BDBM179481 US9675697, Cpd. No. 73

SMILES: COc1cc2c(cc1-c1c(C)noc1C)[nH]c1nc(C)nc(-c3ccnc4ccccc34)c21

InChI Key: InChIKey=AEANZCXROGPSBY-UHFFFAOYSA-N

Data: 9 KI  4 IC50  36 Kd

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 49 hits for monomerid = 179481   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Bromodomain-containing protein 9 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Bromodomain and PHD finger-containing protein 3 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
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Nucleosome-remodeling factor subunit BPTF (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
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Protein polybromo-1 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
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Histone acetyltransferase KAT2B (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
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Probable global transcription activator SNF2L2 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
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Transcription initiation factor TFIID subunit 1 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
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Transcription intermediary factor 1-alpha (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
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Serine/threonine-protein kinase PLK4 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3.90E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 2 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	4.5	n/a	n/a	n/a	n/a	n/a
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Bromodomain adjacent to zinc finger domain protein 2B (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 7 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 8 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
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Protein polybromo-1 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
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Transcription activator BRG1 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Bromodomain-containing protein 4 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	1.80	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	28	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	7.20	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 2 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	1.10	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	8.40	n/a	n/a	n/a	n/a	n/a
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CREB-binding protein (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	520	n/a	n/a	n/a	n/a	n/a
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ATPase family AAA domain-containing protein 2B (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Bromodomain-containing protein 1 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 8 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	28	n/a	n/a	n/a	n/a	n/a	n/a
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Peregrin (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Bromodomain and WD repeat-containing protein 1 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 3 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	0.730	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histone acetyltransferase KAT2A (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain adjacent to zinc finger domain protein 2A (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain testis-specific protein (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	5.5	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 2 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	0.900	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 3 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 3 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	0.690	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain testis-specific protein (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	15	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain testis-specific protein (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	9.70	n/a	n/a	n/a	n/a	n/a
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Chromatin remodeling regulator CECR2 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	1.60E+3	n/a	n/a	n/a	n/a	n/a
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Histone acetyltransferase p300 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
ATPase family AAA domain-containing protein 2 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>4.00E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		1.40	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 3 [326-398] (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		2.60	-11.7	n/a	n/a	n/a	n/a	n/a	n/a	25
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Bromodomain-containing protein 2 [364-436] (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		7.80	-11.1	n/a	n/a	n/a	n/a	n/a	n/a	25
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		8.20	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		8.20	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 2 [364-436] (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		8.70	-11.0	n/a	n/a	n/a	n/a	n/a	n/a	25
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Bromodomain-containing protein 3 [51-123] (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		10	-10.9	n/a	n/a	n/a	n/a	n/a	n/a	25
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Bromodomain-containing protein 2 [91-163] (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		16	-10.6	n/a	n/a	n/a	n/a	n/a	n/a	25
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Bromodomain-containing protein 4 [75-147] (Human)	BDBM179481 (US9675697, Cpd. No. 73) Show SMILES Show InChI	GoogleScholar	UniChem		35	-10.2	n/a	n/a	n/a	n/a	n/a	n/a	25
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