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BDBM178570 US9125913, 129

SMILES: CN(C)CCOc1cccc(c1CN1CCN(CC1)c1ccc(C(=O)NS(=O)(=O)c2ccc(NCC3CCOCC3)c(c2)[N+]([O-])=O)c(Oc2ccc3[nH]ccc3c2)c1)-c1ccc(Cl)cc1

InChI Key: InChIKey=OEPSXIVYHBPSCA-UHFFFAOYSA-N

Data: 5 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 178570
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Apoptosis regulator Bcl-2 (Mouse)	BDBM178570 (US9125913, 129) Show SMILES Show InChI	GoogleScholar	UniChem		0.0560	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Apoptosis regulator Bcl-2 (Human)	BDBM178570 (US9125913, 129) Show SMILES Show InChI	GoogleScholar	UniChem		<0.100	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Apoptosis regulator Bcl-2 (Human)	BDBM178570 (US9125913, 129) Show SMILES Show InChI	GoogleScholar	UniChem		<0.100	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Bcl-2-like protein 1 (Mouse)	BDBM178570 (US9125913, 129) Show SMILES Show InChI	GoogleScholar	UniChem		>660	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Bcl-2-like protein 1 (Human)	BDBM178570 (US9125913, 129) Show SMILES Show InChI	GoogleScholar	UniChem		>660	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair