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BDBM178166 US10307413, Compound 208::US10391089, Compound 208::US10980794, Cmpd No 208::US11591326, Compound C3::US9675614, 208

SMILES: CC(=O)N1CCC(CC1)Nc2cc(ncn2)C(=O)NC[C@@H](CN3CCc4ccccc4C3)O

InChI Key: InChIKey=JLCCNYVTIWRPIZ-UHFFFAOYSA-N

Data: 9 IC50

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 41 hits for monomerid = 178166   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/an/an/a 2n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/an/an/a 2.5n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/an/an/a 2n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/an/an/a 2n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/an/an/a 2n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/an/an/a 2n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/an/an/a 2n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/an/an/a 2n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/an/an/a 2n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/a<100n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/an/an/a 22n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/an/an/a 50n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/an/an/a 55n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/an/an/a 167n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/an/an/a 177n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/an/an/a 212n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/an/an/a 214n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/an/an/a 323n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Mouse)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/a 6.20n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/a<100n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Methylosome protein 50/Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/a<100n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/a<100n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Methylosome protein 50/Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/a 38n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/a 47n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/a 6.20n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Methylosome protein 50/Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/a 6.20n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/a 11n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Human)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/a 12n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Mouse)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/a 19n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Mouse)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/a 6.20n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Mouse)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/a 6n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Mouse)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/a 5.90n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Mouse)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
n/an/a 20n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Mouse)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
3n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Mouse)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
3n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Mouse)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
3.10n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Mouse)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
3.10n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Mouse)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
9.5n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Mouse)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
9.90n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Mouse)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
26n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Mouse)
BDBM178166
PNG
(US9675614, 208 | US10307413, Compound 208 | US1039...)
GoogleScholar
UniChem
43n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair