endothelial growth factor receptor 2 (Human)	BDBM17716 (2,3-diphenyl-N-[2-(piperazin-1-yl)ethyl]furo[2,3-b...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	360	n/a	n/a	n/a	n/a	7.5	22
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Tyrosine-protein kinase Lck (Human)	BDBM17716 (2,3-diphenyl-N-[2-(piperazin-1-yl)ethyl]furo[2,3-b...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	210	n/a	n/a	n/a	n/a	7.5	22
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Activated CDC42 kinase 1 (Human)	BDBM17716 (2,3-diphenyl-N-[2-(piperazin-1-yl)ethyl]furo[2,3-b...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	420	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Human)	BDBM17716 (2,3-diphenyl-N-[2-(piperazin-1-yl)ethyl]furo[2,3-b...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	140	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair